AR102995A1 - Uso de ligandos del receptor sigma en la osteoartritis - Google Patents

Uso de ligandos del receptor sigma en la osteoartritis

Info

Publication number
AR102995A1
AR102995A1 ARP150104064A ARP150104064A AR102995A1 AR 102995 A1 AR102995 A1 AR 102995A1 AR P150104064 A ARP150104064 A AR P150104064A AR P150104064 A ARP150104064 A AR P150104064A AR 102995 A1 AR102995 A1 AR 102995A1
Authority
AR
Argentina
Prior art keywords
osteoartritis
sigma receiver
ligands
sigma
receiver ligands
Prior art date
Application number
ARP150104064A
Other languages
English (en)
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Publication of AR102995A1 publication Critical patent/AR102995A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente se refiere a compuestos de fórmula (1) o fórmula (2) con actividad farmacológica contra el receptor sigma, para su uso en el tratamiento o la prevención de la osteoartritis y el dolor debido a la osteoartritis.
ARP150104064A 2014-12-15 2015-12-14 Uso de ligandos del receptor sigma en la osteoartritis AR102995A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP14382519 2014-12-15

Publications (1)

Publication Number Publication Date
AR102995A1 true AR102995A1 (es) 2017-04-05

Family

ID=52146389

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP150104064A AR102995A1 (es) 2014-12-15 2015-12-14 Uso de ligandos del receptor sigma en la osteoartritis

Country Status (1)

Country Link
AR (1) AR102995A1 (es)

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Legal Events

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