AR110356A1 - Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol - Google Patents

Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol

Info

Publication number
AR110356A1
AR110356A1 ARP170103481A ARP170103481A AR110356A1 AR 110356 A1 AR110356 A1 AR 110356A1 AR P170103481 A ARP170103481 A AR P170103481A AR P170103481 A ARP170103481 A AR P170103481A AR 110356 A1 AR110356 A1 AR 110356A1
Authority
AR
Argentina
Prior art keywords
formula
azetidin
fluoromethyl
tetrahydro
oxy
Prior art date
Application number
ARP170103481A
Other languages
English (en)
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR110356A1 publication Critical patent/AR110356A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
ARP170103481A 2016-12-12 2017-12-13 Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol AR110356A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662432837P 2016-12-12 2016-12-12

Publications (1)

Publication Number Publication Date
AR110356A1 true AR110356A1 (es) 2019-03-20

Family

ID=60935792

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170103481A AR110356A1 (es) 2016-12-12 2017-12-13 Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol

Country Status (2)

Country Link
AR (1) AR110356A1 (fr)
WO (1) WO2018108954A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI702219B (zh) 2018-07-12 2020-08-21 美商美國禮來大藥廠 選擇性雌激素受體降解劑
CN114933551B (zh) * 2022-06-28 2023-06-30 吉尔多肽生物制药(大连市)有限公司 一种手性Fmoc-3-氨基-2-(叔丁氧基甲基)丙酸的合成方法
CN117003681A (zh) * 2023-07-04 2023-11-07 苏州汉德创宏生化科技有限公司 一种抑制剂类中间体及其合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006033633A1 (fr) * 2004-09-24 2006-03-30 Astrazeneca Ab Composes, compositions contenant ces composes, preparation et utilisations de ces derniers
CN101198590B (zh) * 2005-08-24 2012-05-09 卫材R&D管理有限公司 吡啶衍生物及嘧啶衍生物(3)
WO2013090829A1 (fr) 2011-12-14 2013-06-20 Aragon Pharmaceuticals, Inc. Modulateurs des récepteurs des œstrogènes et ses utilisations
CA2915534A1 (fr) 2013-06-19 2014-12-24 Seragon Pharmaceuticals, Inc. Modulateurs azetidine des recepteurs d'oestrogenes et leurs utilisations
EA031077B1 (ru) 2013-06-19 2018-11-30 Серагон Фармасьютикалз, Инк. Модулятор рецептора эстрогена и его применения
TWI874834B (zh) 2014-12-18 2025-03-01 瑞士商赫孚孟拉羅股份公司 四氫-吡啶并[3,4-b]吲哚雌激素受體調節劑及其用途
US20160175284A1 (en) 2014-12-18 2016-06-23 Genentech, Inc. Estrogen receptor modulators and uses thereof
WO2016097071A1 (fr) 2014-12-18 2016-06-23 F. Hoffmann-La Roche Ag Modulateurs du récepteur des œstrogènes et leurs utilisations

Also Published As

Publication number Publication date
WO2018108954A1 (fr) 2018-06-21

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