AR110356A1 - Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol - Google Patents
Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-olInfo
- Publication number
- AR110356A1 AR110356A1 ARP170103481A ARP170103481A AR110356A1 AR 110356 A1 AR110356 A1 AR 110356A1 AR P170103481 A ARP170103481 A AR P170103481A AR P170103481 A ARP170103481 A AR P170103481A AR 110356 A1 AR110356 A1 AR 110356A1
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- azetidin
- fluoromethyl
- tetrahydro
- oxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662432837P | 2016-12-12 | 2016-12-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR110356A1 true AR110356A1 (es) | 2019-03-20 |
Family
ID=60935792
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP170103481A AR110356A1 (es) | 2016-12-12 | 2017-12-13 | Proceso para la preparación de 2-(3-(fluormetil)azetidin-1-il)etan-1-ol |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR110356A1 (fr) |
| WO (1) | WO2018108954A1 (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI702219B (zh) | 2018-07-12 | 2020-08-21 | 美商美國禮來大藥廠 | 選擇性雌激素受體降解劑 |
| CN114933551B (zh) * | 2022-06-28 | 2023-06-30 | 吉尔多肽生物制药(大连市)有限公司 | 一种手性Fmoc-3-氨基-2-(叔丁氧基甲基)丙酸的合成方法 |
| CN117003681A (zh) * | 2023-07-04 | 2023-11-07 | 苏州汉德创宏生化科技有限公司 | 一种抑制剂类中间体及其合成方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006033633A1 (fr) * | 2004-09-24 | 2006-03-30 | Astrazeneca Ab | Composes, compositions contenant ces composes, preparation et utilisations de ces derniers |
| CN101198590B (zh) * | 2005-08-24 | 2012-05-09 | 卫材R&D管理有限公司 | 吡啶衍生物及嘧啶衍生物(3) |
| WO2013090829A1 (fr) | 2011-12-14 | 2013-06-20 | Aragon Pharmaceuticals, Inc. | Modulateurs des récepteurs des œstrogènes et ses utilisations |
| CA2915534A1 (fr) | 2013-06-19 | 2014-12-24 | Seragon Pharmaceuticals, Inc. | Modulateurs azetidine des recepteurs d'oestrogenes et leurs utilisations |
| EA031077B1 (ru) | 2013-06-19 | 2018-11-30 | Серагон Фармасьютикалз, Инк. | Модулятор рецептора эстрогена и его применения |
| TWI874834B (zh) | 2014-12-18 | 2025-03-01 | 瑞士商赫孚孟拉羅股份公司 | 四氫-吡啶并[3,4-b]吲哚雌激素受體調節劑及其用途 |
| US20160175284A1 (en) | 2014-12-18 | 2016-06-23 | Genentech, Inc. | Estrogen receptor modulators and uses thereof |
| WO2016097071A1 (fr) | 2014-12-18 | 2016-06-23 | F. Hoffmann-La Roche Ag | Modulateurs du récepteur des œstrogènes et leurs utilisations |
-
2017
- 2017-12-12 WO PCT/EP2017/082493 patent/WO2018108954A1/fr not_active Ceased
- 2017-12-13 AR ARP170103481A patent/AR110356A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2018108954A1 (fr) | 2018-06-21 |
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| FB | Suspension of granting procedure |