AR110451A1 - Compuesto tricíclico que tiene sulfinilo y composición farmacéutica que lo comprende - Google Patents

Compuesto tricíclico que tiene sulfinilo y composición farmacéutica que lo comprende

Info

Publication number
AR110451A1
AR110451A1 ARP170103676A ARP170103676A AR110451A1 AR 110451 A1 AR110451 A1 AR 110451A1 AR P170103676 A ARP170103676 A AR P170103676A AR P170103676 A ARP170103676 A AR P170103676A AR 110451 A1 AR110451 A1 AR 110451A1
Authority
AR
Argentina
Prior art keywords
sulfinyl
pharmaceutical composition
tricyclic compound
compound
tricyclic
Prior art date
Application number
ARP170103676A
Other languages
English (en)
Inventor
Jun Sato
Katsuki Yokoo
Kenji Yamawaki
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of AR110451A1 publication Critical patent/AR110451A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

Reivindicación 1: Un compuesto caracterizado porque es cualquiera de la fórmula seleccionada del grupo de fórmulas (1); su forma de éster o una de sus sales o hidratos farmacéuticamente aceptables.
ARP170103676A 2016-12-26 2017-12-22 Compuesto tricíclico que tiene sulfinilo y composición farmacéutica que lo comprende AR110451A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2016251861 2016-12-26

Publications (1)

Publication Number Publication Date
AR110451A1 true AR110451A1 (es) 2019-03-27

Family

ID=62707667

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170103676A AR110451A1 (es) 2016-12-26 2017-12-22 Compuesto tricíclico que tiene sulfinilo y composición farmacéutica que lo comprende

Country Status (4)

Country Link
JP (1) JP2018104420A (es)
AR (1) AR110451A1 (es)
TW (1) TW201833119A (es)
WO (1) WO2018123920A1 (es)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02289584A (ja) * 1989-02-17 1990-11-29 Takeda Chem Ind Ltd セファロスポリンγ―ラクトン化合物
US6599893B2 (en) * 2000-08-29 2003-07-29 Essential Therapeutics, Inc. Cephalosporin antibiotics and prodrugs thereof
TW200305422A (en) * 2002-03-18 2003-11-01 Shionogi & Co Broad spectrum cefem compounds
EP2703406A4 (en) * 2011-04-28 2015-08-05 Shionogi & Co NOVEL CEPHEM COMPOUND HAVING THE CATÉCHOL STRUCTURE OR A STRUCTURE CLOSE TO CATÉCHOL
JPWO2016175223A1 (ja) * 2015-04-28 2018-02-15 塩野義製薬株式会社 三環性化合物、およびそれらの使用
US20180186814A1 (en) * 2015-06-30 2018-07-05 Shionogi & Co., Ltd. Tricyclic compound having sulfinyl or sulfonyl

Also Published As

Publication number Publication date
TW201833119A (zh) 2018-09-16
WO2018123920A1 (ja) 2018-07-05
JP2018104420A (ja) 2018-07-05

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