AT344332B - METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS - Google Patents

METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS

Info

Publication number
AT344332B
AT344332B AT153875A AT153875A AT344332B AT 344332 B AT344332 B AT 344332B AT 153875 A AT153875 A AT 153875A AT 153875 A AT153875 A AT 153875A AT 344332 B AT344332 B AT 344332B
Authority
AT
Austria
Prior art keywords
benzomorphanes
tetrahydrofurfuryl
acid addition
addition salts
producing new
Prior art date
Application number
AT153875A
Other languages
German (de)
Other versions
ATA153875A (en
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of ATA153875A publication Critical patent/ATA153875A/en
Application granted granted Critical
Publication of AT344332B publication Critical patent/AT344332B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT153875A 1974-03-09 1975-02-28 METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS AT344332B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2411382A DE2411382C3 (en) 1974-03-09 1974-03-09 2-Tetrahydrofurfuryl-6,7-benzomorphane, process for the preparation and their use

Publications (2)

Publication Number Publication Date
ATA153875A ATA153875A (en) 1977-11-15
AT344332B true AT344332B (en) 1978-07-10

Family

ID=5909593

Family Applications (1)

Application Number Title Priority Date Filing Date
AT153875A AT344332B (en) 1974-03-09 1975-02-28 METHOD FOR PRODUCING NEW 2-TETRAHYDROFURFURYL-6,7-BENZOMORPHANES AND THEIR ACID ADDITION SALTS

Country Status (25)

Country Link
JP (1) JPS5827275B2 (en)
AT (1) AT344332B (en)
BE (1) BE826440A (en)
BG (3) BG24813A4 (en)
CA (1) CA1049511A (en)
CH (8) CH612425A5 (en)
CS (1) CS188221B2 (en)
DD (1) DD119236A5 (en)
DE (1) DE2411382C3 (en)
DK (1) DK137188C (en)
ES (6) ES440346A1 (en)
FI (1) FI63571C (en)
FR (1) FR2262984B1 (en)
GB (1) GB1496418A (en)
HU (1) HU177408B (en)
IE (1) IE40945B1 (en)
IL (1) IL46760A (en)
NL (1) NL7502724A (en)
NO (1) NO141800C (en)
PH (1) PH14127A (en)
PL (3) PL93700B1 (en)
RO (2) RO70051A (en)
SE (1) SE421919B (en)
SU (3) SU577982A3 (en)
ZA (1) ZA751394B (en)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2716687A1 (en) * 1977-04-15 1978-10-19 Boehringer Sohn Ingelheim 2'-HYDROXY-2- (5-ISOXAZOLYLMETHYL) -6.7BENZOMORPHANES, THEIR ACID ADDITIONAL SALTS AND MEDICINAL PRODUCTS CONTAINING THEM
DE2828039A1 (en) * 1978-06-26 1980-01-10 Boehringer Sohn Ingelheim 2- (2-ALKOXYETHYL) -2'-HYDROXY-6,7-BENZOMORPHANES THEIR ACID ADDITION SALTS, THESE MEDICINAL PRODUCTS, AND METHOD FOR THE PRODUCTION THEREOF
HU225148B1 (en) * 1995-03-10 2006-07-28 Photocure Asa Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy or diagnosis, products and kits comprising thereof and method of in vitro diagnosis by their using
US7530461B2 (en) 1995-03-10 2009-05-12 Photocure Asa Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
US6492420B2 (en) 1995-03-10 2002-12-10 Photocure As Esters of 5-aminolevulinic acid as photosensitizing agents in photochemotherapy
US6992107B1 (en) 1995-03-10 2006-01-31 Photocure Asa Esters of 5-aminolevulinic acid and their use as photosensitizing compounds in photochemotherapy
GB0018528D0 (en) 2000-07-27 2000-09-13 Photocure Asa Compounds
US6723750B2 (en) 2002-03-15 2004-04-20 Allergan, Inc. Photodynamic therapy for pre-melanomas
JP5470557B2 (en) 2007-07-26 2014-04-16 ヴァイティー ファーマシューティカルズ,インコーポレイテッド Synthesis of inhibitors of 11β-hydroxysteroid dehydrogenase type 1
TW200927115A (en) 2007-11-16 2009-07-01 Boehringer Ingelheim Int Aryl-and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use
US8440658B2 (en) 2007-12-11 2013-05-14 Vitae Pharmaceuticals, Inc. Cyclic urea inhibitors of 11β-hydroxysteroid dehydrogenase 1
TW200934490A (en) 2008-01-07 2009-08-16 Vitae Pharmaceuticals Inc Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1
WO2009094169A1 (en) 2008-01-24 2009-07-30 Vitae Pharmaceuticals, Inc. Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8598160B2 (en) 2008-02-15 2013-12-03 Vitae Pharmaceuticals, Inc. Cycloalkyl lactame derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
JP5696037B2 (en) 2008-05-01 2015-04-08 ヴァイティー ファーマシューティカルズ,インコーポレイテッド Cyclic inhibitor of 11β-hydroxysteroid dehydrogenase 1
EP2291370B1 (en) 2008-05-01 2013-11-27 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
RU2531272C2 (en) 2008-05-01 2014-10-20 Вайтаи Фармасьютиклз, Инк. Cyclic inhibitors of 11beta-hydroxysteroid-dehydrogenase 1
AR071719A1 (en) 2008-05-13 2010-07-07 Boehringer Ingelheim Int ALICICLIC DERIVATIVES OF CARBOXILIC ACID OF BENZOMORPHANS AND RELATED STRUCTURES, MEDICINES CONTAINING THESE COMPOUNDS AND THEIR USE. OBTAINING PROCESSES
NZ590495A (en) 2008-07-25 2012-10-26 Vitae Pharmaceuticals Inc Dihydropyridin-phenyl-3-oxazinan-2-ones as inhibitors of 11beta-hydroxysteroid dehydrogenase 1
WO2010010157A2 (en) 2008-07-25 2010-01-28 Boehringer Ingelheim International Gmbh INHIBITORS OF 11beta-HYDROXYSTEROID DEHYDROGENASE 1
US8680093B2 (en) 2009-04-30 2014-03-25 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1
US8927539B2 (en) 2009-06-11 2015-01-06 Vitae Pharmaceuticals, Inc. Cyclic inhibitors of 11β-hydroxysteroid dehydrogenase 1 based on the 1,3-oxazinan-2-one structure
AR078887A1 (en) 2009-11-06 2011-12-07 Boehringer Ingelheim Int ARILO AND HETEROARILCARBONILO DERIVATIVES OF HEXAHYDROINDENOPIRIDINE AND OCTAHYDROBENZOQUINOLINE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
WO2011159760A1 (en) 2010-06-16 2011-12-22 Vitae Pharmaceuticals, Inc. Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use
TWI537258B (en) 2010-11-05 2016-06-11 百靈佳殷格翰國際股份有限公司 Aryl-and heteroarylcarbonyl derivatives of hexahydroindenopyridine and octahydrobenzoquinoline
WO2013025664A1 (en) 2011-08-17 2013-02-21 Boehringer Ingelheim International Gmbh Indenopyridine derivatives

Also Published As

Publication number Publication date
DE2411382B2 (en) 1979-01-18
ES440347A1 (en) 1977-06-01
FI63571C (en) 1983-07-11
ES440346A1 (en) 1977-03-01
JPS50123675A (en) 1975-09-29
IL46760A (en) 1978-12-17
NO141800C (en) 1980-06-04
DE2411382A1 (en) 1975-09-18
ES440349A1 (en) 1977-03-01
JPS5827275B2 (en) 1983-06-08
RO69617A (en) 1980-08-15
RO70051A (en) 1980-12-30
HU177408B (en) 1981-10-28
NO750773L (en) 1975-09-10
DK92975A (en) 1975-09-10
PL93699B1 (en) 1977-06-30
CH622017A5 (en) 1981-03-13
CS188221B2 (en) 1979-02-28
SE7502592L (en) 1975-09-10
BG24813A4 (en) 1978-05-12
IE40945L (en) 1975-09-09
FR2262984A1 (en) 1975-10-03
DE2411382C3 (en) 1979-09-06
BG25087A3 (en) 1978-07-12
FI750652A7 (en) 1975-09-10
ATA153875A (en) 1977-11-15
CH620439A5 (en) 1980-11-28
DD119236A5 (en) 1976-04-12
ES440350A1 (en) 1977-03-16
CH612425A5 (en) 1979-07-31
NO141800B (en) 1980-02-04
SU577983A3 (en) 1977-10-25
AU7894275A (en) 1976-09-16
IE40945B1 (en) 1979-09-12
FI63571B (en) 1983-03-31
ES440348A1 (en) 1977-06-01
BE826440A (en) 1975-09-08
SU577982A3 (en) 1977-10-25
ES440345A1 (en) 1977-03-01
IL46760A0 (en) 1975-05-22
CA1049511A (en) 1979-02-27
ZA751394B (en) 1976-11-24
BG24814A4 (en) 1978-05-12
CH622016A5 (en) 1981-03-13
PL93499B1 (en) 1977-05-30
FR2262984B1 (en) 1978-07-28
SU588916A3 (en) 1978-01-15
SE421919B (en) 1982-02-08
DK137188B (en) 1978-01-30
CH620440A5 (en) 1980-11-28
CH620681A5 (en) 1980-12-15
NL7502724A (en) 1975-09-11
CH622014A5 (en) 1981-03-13
DK137188C (en) 1978-07-03
PH14127A (en) 1981-02-26
PL93700B1 (en) 1977-06-30
CH622015A5 (en) 1981-03-13
GB1496418A (en) 1977-12-30

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Legal Events

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ELJ Ceased due to non-payment of the annual fee
REN Ceased due to non-payment of the annual fee