ATA277774A - PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT - Google Patents

PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT

Info

Publication number
ATA277774A
ATA277774A AT277774A AT277774A ATA277774A AT A277774 A ATA277774 A AT A277774A AT 277774 A AT277774 A AT 277774A AT 277774 A AT277774 A AT 277774A AT A277774 A ATA277774 A AT A277774A
Authority
AT
Austria
Prior art keywords
salt
production
piperazine derivatives
new piperazine
new
Prior art date
Application number
AT277774A
Other languages
German (de)
Other versions
AT340931B (en
Inventor
Shinsaku Minami
Junichi Matsumoto
Kazuyo Kawaguchi
Shinsaku Mishio
Masanao Shimizu
Yoshiyuki Takase
Shinichi Nakamura
Original Assignee
Dainippon Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP3845373A external-priority patent/JPS5546400B2/ja
Priority claimed from JP5654473A external-priority patent/JPS565753B2/ja
Priority claimed from JP6446473A external-priority patent/JPS565755B2/ja
Application filed by Dainippon Pharmaceutical Co filed Critical Dainippon Pharmaceutical Co
Publication of ATA277774A publication Critical patent/ATA277774A/en
Application granted granted Critical
Publication of AT340931B publication Critical patent/AT340931B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT277774A 1973-04-03 1974-04-03 PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT AT340931B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP3845373A JPS5546400B2 (en) 1973-04-03 1973-04-03
JP5654473A JPS565753B2 (en) 1973-05-21 1973-05-21
JP6446473A JPS565755B2 (en) 1973-06-07 1973-06-07

Publications (2)

Publication Number Publication Date
ATA277774A true ATA277774A (en) 1977-05-15
AT340931B AT340931B (en) 1978-01-10

Family

ID=27289838

Family Applications (1)

Application Number Title Priority Date Filing Date
AT277774A AT340931B (en) 1973-04-03 1974-04-03 PROCESS FOR THE PRODUCTION OF NEW PIPERAZINE DERIVATIVES AND THEIR SALT

Country Status (11)

Country Link
AR (2) AR204003A1 (en)
AT (1) AT340931B (en)
CA (1) CA1066701A (en)
CH (1) CH593281A5 (en)
ES (1) ES424851A1 (en)
FI (1) FI56011C (en)
IE (1) IE39102B1 (en)
NL (1) NL186087C (en)
NO (1) NO142221C (en)
PH (2) PH10529A (en)
SE (1) SE416051B (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1209163B (en) * 1979-12-21 1989-07-10 Unibios S P A Trecate Novara PROCEDURE FOR THE MANUFACTURE OF: 6-ALCOSSICARBONIL-8-ETHYL-5-OXO-5,8 DIIDRO-APERTA PAR. SQUARE 2,3-DCHIUSA PAR. SQUARE-PRIMIDINE 2-REPLACED AND ACID CORRESPONDING BOOKS.
EP2845856A1 (en) 2009-06-29 2015-03-11 Incyte Corporation Pyrimidinones as PI3K inhibitors
WO2011075630A1 (en) 2009-12-18 2011-06-23 Incyte Corporation Substituted fused aryl and heteroaryl derivatives as pi3k inhibitors
US8759359B2 (en) 2009-12-18 2014-06-24 Incyte Corporation Substituted heteroaryl fused derivatives as PI3K inhibitors
TW201249844A (en) 2010-12-20 2012-12-16 Incyte Corp N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors
UA121539C2 (en) 2011-09-02 2020-06-25 Інсайт Холдинґс Корпорейшн HETEROCYCLYLAMINE AS RI3K INHIBITORS
AR090548A1 (en) 2012-04-02 2014-11-19 Incyte Corp BICYCLIC AZAHETEROCICLOBENCILAMINS AS PI3K INHIBITORS
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
UA122332C2 (en) 2015-02-27 2020-10-26 Інсайт Корпорейшн Salts of pi3k inhibitor and processes for their preparation
WO2016183060A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Process for the synthesis of a phosphoinositide 3-kinase inhibitor
WO2016183063A1 (en) 2015-05-11 2016-11-17 Incyte Corporation Crystalline forms of a pi3k inhibitor
MX2020012826A (en) 2018-06-01 2021-03-09 Incyte Corp DOSAGE REGIMEN FOR THE TREATMENT OF DISORDERS RELATED TO PHOSPHATIDYLINOSITOL 3-KINASES (PI3K).

Also Published As

Publication number Publication date
CH593281A5 (en) 1977-11-30
FI56011C (en) 1979-11-12
NO740349L (en) 1974-10-04
CA1066701A (en) 1979-11-20
ES424851A1 (en) 1976-06-01
PH10984A (en) 1977-10-18
AR204003A1 (en) 1975-11-12
NL186087C (en) 1990-09-17
NL7401509A (en) 1974-10-07
IE39102B1 (en) 1978-08-02
NO142221C (en) 1980-07-16
PH10529A (en) 1977-05-30
FI56011B (en) 1979-07-31
AR204660A1 (en) 1976-02-20
IE39102L (en) 1974-10-03
AT340931B (en) 1978-01-10
NO142221B (en) 1980-04-08
NL186087B (en) 1990-04-17
SE416051B (en) 1980-11-24

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Legal Events

Date Code Title Description
ELA Expired due to lapse of time