ATA72783A - METHOD FOR PRODUCING NEW 1-SUBSTITUTED N- (8 ALPHA -ERGOLINYL) -N'-N'DI | THYL UREAS - Google Patents

METHOD FOR PRODUCING NEW 1-SUBSTITUTED N- (8 ALPHA -ERGOLINYL) -N'-N'DI | THYL UREAS

Info

Publication number
ATA72783A
ATA72783A AT0072783A AT72783A ATA72783A AT A72783 A ATA72783 A AT A72783A AT 0072783 A AT0072783 A AT 0072783A AT 72783 A AT72783 A AT 72783A AT A72783 A ATA72783 A AT A72783A
Authority
AT
Austria
Prior art keywords
ergolinyl
thyl
ureas
alpha
substituted
Prior art date
Application number
AT0072783A
Other languages
German (de)
Other versions
AT383349B (en
Original Assignee
Spofa Vereinigte Pharma Werke
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Spofa Vereinigte Pharma Werke filed Critical Spofa Vereinigte Pharma Werke
Publication of ATA72783A publication Critical patent/ATA72783A/en
Application granted granted Critical
Publication of AT383349B publication Critical patent/AT383349B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Endocrinology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT0072783A 1982-03-12 1983-03-02 METHOD FOR PRODUCING NEW 1-SUBSTITUTED N- (8 ALPHA -ERGOLINYL) -N'-N'DI | THYL UREAS AT383349B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS821734A CS231214B1 (en) 1982-03-12 1982-03-12 Processing method of 1-substituted n+l8alpha-ergoline+p-n,diethyl urea

Publications (2)

Publication Number Publication Date
ATA72783A true ATA72783A (en) 1986-11-15
AT383349B AT383349B (en) 1987-06-25

Family

ID=5352449

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0072783A AT383349B (en) 1982-03-12 1983-03-02 METHOD FOR PRODUCING NEW 1-SUBSTITUTED N- (8 ALPHA -ERGOLINYL) -N'-N'DI | THYL UREAS

Country Status (15)

Country Link
JP (1) JPS58180484A (en)
AT (1) AT383349B (en)
AU (1) AU555961B2 (en)
BE (1) BE896122A (en)
CA (1) CA1203531A (en)
CH (1) CH652125A5 (en)
CS (1) CS231214B1 (en)
DE (1) DE3308719A1 (en)
DK (1) DK84683A (en)
FI (1) FI830754A7 (en)
FR (1) FR2523131B1 (en)
GB (1) GB2116548B (en)
IT (1) IT1161209B (en)
NL (1) NL8300829A (en)
SE (1) SE452321B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3309493A1 (en) * 1983-03-14 1984-09-20 Schering AG, 1000 Berlin und 4709 Bergkamen NEW ERGOLIN DERIVATIVES, PROCESS FOR THEIR PRODUCTION AND USE AS A MEDICINAL PRODUCT
EP0208417A3 (en) * 1985-06-12 1989-09-06 SPOFA Spojené Podniky Pro Zdravotnickou Vyrobu Use of 1-(8-alpha-ergolinyl)-3,3-diethyl urea derivatives in the treatment of endometritis
DE3522894A1 (en) * 1985-06-24 1987-01-02 Schering Ag USE OF TERGURID AS GERIATRIC
FR2584720B1 (en) * 1985-07-11 1987-10-02 Rhone Poulenc Sante PROCESS FOR THE PREPARATION OF N-METHYL DERIVATIVES OF ERGOLINE
DE3620293A1 (en) * 1986-06-16 1987-12-17 Schering Ag 1 AND / OR 2 SUBSTITUTED ERGOL DERIVATIVES
DE3623503A1 (en) * 1986-07-09 1988-01-21 Schering Ag 1-ARYL-ERGOLINYL-UREA DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THE USE OF THESE COMPOUNDS AS A MEDICINAL PRODUCT
DE10212564B4 (en) * 2002-03-12 2007-04-19 Neurobiotec Gmbh 1-Allyl ergot alkaloid derivatives and their use for the prophylaxis and treatment of migraine
CN103476402A (en) * 2010-11-11 2013-12-25 西诺克萨医药有限公司 Lisuride, terguride and derivatives thereof for preventing and/or treating fibrotic lesions
JP6856532B2 (en) 2015-01-20 2021-04-07 エックスオーシー ファーマシューティカルズ インコーポレイテッドXoc Pharmaceuticals, Inc Ergoline compounds and their use
JP2018502889A (en) 2015-01-20 2018-02-01 エックスオーシー ファーマシューティカルズ インコーポレイテッドXoc Pharmaceuticals, Inc Isoergoline compounds and uses thereof
EP3630758A1 (en) 2017-06-01 2020-04-08 Xoc Pharmaceuticals, Inc Ergoline derivatives for use in medicine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH344731A (en) * 1956-05-18 1960-02-29 Sandoz Ag Process for the production of new derivatives of the lysergic acid series alkylated on the indole nitrogen
AT231082B (en) * 1960-10-12 1964-01-10 Sandoz Ag Process for the production of new urea derivatives
EP0021206B1 (en) * 1979-06-13 1983-06-22 Schering Aktiengesellschaft (ergolin-yl)-n', n'-diethyl urea derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
CH652125A5 (en) 1985-10-31
GB2116548A (en) 1983-09-28
AT383349B (en) 1987-06-25
CS231214B1 (en) 1984-10-15
FI830754L (en) 1983-09-13
IT8319935A0 (en) 1983-03-07
FI830754A0 (en) 1983-03-07
CA1203531A (en) 1986-04-22
DK84683D0 (en) 1983-02-24
FR2523131A1 (en) 1983-09-16
GB8305735D0 (en) 1983-04-07
DK84683A (en) 1983-09-13
AU1216783A (en) 1983-09-15
GB2116548B (en) 1985-03-20
BE896122A (en) 1983-07-01
SE8301257D0 (en) 1983-03-08
IT1161209B (en) 1987-03-18
SE8301257L (en) 1983-09-13
AU555961B2 (en) 1986-10-16
FR2523131B1 (en) 1987-08-28
NL8300829A (en) 1983-10-03
SE452321B (en) 1987-11-23
DE3308719A1 (en) 1983-09-22
JPS58180484A (en) 1983-10-21
FI830754A7 (en) 1983-09-13

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Legal Events

Date Code Title Description
ELJ Ceased due to non-payment of the annual fee
REN Ceased due to non-payment of the annual fee