ATE111467T1 - 4h-pyrrolo(1,2-a>thieno(3,2- f>(1,4>diazepinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen. - Google Patents

4h-pyrrolo(1,2-a>thieno(3,2- f>(1,4>diazepinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen.

Info

Publication number: ATE111467T1
Authority: AT; Austria
Prior art keywords: thieno; pyrrolo; preparation; radical; pharmaceutical preparations
Prior art date: 1990-03-08

Application number

AT91400620T

Other languages

English (en)

Inventor

Sylvain Rault

Michel Boulouard

Patrick Dallemagne

Max Robba

Beatrice Guardiola

Michelle Devissaguet

Original Assignee

Adir

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-03-08

Filing date

1991-03-07

Publication date

1994-09-15

1991-03-07 Application filed by Adir filed Critical Adir

1994-09-15 Application granted granted Critical

1994-09-15 Publication of ATE111467T1 publication Critical patent/ATE111467T1/de

Links

AAOVKJBEBIDNHE-UHFFFAOYSA-N diazepam Chemical class N=1CC(=O)N(C)C2=CC=C(Cl)C=C2C=1C1=CC=CC=C1 AAOVKJBEBIDNHE-UHFFFAOYSA-N 0.000 title 1
238000000034 method Methods 0.000 title 1
239000000825 pharmaceutical preparation Substances 0.000 title 1
238000002360 preparation method Methods 0.000 title 1
HNDGEYCCZGRMTN-UHFFFAOYSA-N thieno[3,2-f:4,5-f]bis[1]benzothiophene Chemical compound S1C2=CC=3SC=CC=3C=C2C2=C1C=C(SC=C1)C1=C2 HNDGEYCCZGRMTN-UHFFFAOYSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 1
229940079593 drug Drugs 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
238000002483 medication Methods 0.000 abstract 1
HZVOZRGWRWCICA-UHFFFAOYSA-N methanediyl Chemical compound [CH2] HZVOZRGWRWCICA-UHFFFAOYSA-N 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Vascular Medicine (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Hematology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AT91400620T 1990-03-08 1991-03-07 4h-pyrrolo(1,2-a>thieno(3,2- f>(1,4>diazepinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen. ATE111467T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9002933A FR2659331A1 (fr)	1990-03-08	1990-03-08	Nouveaux derives de la 4h-pyrrolo [1,2-a] thieno [3,2-f] [1,4]-diazepine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number	Publication Date
ATE111467T1 true ATE111467T1 (de)	1994-09-15

Family

ID=9394511

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT91400620T ATE111467T1 (de)	1990-03-08	1991-03-07	4h-pyrrolo(1,2-a>thieno(3,2- f>(1,4>diazepinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen.

Country Status (14)

Country	Link
US (1)	US5190939A (de)
EP (1)	EP0446133B1 (de)
JP (1)	JPH04234889A (de)
AT (1)	ATE111467T1 (de)
AU (1)	AU632906B2 (de)
CA (1)	CA2037654A1 (de)
DE (1)	DE69103934T2 (de)
ES (1)	ES2064054T3 (de)
FR (1)	FR2659331A1 (de)
IE (1)	IE910769A1 (de)
NZ (1)	NZ237365A (de)
OA (1)	OA09486A (de)
PT (1)	PT96964A (de)
ZA (1)	ZA911727B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2660310B1 (fr) *	1990-03-27	1992-06-05	Adir	Nouveaux derives de la 4h-pyrrolo[1,2a] thieno[2,3-f] diazepine[1,4], leur procede de preparation et les compositions pharmaceutiques les renfermant.
WO1995032963A1 (en) *	1994-06-01	1995-12-07	Yoshitomi Pharmaceutical Industries, Ltd.	Thienylazole compound and thienotriazolodiazepine compound
HU214588B (hu) *	1994-07-01	1998-04-28	EGIS Gyógyszergyár Rt.	Eljárás bicikloheptán-származékot tartalmazó, CCK-rendszer gátló hatású gyógyászati készítmények előállítására

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1332410C (en) *	1984-06-26	1994-10-11	Roger M. Freidinger	Benzodiazepine analogs
EP0368175A1 (de) *	1988-11-06	1990-05-16	Boehringer Ingelheim Kg	3S,7S-3-(Morpholinocarbonyl)-5-(2-chlorphenyl)-7,10-dimethyl-3,4-dihydro-2H,7H-cyclopenta[4,5]thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin.

1990
- 1990-03-08 FR FR9002933A patent/FR2659331A1/fr active Pending
1991
- 1991-03-06 CA CA002037654A patent/CA2037654A1/fr not_active Abandoned
- 1991-03-07 ES ES91400620T patent/ES2064054T3/es not_active Expired - Lifetime
- 1991-03-07 DE DE69103934T patent/DE69103934T2/de not_active Expired - Fee Related
- 1991-03-07 AU AU72710/91A patent/AU632906B2/en not_active Ceased
- 1991-03-07 AT AT91400620T patent/ATE111467T1/de not_active IP Right Cessation
- 1991-03-07 EP EP91400620A patent/EP0446133B1/de not_active Expired - Lifetime
- 1991-03-07 US US07/665,812 patent/US5190939A/en not_active Expired - Fee Related
- 1991-03-07 PT PT96964A patent/PT96964A/pt not_active Application Discontinuation
- 1991-03-08 IE IE076991A patent/IE910769A1/en unknown
- 1991-03-08 OA OA59970A patent/OA09486A/xx unknown
- 1991-03-08 NZ NZ237365A patent/NZ237365A/en unknown
- 1991-03-08 JP JP3125608A patent/JPH04234889A/ja active Pending
- 1991-03-08 ZA ZA911727A patent/ZA911727B/xx unknown

Also Published As

Publication number	Publication date
IE910769A1 (en)	1991-09-11
ES2064054T3 (es)	1995-01-16
DE69103934T2 (de)	1995-04-20
AU632906B2 (en)	1993-01-14
ZA911727B (en)	1991-12-24
PT96964A (pt)	1991-10-31
EP0446133B1 (de)	1994-09-14
FR2659331A1 (fr)	1991-09-13
US5190939A (en)	1993-03-02
AU7271091A (en)	1991-09-12
JPH04234889A (ja)	1992-08-24
CA2037654A1 (fr)	1991-09-09
DE69103934D1 (de)	1994-10-20
EP0446133A1 (de)	1991-09-11
NZ237365A (en)	1991-12-23
OA09486A (fr)	1992-11-15

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Legal Events

Date	Code	Title	Description
1995-04-15	UEP	Publication of translation of european patent specification
1996-12-15	REN	Ceased due to non-payment of the annual fee