ATE120368T1 - Estradiol enthaltende transdermale zubereitung. - Google Patents
Estradiol enthaltende transdermale zubereitung.Info
- Publication number
- ATE120368T1 ATE120368T1 AT91908854T AT91908854T ATE120368T1 AT E120368 T1 ATE120368 T1 AT E120368T1 AT 91908854 T AT91908854 T AT 91908854T AT 91908854 T AT91908854 T AT 91908854T AT E120368 T1 ATE120368 T1 AT E120368T1
- Authority
- AT
- Austria
- Prior art keywords
- polymer
- preparation containing
- containing estradiol
- block
- transdermal preparation
- Prior art date
Links
- VOXZDWNPVJITMN-ZBRFXRBCSA-N 17β-estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 VOXZDWNPVJITMN-ZBRFXRBCSA-N 0.000 title abstract 2
- 229960005309 estradiol Drugs 0.000 title abstract 2
- 229930182833 estradiol Natural products 0.000 title abstract 2
- 229920000642 polymer Polymers 0.000 abstract 4
- 239000002250 absorbent Substances 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 150000001491 aromatic compounds Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229920001577 copolymer Polymers 0.000 abstract 1
- DNTGGZPQPQTDQF-XBXARRHUSA-N crotamiton Chemical compound C/C=C/C(=O)N(CC)C1=CC=CC=C1C DNTGGZPQPQTDQF-XBXARRHUSA-N 0.000 abstract 1
- 229960003338 crotamiton Drugs 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
- A61K9/7061—Polyacrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7069—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained otherwise than by reactions only involving carbon to carbon unsaturated bonds, e.g. polysiloxane, polyesters, polyurethane, polyethylene oxide
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP12816090 | 1990-05-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE120368T1 true ATE120368T1 (de) | 1995-04-15 |
Family
ID=14977874
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT91908854T ATE120368T1 (de) | 1990-05-17 | 1991-04-26 | Estradiol enthaltende transdermale zubereitung. |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5248676A (de) |
| EP (1) | EP0483370B1 (de) |
| AT (1) | ATE120368T1 (de) |
| AU (1) | AU633733B2 (de) |
| CA (1) | CA2066249C (de) |
| DE (1) | DE69108512T2 (de) |
| WO (1) | WO1991017752A1 (de) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2971224B2 (ja) | 1991-11-30 | 1999-11-02 | 久光製薬株式会社 | エストラジオール経皮吸収貼付剤 |
| US7134236B2 (en) | 1994-04-19 | 2006-11-14 | Applied Elastomerics, Inc. | Gelatinous elastomer compositions and articles for use as fishing bait |
| US7208184B2 (en) | 2002-07-20 | 2007-04-24 | Applied Elastomerics, Inc. | Gelatinous food elastomer compositions and articles for use as fishing bait |
| US7108873B2 (en) | 1994-04-19 | 2006-09-19 | Applied Elastomerics, Inc. | Gelatinous food elastomer compositions and articles |
| DE4237453C1 (de) * | 1992-11-06 | 1993-08-19 | Lts Lohmann Therapie-Systeme Gmbh & Co Kg, 5450 Neuwied, De | |
| DE4336557C2 (de) | 1993-05-06 | 1997-07-17 | Lohmann Therapie Syst Lts | Estradiolhaltiges transdermales therapeutisches System, Verfahren zu seiner Herstellung und seine Verwendung |
| DE4400770C1 (de) * | 1994-01-13 | 1995-02-02 | Lohmann Therapie Syst Lts | Wirkstoffhaltiges Pflaster zur Abgabe von Estradiol mit mindestens einem Penetrationsverstärker, Verfahren zu seiner Herstellung und seine Verwendung |
| FR2717688B1 (fr) * | 1994-03-28 | 1996-07-05 | Lhd Lab Hygiene Dietetique | Système matriciel transdermique d'administration d'un oestrogène et/ou un progestatif à base d'EVA. |
| FR2717689B1 (fr) * | 1994-03-28 | 1996-07-05 | Lhd Lab Hygiene Dietetique | Système matriciel transdermique d'administration d'un oestrogène et/ou un progestatif à base de copolymère styrène-isoprène-styrène. |
| US7290367B2 (en) | 1994-04-19 | 2007-11-06 | Applied Elastomerics, Inc. | Tear resistant gel articles for various uses |
| US7234560B2 (en) | 1994-04-19 | 2007-06-26 | Applied Elastomerics, Inc. | Inflatable restraint cushions and other uses |
| US7226484B2 (en) | 1994-04-19 | 2007-06-05 | Applied Elastomerics, Inc. | Tear resistant gels and articles for every uses |
| GR1002079B (en) * | 1994-07-26 | 1995-12-05 | Lavipharm A E | System of a special structure and composition for the rapid transdermal administration of oestrogens. |
| EP0787488A4 (de) * | 1994-11-18 | 1998-06-03 | Hisamitsu Pharmaceutical Co | Transdermal absorbierbares pflaster |
| US5861431A (en) * | 1995-06-07 | 1999-01-19 | Iotek, Inc. | Incontinence treatment |
| AU7238896A (en) * | 1995-09-14 | 1997-04-01 | Cygnus, Inc. | High capacity, superabsorbent drug reservoirs for use in transdermal drug delivery systems |
| FR2739031B1 (fr) * | 1995-09-27 | 1997-11-21 | Lhd Lab Hygiene Dietetique | Systeme matriciel transdermique d'administration d'un oestrogene et/ou d'un progestatif a base de copolymere styrene-isoprene-styrene, procede de preparation et utilisation en therapeutique |
| DE19705138A1 (de) * | 1997-02-11 | 1998-08-13 | Lohmann Therapie Syst Lts | Dehnbares transdermales therapeutisches System |
| CA2287463A1 (en) * | 1997-04-16 | 1998-10-22 | Munehiko Hirano | Base composition for percutaneous absorption and percutaneously absorbable preparation containing the base composition |
| GB9828480D0 (en) * | 1998-12-24 | 1999-02-17 | Dermatech Limited | Transdermal drug delivery system |
| US8124122B2 (en) | 2002-08-09 | 2012-02-28 | Teikoku Seiyaku Co., Ltd. | Female hormone-containing patch |
| SI1594483T1 (sl) * | 2003-02-21 | 2006-12-31 | Schering Ag | UV-stabilni transdermalni terapevtski obliz |
| US8668925B2 (en) | 2003-12-12 | 2014-03-11 | Bayer Intellectual Property Gmbh | Transdermal delivery of hormones without the need of penetration enhancers |
| US8962013B2 (en) | 2005-05-02 | 2015-02-24 | Bayer Intellectual Property Gmbh | Multi-layered transdermal system with triazine UV absorber |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2045618B (en) * | 1979-04-03 | 1983-05-11 | Hisamitsu Pharmaceutical Co | Adhesive plaster |
| JPS60188314A (ja) * | 1984-03-07 | 1985-09-25 | Yamanouchi Pharmaceut Co Ltd | 鎮痒プラスタ− |
| JPS60188315A (ja) * | 1984-03-07 | 1985-09-25 | Yamanouchi Pharmaceut Co Ltd | グリチルレチン酸配合鎮痒プラスター |
| DE3587616D1 (de) * | 1984-12-22 | 1993-11-11 | Sanol Arznei Schwarz Gmbh | Wirkstoffpflaster. |
| US4788062A (en) * | 1987-02-26 | 1988-11-29 | Alza Corporation | Transdermal administration of progesterone, estradiol esters, and mixtures thereof |
| CH674618A5 (de) * | 1987-04-02 | 1990-06-29 | Ciba Geigy Ag | |
| US4994267A (en) * | 1988-03-04 | 1991-02-19 | Noven Pharmaceuticals, Inc. | Transdermal acrylic multipolymer drug delivery system |
| AU622162B2 (en) * | 1988-04-22 | 1992-04-02 | Ciba-Geigy Ag | Transdermal monolith systems |
| JP2849937B2 (ja) * | 1990-04-18 | 1999-01-27 | 日東電工株式会社 | 医療用貼付剤 |
-
1991
- 1991-04-26 AT AT91908854T patent/ATE120368T1/de not_active IP Right Cessation
- 1991-04-26 US US07/834,335 patent/US5248676A/en not_active Expired - Fee Related
- 1991-04-26 EP EP91908854A patent/EP0483370B1/de not_active Expired - Lifetime
- 1991-04-26 WO PCT/JP1991/000578 patent/WO1991017752A1/ja not_active Ceased
- 1991-04-26 CA CA002066249A patent/CA2066249C/en not_active Expired - Fee Related
- 1991-04-26 AU AU77800/91A patent/AU633733B2/en not_active Ceased
- 1991-04-26 DE DE69108512T patent/DE69108512T2/de not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2066249A1 (en) | 1991-11-18 |
| CA2066249C (en) | 1997-12-16 |
| DE69108512D1 (de) | 1995-05-04 |
| EP0483370A4 (en) | 1992-10-28 |
| WO1991017752A1 (en) | 1991-11-28 |
| US5248676A (en) | 1993-09-28 |
| EP0483370A1 (de) | 1992-05-06 |
| EP0483370B1 (de) | 1995-03-29 |
| AU633733B2 (en) | 1993-02-04 |
| DE69108512T2 (de) | 1995-08-03 |
| AU7780091A (en) | 1991-12-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |