ATE122669T1 - Zearalanol-derivate mit anabolytischer wirkung. - Google Patents

Zearalanol-derivate mit anabolytischer wirkung.

Info

Publication number: ATE122669T1
Authority: AT; Austria
Prior art keywords: anabolytic; action; hydrogen; hydroxyl; compounds
Prior art date: 1987-10-13

Application number

AT88309598T

Other languages

English (en)

Inventor

Martin J Jacobs

Original Assignee

Mallinckrodt Veterinary Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-10-13

Filing date

1988-10-13

Publication date

1995-06-15

1988-10-13 Application filed by Mallinckrodt Veterinary Inc filed Critical Mallinckrodt Veterinary Inc

1995-06-15 Application granted granted Critical

1995-06-15 Publication of ATE122669T1 publication Critical patent/ATE122669T1/de

Links

FPQFYIAXQDXNOR-QDKLYSGJSA-N alpha-Zearalenol Chemical class O=C1O[C@@H](C)CCC[C@H](O)CCC\C=C\C2=CC(O)=CC(O)=C21 FPQFYIAXQDXNOR-QDKLYSGJSA-N 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 3
229910052739 hydrogen Inorganic materials 0.000 abstract 3
239000001257 hydrogen Substances 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
150000001875 compounds Chemical class 0.000 abstract 2
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
229930194542 Keto Natural products 0.000 abstract 1
241001465754 Metazoa Species 0.000 abstract 1
229940124325 anabolic agent Drugs 0.000 abstract 1
239000003263 anabolic agent Substances 0.000 abstract 1
230000000845 anti-microbial effect Effects 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
230000003054 hormonal effect Effects 0.000 abstract 1
125000000468 ketone group Chemical group 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Beans For Foods Or Fodder (AREA)
Compounds Of Unknown Constitution (AREA)
Cephalosporin Compounds (AREA)
Pyrane Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

AT88309598T 1987-10-13 1988-10-13 Zearalanol-derivate mit anabolytischer wirkung. ATE122669T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/108,539 US4849447A (en)	1987-10-13	1987-10-13	Zearalanol derivatives with anabolic activity

Publications (1)

Publication Number	Publication Date
ATE122669T1 true ATE122669T1 (de)	1995-06-15

Family

ID=22322783

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT88309598T ATE122669T1 (de)	1987-10-13	1988-10-13	Zearalanol-derivate mit anabolytischer wirkung.

Country Status (6)

Country	Link
US (1)	US4849447A (de)
EP (1)	EP0312353B1 (de)
JP (1)	JPH01199960A (de)
AT (1)	ATE122669T1 (de)
DE (1)	DE3853804T2 (de)
ES (1)	ES2072264T3 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5185365A (en) *	1992-06-24	1993-02-09	Cornell Research Foundation, Inc.	Insect deterrent azamcrolides
JP5465006B2 (ja)	2006-08-11	2014-04-09	ユニベルシテ・ドウ・ストラスブール	キナーゼおよびｈｓｐ９０の阻害剤として有用な大環状化合物
ES2581765T3 (es)	2006-08-24	2016-09-07	University Of Tennessee Research Foundation	Acilanilidas sustituidas y métodos de uso de las mismas
US20110190237A1 (en) *	2008-01-15	2011-08-04	Nexgenix Pharmaceuticals	Macrocyclic Prodrug Compounds Useful as Therapeutics
US9622992B2 (en)	2012-07-13	2017-04-18	Gtx, Inc.	Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs)
US9744149B2 (en)	2012-07-13	2017-08-29	Gtx, Inc.	Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs)
LT2872482T (lt)	2012-07-13	2020-12-28	Oncternal Therapeutics, Inc.	Krūties vėžių gydymo būdas selektyviu androgeno receptoriaus moduliatoriumi
US10987334B2 (en)	2012-07-13	2021-04-27	University Of Tennessee Research Foundation	Method of treating ER mutant expressing breast cancers with selective androgen receptor modulators (SARMs)
US10258596B2 (en)	2012-07-13	2019-04-16	Gtx, Inc.	Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS)
US9969683B2 (en)	2012-07-13	2018-05-15	Gtx, Inc.	Method of treating estrogen receptor (ER)-positive breast cancers with selective androgen receptor modulator (SARMS)
US10314807B2 (en)	2012-07-13	2019-06-11	Gtx, Inc.	Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3453367A (en) *	1966-06-29	1969-07-01	Commercial Solvents Corp	Methods for treating inflammation with estrogenic compounds
FR96016E (fr) *	1966-06-29	1972-05-19	Commercial Solvents Corp	Composé utilisable comme supplément alimentaire pour les animaux.
FR96046E (fr) *	1966-06-29	1972-05-19	Commercial Solvents Corp	Composé utilisable comme supplément alimentaire pour les animaux.
US3373037A (en) *	1966-06-29	1968-03-12	Commercial Solvents Corp	Estrogenic compounds and animal growth promoters
US3887583A (en) *	1968-05-15	1975-06-03	Commercial Solvents Corp	Products and process
US3957825A (en) *	1972-04-25	1976-05-18	Commercial Solvents Corporation	Process for synthesizing zearalanone and related compounds
US4024602A (en) *	1975-02-10	1977-05-24	Actionite Company, Inc.	Apparatus for decasing food links
US4148808A (en) *	1975-08-22	1979-04-10	Int Minerals & Chem Corp	Method for reducing zearalenone
US4239772A (en) *	1979-05-30	1980-12-16	International Minerals & Chemical Corp.	Allyl and propyl zearalenone derivatives and their use as growth promoting agents
US4443470A (en) *	1981-09-03	1984-04-17	International Minerals & Chemical Corp.	Method of promoting growth and enhancing feed efficiency in meat producing animals

1987
- 1987-10-13 US US07/108,539 patent/US4849447A/en not_active Expired - Fee Related
1988
- 1988-10-12 JP JP63255019A patent/JPH01199960A/ja active Pending
- 1988-10-13 ES ES88309598T patent/ES2072264T3/es not_active Expired - Lifetime
- 1988-10-13 EP EP88309598A patent/EP0312353B1/de not_active Expired - Lifetime
- 1988-10-13 AT AT88309598T patent/ATE122669T1/de not_active IP Right Cessation
- 1988-10-13 DE DE3853804T patent/DE3853804T2/de not_active Expired - Fee Related

Also Published As

Publication number	Publication date
ES2072264T3 (es)	1995-07-16
EP0312353B1 (de)	1995-05-17
EP0312353A2 (de)	1989-04-19
US4849447A (en)	1989-07-18
JPH01199960A (ja)	1989-08-11
DE3853804D1 (de)	1995-06-22
DE3853804T2 (de)	1995-11-02
EP0312353A3 (en)	1990-06-20

Legal Events

Date	Code	Title	Description
1995-11-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
NO873939D0 (no)	1987-09-21	Fremgangsmaate for fremstilling av terapeutisk aktive retinsyrederivater.
ES2166359T3 (es)	2002-04-16	Derivado de depsipeptido, su produccion y uso.
EP0256503A3 (en)	1989-07-19	Pyridinecarboxamide derivatives and their use as fungicide
ATE223378T1 (de)	2002-09-15	Prolineamid-derivate
ATE132862T1 (de)	1996-01-15	Aryl- und heteroaryl-piperazinylcarboxamide mit wirkung auf das zentrale nervensystem
FI914187A0 (fi)	1991-09-05	Menetelmä valmistaa kaavan /I/ mukaista 1-metyylikarbapeneemijohdosta
ATE122669T1 (de)	1995-06-15	Zearalanol-derivate mit anabolytischer wirkung.
DE69215694D1 (de)	1997-01-16	Benzamid-derivate
DE3665711D1 (de)	1989-10-26	Novel guanidinomethylbenzoic acid derivatives
DE69125360D1 (de)	1997-04-30	Alkylester von oxidiertem Glutathion
SE8100403L (sv)	1981-07-30	Cyklohexen-derivat
FR2681864B1 (fr)	1995-03-31	Nouveaux derives bicycliques azotes, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
DE69123757D1 (de)	1997-01-30	Epoxysuccinamidsäurederivat
AR246965A1 (es)	1994-10-31	Procedimiento para fabricar un derivado del acido 1-3-dioxan-alquenoico.
SE8200679L (sv)	1982-09-22	1-bensyl-4-(4-(2-pyrimidinylamino) bensyl 1-2,3-dioxopiperazinderivat, salter derav, forfarande for framstellning derav och karcinostatiska medel der de ingar
IE873442L (en)	1988-06-18	Cephalosporin derivative
ES2096628T3 (es)	1997-03-16	Derivados heterociclicos.
ATE53163T1 (de)	1990-06-15	Desinfektionszusammensetzungen.
EG18407A (en)	1993-02-28	Stable injectable antiemetic compositions
ES2059097T3 (es)	1994-11-01	Derivados de la ergolina.
DE3782229D1 (de)	1992-11-19	Verwendung von 2-oxo-imidazolidin-derivaten zur behandlung von nierenkrankheiten.