ATE159725T1 - 2-aminozuckermakrolid-derivate - Google Patents

2-aminozuckermakrolid-derivate

Info

Publication number
ATE159725T1
ATE159725T1 AT93903554T AT93903554T ATE159725T1 AT E159725 T1 ATE159725 T1 AT E159725T1 AT 93903554 T AT93903554 T AT 93903554T AT 93903554 T AT93903554 T AT 93903554T AT E159725 T1 ATE159725 T1 AT E159725T1
Authority
AT
Austria
Prior art keywords
pct
amino sugar
group
macrolide derivatives
sec
Prior art date
Application number
AT93903554T
Other languages
English (en)
Inventor
Kevin Koch
Gary R Schulte
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE159725T1 publication Critical patent/ATE159725T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT93903554T 1992-03-02 1993-01-27 2-aminozuckermakrolid-derivate ATE159725T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US84433992A 1992-03-02 1992-03-02

Publications (1)

Publication Number Publication Date
ATE159725T1 true ATE159725T1 (de) 1997-11-15

Family

ID=25292446

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93903554T ATE159725T1 (de) 1992-03-02 1993-01-27 2-aminozuckermakrolid-derivate

Country Status (11)

Country Link
US (1) US5631235A (de)
EP (1) EP0636136B1 (de)
JP (1) JP2562001B2 (de)
AT (1) ATE159725T1 (de)
CA (1) CA2131373C (de)
DE (1) DE69314947T2 (de)
DK (1) DK0636136T3 (de)
ES (1) ES2108261T3 (de)
FI (1) FI107537B (de)
GR (1) GR3025672T3 (de)
WO (1) WO1993018048A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP584198A0 (en) * 1998-09-14 1998-10-08 Fujisawa Pharmaceutical Co., Ltd. New use
US7160867B2 (en) 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
EP1768662A2 (de) 2004-06-24 2007-04-04 Novartis Vaccines and Diagnostics, Inc. Immunstimulatoren kleiner moleküle und assays für deren nachweis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
JPH05504944A (ja) * 1989-08-18 1993-07-29 藤沢薬品工業株式会社 巨大環式化合物
EP0427680B1 (de) * 1989-11-09 1995-08-23 Sandoz Ltd. Heteroatome enthaltende tricyclische Verbindungen
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism

Also Published As

Publication number Publication date
EP0636136A1 (de) 1995-02-01
CA2131373C (en) 1999-01-26
CA2131373A1 (en) 1993-09-16
WO1993018048A1 (en) 1993-09-16
DK0636136T3 (da) 1997-12-22
DE69314947D1 (de) 1997-12-04
FI944015A0 (fi) 1994-09-01
GR3025672T3 (en) 1998-03-31
DE69314947T2 (de) 1998-03-05
ES2108261T3 (es) 1997-12-16
FI944015L (fi) 1994-09-01
FI107537B (fi) 2001-08-31
US5631235A (en) 1997-05-20
JPH07500350A (ja) 1995-01-12
JP2562001B2 (ja) 1996-12-11
EP0636136B1 (de) 1997-10-29

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee