ES2108261T3 - Derivados 2-aminoazucar de macrolidos. - Google Patents
Derivados 2-aminoazucar de macrolidos.Info
- Publication number
- ES2108261T3 ES2108261T3 ES93903554T ES93903554T ES2108261T3 ES 2108261 T3 ES2108261 T3 ES 2108261T3 ES 93903554 T ES93903554 T ES 93903554T ES 93903554 T ES93903554 T ES 93903554T ES 2108261 T3 ES2108261 T3 ES 2108261T3
- Authority
- ES
- Spain
- Prior art keywords
- macrolides
- azucar
- derivatives
- amino
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 239000003120 macrolide antibiotic agent Substances 0.000 title abstract 2
- 229940041033 macrolides Drugs 0.000 title abstract 2
- GOJUJUVQIVIZAV-UHFFFAOYSA-N 2-amino-4,6-dichloropyrimidine-5-carbaldehyde Chemical compound NC1=NC(Cl)=C(C=O)C(Cl)=N1 GOJUJUVQIVIZAV-UHFFFAOYSA-N 0.000 title 1
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 201000004681 Psoriasis Diseases 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
LOS MACROLIDOS DE LA FORMULA (I) Y LOS METODOS DE TRATAMIENTO DE RESISTENCIA A LOS TRANSPLANTES, INFECCIONES DE HONGOS Y ENFERMEDADES AUTOINMUNES TALES COMO ARTRITIS REUMATOIDE Y PSORIASIS QUE USAN DICHOS MACROLIDOS DE LA FORMULA (I), EN DONDE N ES 1 O 2; A Y B VAN JUNTOS Y FORMAN =O O A Y B VAN SEPARADAMENTE Y SON CADA UNO H O A ES OH Y B ES H; R1 ES UN GRUPO 2-AMINOGLICOSIL; R2 ES OH O UN GRUPO GLICOSILOXI; Y R3 ES UN GRUPO ALQUILO O ALILO.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US84433992A | 1992-03-02 | 1992-03-02 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2108261T3 true ES2108261T3 (es) | 1997-12-16 |
Family
ID=25292446
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES93903554T Expired - Lifetime ES2108261T3 (es) | 1992-03-02 | 1993-01-27 | Derivados 2-aminoazucar de macrolidos. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US5631235A (es) |
| EP (1) | EP0636136B1 (es) |
| JP (1) | JP2562001B2 (es) |
| AT (1) | ATE159725T1 (es) |
| CA (1) | CA2131373C (es) |
| DE (1) | DE69314947T2 (es) |
| DK (1) | DK0636136T3 (es) |
| ES (1) | ES2108261T3 (es) |
| FI (1) | FI107537B (es) |
| GR (1) | GR3025672T3 (es) |
| WO (1) | WO1993018048A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPP584198A0 (en) * | 1998-09-14 | 1998-10-08 | Fujisawa Pharmaceutical Co., Ltd. | New use |
| US7160867B2 (en) | 2003-05-16 | 2007-01-09 | Isotechnika, Inc. | Rapamycin carbohydrate derivatives |
| EP1768662A2 (en) | 2004-06-24 | 2007-04-04 | Novartis Vaccines and Diagnostics, Inc. | Small molecule immunopotentiators and assays for their detection |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4894366A (en) * | 1984-12-03 | 1990-01-16 | Fujisawa Pharmaceutical Company, Ltd. | Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same |
| JPH05504944A (ja) * | 1989-08-18 | 1993-07-29 | 藤沢薬品工業株式会社 | 巨大環式化合物 |
| EP0427680B1 (en) * | 1989-11-09 | 1995-08-23 | Sandoz Ltd. | Heteroatoms-containing tricyclic compounds |
| IE904050A1 (en) * | 1989-11-13 | 1991-05-22 | Merck & Co Inc | Aminomacrolides and derivatives having immunosuppressive¹activity |
| EP0466365A3 (en) * | 1990-07-03 | 1992-04-15 | Merck & Co. Inc. | Novel immunosuppressant fermentation products of a microorganism |
-
1993
- 1993-01-27 WO PCT/US1993/000427 patent/WO1993018048A1/en not_active Ceased
- 1993-01-27 JP JP5515659A patent/JP2562001B2/ja not_active Expired - Fee Related
- 1993-01-27 CA CA002131373A patent/CA2131373C/en not_active Expired - Fee Related
- 1993-01-27 ES ES93903554T patent/ES2108261T3/es not_active Expired - Lifetime
- 1993-01-27 DK DK93903554.9T patent/DK0636136T3/da active
- 1993-01-27 AT AT93903554T patent/ATE159725T1/de not_active IP Right Cessation
- 1993-01-27 EP EP93903554A patent/EP0636136B1/en not_active Expired - Lifetime
- 1993-01-27 DE DE69314947T patent/DE69314947T2/de not_active Expired - Fee Related
- 1993-01-27 US US08/284,687 patent/US5631235A/en not_active Expired - Fee Related
-
1994
- 1994-09-01 FI FI944015A patent/FI107537B/fi active
-
1997
- 1997-12-16 GR GR970403321T patent/GR3025672T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0636136A1 (en) | 1995-02-01 |
| CA2131373C (en) | 1999-01-26 |
| ATE159725T1 (de) | 1997-11-15 |
| CA2131373A1 (en) | 1993-09-16 |
| WO1993018048A1 (en) | 1993-09-16 |
| DK0636136T3 (da) | 1997-12-22 |
| DE69314947D1 (de) | 1997-12-04 |
| FI944015A0 (fi) | 1994-09-01 |
| GR3025672T3 (en) | 1998-03-31 |
| DE69314947T2 (de) | 1998-03-05 |
| FI944015L (fi) | 1994-09-01 |
| FI107537B (fi) | 2001-08-31 |
| US5631235A (en) | 1997-05-20 |
| JPH07500350A (ja) | 1995-01-12 |
| JP2562001B2 (ja) | 1996-12-11 |
| EP0636136B1 (en) | 1997-10-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG2A | Definitive protection |
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