ATE163850T1 - Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen - Google Patents

Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Info

Publication number
ATE163850T1
ATE163850T1 AT93909884T AT93909884T ATE163850T1 AT E163850 T1 ATE163850 T1 AT E163850T1 AT 93909884 T AT93909884 T AT 93909884T AT 93909884 T AT93909884 T AT 93909884T AT E163850 T1 ATE163850 T1 AT E163850T1
Authority
AT
Austria
Prior art keywords
pct
rectal administration
agonistic
pharmaceutical compositions
sec
Prior art date
Application number
AT93909884T
Other languages
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Wellcome Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Lab filed Critical Glaxo Wellcome Lab
Application granted granted Critical
Publication of ATE163850T1 publication Critical patent/ATE163850T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
AT93909884T 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen ATE163850T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions

Publications (1)

Publication Number Publication Date
ATE163850T1 true ATE163850T1 (de) 1998-03-15

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93909884T ATE163850T1 (de) 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Country Status (33)

Country Link
US (1) US5705506A (de)
EP (1) EP0639072B1 (de)
JP (1) JPH07506570A (de)
KR (1) KR100253111B1 (de)
AT (1) ATE163850T1 (de)
AU (1) AU670083B2 (de)
BE (1) BE1007024A5 (de)
BG (1) BG62120B1 (de)
BR (1) BR1100108A (de)
CA (1) CA2135179C (de)
CH (1) CH685920A5 (de)
CY (1) CY2039B1 (de)
CZ (1) CZ283512B6 (de)
DE (1) DE69317418T2 (de)
ES (1) ES2113533T3 (de)
FR (1) FR2690847B1 (de)
GB (2) GB9209882D0 (de)
GR (1) GR3026584T3 (de)
HK (1) HK95697A (de)
HU (2) HU227338B1 (de)
IE (1) IE75203B1 (de)
IL (1) IL105468A (de)
IT (1) IT1261471B (de)
NO (1) NO306700B1 (de)
NZ (1) NZ252132A (de)
OA (1) OA10109A (de)
RO (1) RO112993B1 (de)
RU (1) RU2118527C1 (de)
SG (1) SG46649A1 (de)
TW (1) TW231970B (de)
UA (1) UA37206C2 (de)
WO (1) WO1993021916A1 (de)
ZA (1) ZA933178B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997044062A1 (en) * 1996-05-23 1997-11-27 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
PT2198858E (pt) * 1998-03-26 2011-09-01 Astellas Pharma Inc Composição farmacêutica de libertação constante que contém um macrólido como o tacrolimus
AU3731400A (en) * 1999-03-05 2000-09-21 Trustees Of University Technology Corporation, The Methods and compositions useful in inhibiting apoptosis
AR056690A1 (es) * 2005-10-14 2007-10-17 Athersys Inc Derivados de indol como inhibidores de indol como inhibidores del receptor 3 de histamina para el tartamiento de trastornos del sueno y cognitivos obesidad y otros trastornos de snc
JP2010522135A (ja) 2006-10-09 2010-07-01 チャールストン ラボラトリーズ，インコーポレイテッド 医薬組成物
JP5714910B2 (ja) 2008-01-09 2015-05-07 チャールストン ラボラトリーズ，インコーポレイテッド 薬学的組成物
EP3311667A1 (de) 2009-07-08 2018-04-25 Charleston Laboratories, Inc. Pharmazeutische zusammensetzungen
KR101825972B1 (ko) 2010-10-15 2018-02-06 콘테라 파르마 에이피에스 운동 장애 치료를 위한 세로토닌 수용체 작용제의 조합
PT2838517T (pt) 2012-04-18 2018-01-04 Contera Pharma Aps Formulação farmacêutica disponível sob forma oral adequada para a melhoria da gestão dos distúrbios da mobilidade
JP2019507181A (ja) 2016-03-04 2019-03-14 チャールストン ラボラトリーズ，インコーポレイテッド 医薬組成物
CA3030089C (en) 2016-07-11 2024-04-23 Contera Pharma Aps Pulsatile drug delivery system for treating morning akinesia

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1171450B (it) * 1980-08-12 1987-06-10 Glaxo Group Ltd Composti eterociclici indolici, procedimento per produrli e composizioni farmaceutiche che li contengono
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
HU196752B (en) * 1983-12-06 1989-01-30 Glaxo Group Ltd Process for production of medical compositions containing indole-derivatives and these compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
IT1181741B (it) * 1984-12-04 1987-09-30 Glaxo Group Ltd Derivati di indolo,procedimento per prepararli e composizioni farmaceutiche che li contengono
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
US4833153A (en) * 1985-11-08 1989-05-23 Glaxo Group Limited Indole derivatives
DK172696B1 (da) * 1987-08-13 1999-05-31 Glaxo Group Ltd Indolderivater, fremgangsmåde til fremstilling deraf og farmaceutiske præparater indeholdende forbindelserne
KR100215627B1 (ko) * 1990-06-07 1999-08-16 레슬리 제인 에드워즈 치료용 헤테로사이클 화합물

Also Published As

Publication number Publication date
SG46649A1 (en) 1998-02-20
CY2039B1 (en) 1998-04-30
HU227338B1 (en) 2011-04-28
CA2135179A1 (en) 1993-11-11
IE75203B1 (en) 1997-08-27
NO944214L (no) 1994-11-07
AU4064093A (en) 1993-11-29
ES2113533T3 (es) 1998-05-01
NO944214D0 (no) 1994-11-04
ITRM930286A0 (it) 1993-05-06
IL105468A0 (en) 1993-08-18
GB9209882D0 (en) 1992-06-24
OA10109A (en) 1996-12-18
DE69317418D1 (de) 1998-04-16
CA2135179C (en) 2000-12-05
GR3026584T3 (en) 1998-07-31
WO1993021916A1 (en) 1993-11-11
UA37206C2 (uk) 2001-05-15
US5705506A (en) 1998-01-06
HK95697A (en) 1997-08-08
JPH07506570A (ja) 1995-07-20
BE1007024A5 (fr) 1995-02-21
AU670083B2 (en) 1996-07-04
FR2690847A1 (fr) 1993-11-12
DE69317418T2 (de) 1998-07-30
BG99167A (bg) 1995-06-30
EP0639072A1 (de) 1995-02-22
RO112993B1 (ro) 1998-03-30
KR100253111B1 (en) 2000-07-01
NO306700B1 (no) 1999-12-13
EP0639072B1 (de) 1998-03-11
GB2266665A (en) 1993-11-10
IT1261471B (it) 1996-05-23
BR1100108A (pt) 1999-12-07
FR2690847B1 (fr) 1995-06-09
HU211638A9 (en) 1995-12-28
IE930339A1 (en) 1993-11-17
TW231970B (de) 1994-10-11
IL105468A (en) 1998-09-24
ITRM930286A1 (it) 1994-11-06
HUT71418A (en) 1995-11-28
CZ283512B6 (cs) 1998-04-15
RU2118527C1 (ru) 1998-09-10
BG62120B1 (bg) 1999-03-31
GB9309209D0 (en) 1993-06-16
CZ272394A3 (en) 1995-10-18
CH685920A5 (fr) 1995-11-15
NZ252132A (en) 1996-09-25
GB2266665B (en) 1996-05-22
ZA933178B (en) 1994-01-10

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