ATE167057T1 - Sublinguales oder bukkales arzneimittel - Google Patents

Sublinguales oder bukkales arzneimittel

Info

Publication number
ATE167057T1
ATE167057T1 AT95912188T AT95912188T ATE167057T1 AT E167057 T1 ATE167057 T1 AT E167057T1 AT 95912188 T AT95912188 T AT 95912188T AT 95912188 T AT95912188 T AT 95912188T AT E167057 T1 ATE167057 T1 AT E167057T1
Authority
AT
Austria
Prior art keywords
sublingual
buccal
pct
medicinal product
sec
Prior art date
Application number
AT95912188T
Other languages
English (en)
Inventor
Leonardus Petrus C Delbressine
Johannes Hubertus Wieringa
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE167057(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Application granted granted Critical
Publication of ATE167057T1 publication Critical patent/ATE167057T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT95912188T 1994-03-02 1995-03-01 Sublinguales oder bukkales arzneimittel ATE167057T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02

Publications (1)

Publication Number Publication Date
ATE167057T1 true ATE167057T1 (de) 1998-06-15

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95912188T ATE167057T1 (de) 1994-03-02 1995-03-01 Sublinguales oder bukkales arzneimittel

Country Status (23)

Country Link
US (1) US5763476A (de)
EP (1) EP0746317B1 (de)
JP (2) JP4099224B2 (de)
KR (1) KR100330942B1 (de)
CN (1) CN1079670C (de)
AT (1) ATE167057T1 (de)
AU (1) AU692530B2 (de)
BR (2) BR9506924A (de)
CA (1) CA2182981C (de)
CZ (1) CZ284633B6 (de)
DE (2) DE122010000050I2 (de)
DK (1) DK0746317T3 (de)
ES (1) ES2118584T3 (de)
FI (1) FI117923B (de)
FR (1) FR10C0056I2 (de)
HK (1) HK1008417A1 (de)
HU (1) HU225051B1 (de)
LU (1) LU91751I2 (de)
NO (2) NO308772B1 (de)
NZ (1) NZ282394A (de)
PL (1) PL180465B1 (de)
RU (1) RU2139051C1 (de)
WO (1) WO1995023600A1 (de)

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US7276246B2 (en) * 2003-05-09 2007-10-02 Cephalon, Inc. Dissolvable backing layer for use with a transmucosal delivery device
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TWI327915B (en) * 2003-06-12 2010-08-01 Organon Nv Pharmaceutical composition comprising antipsychotic agent and use of the antipsychotic agent for treating patients with overweight
BRPI0414321B8 (pt) * 2003-09-22 2021-06-22 Baxter Healthcare Sa esterilização à alta pressão para esterilização final de preparações farmacêuticas e produtos médicos
WO2005107808A2 (en) * 2004-05-11 2005-11-17 Pfizer Products Inc. Combination of atypical antipsychotics and 5-ht1b receptor antagonists
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AU2006231281B2 (en) 2005-04-07 2011-04-28 Msd Oss B.V. Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
US7741358B2 (en) * 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
US7875729B2 (en) 2007-01-05 2011-01-25 Synthon Bv Process for making asenapine
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JP2011526881A (ja) * 2008-06-25 2011-10-20 ファイザー・インク ジアリール化合物およびそれらの使用
WO2010127674A1 (en) * 2009-05-06 2010-11-11 Sunin K/S Transdermal compositions of asenapine for the treatment of psychiatric disorders
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EP2598496B1 (de) 2010-07-29 2014-03-19 Laboratorios Lesvi, S.L. Neuartiges verfahren zur herstellung von asenapin
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Also Published As

Publication number Publication date
NO308772B1 (no) 2000-10-30
BR1100625A (pt) 1999-12-28
BR9506924A (pt) 1997-09-30
HU9602383D0 (en) 1996-10-28
KR100330942B1 (ko) 2002-11-16
JPH09509674A (ja) 1997-09-30
MX9603713A (es) 1997-12-31
FI117923B (fi) 2007-04-30
PL180465B1 (pl) 2001-02-28
NO2010024I1 (no) 2011-01-03
WO1995023600A1 (en) 1995-09-08
HU225051B1 (en) 2006-05-29
HUT76319A (en) 1997-08-28
EP0746317B1 (de) 1998-06-10
NO2010024I2 (no) 2012-04-10
PL316080A1 (en) 1996-12-23
LU91751I2 (fr) 2011-01-04
ES2118584T3 (es) 1998-09-16
DE122010000050I1 (de) 2011-05-05
FR10C0056I1 (de) 2011-01-28
FR10C0056I2 (de) 2011-11-25
JP4099224B2 (ja) 2008-06-11
FI963398A0 (fi) 1996-08-30
DE122010000050I2 (de) 2011-07-21
CA2182981C (en) 2006-10-17
HK1008417A1 (en) 1999-05-07
NO963639L (no) 1996-10-30
AU1947895A (en) 1995-09-18
CN1079670C (zh) 2002-02-27
DK0746317T3 (da) 1999-03-22
CN1143320A (zh) 1997-02-19
DE69502939T2 (de) 1998-10-22
FI963398L (fi) 1996-08-30
AU692530B2 (en) 1998-06-11
US5763476A (en) 1998-06-09
DE69502939D1 (de) 1998-07-16
RU2139051C1 (ru) 1999-10-10
JP4616810B2 (ja) 2011-01-19
CZ254196A3 (en) 1997-10-15
EP0746317A1 (de) 1996-12-11
NZ282394A (en) 1997-12-19
NO963639D0 (no) 1996-08-30
JP2006342178A (ja) 2006-12-21
CA2182981A1 (en) 1995-09-08
CZ284633B6 (cs) 1999-01-13

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