LU91751I2 - Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) - Google Patents

Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Info

Publication number
LU91751I2
LU91751I2 LU91751C LU91751C LU91751I2 LU 91751 I2 LU91751 I2 LU 91751I2 LU 91751 C LU91751 C LU 91751C LU 91751 C LU91751 C LU 91751C LU 91751 I2 LU91751 I2 LU 91751I2
Authority
LU
Luxembourg
Prior art keywords
pharmaceutically acceptable
pct
sublingual
asenapin
sycrest
Prior art date
Application number
LU91751C
Other languages
English (en)
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU91751(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Nv filed Critical Organon Nv
Publication of LU91751I2 publication Critical patent/LU91751I2/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LU91751C 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) LU91751I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02
EP95912188A EP0746317B1 (fr) 1994-03-02 1995-03-01 Composition pharmaceutique sublinguale ou buccale
PCT/EP1995/000765 WO1995023600A1 (fr) 1994-03-02 1995-03-01 Composition pharmaceutique sublinguale ou buccale

Publications (1)

Publication Number Publication Date
LU91751I2 true LU91751I2 (fr) 2011-01-04

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91751C LU91751I2 (fr) 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Country Status (23)

Country Link
US (1) US5763476A (fr)
EP (1) EP0746317B1 (fr)
JP (2) JP4099224B2 (fr)
KR (1) KR100330942B1 (fr)
CN (1) CN1079670C (fr)
AT (1) ATE167057T1 (fr)
AU (1) AU692530B2 (fr)
BR (2) BR9506924A (fr)
CA (1) CA2182981C (fr)
CZ (1) CZ284633B6 (fr)
DE (2) DE122010000050I2 (fr)
DK (1) DK0746317T3 (fr)
ES (1) ES2118584T3 (fr)
FI (1) FI117923B (fr)
FR (1) FR10C0056I2 (fr)
HK (1) HK1008417A1 (fr)
HU (1) HU225051B1 (fr)
LU (1) LU91751I2 (fr)
NO (2) NO308772B1 (fr)
NZ (1) NZ282394A (fr)
PL (1) PL180465B1 (fr)
RU (1) RU2139051C1 (fr)
WO (1) WO1995023600A1 (fr)

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WO1999032108A1 (fr) * 1997-12-19 1999-07-01 Akzo Nobel N.V. Traitement pour la depression
WO2003068604A1 (fr) * 2002-02-13 2003-08-21 Weibel Michael K Forme posologique medicamenteuse et procede de fabrication
US7306812B2 (en) 2003-05-09 2007-12-11 Cephalon, Inc. Dissolvable backing layer for use with a transmucosal delivery device
US7276246B2 (en) * 2003-05-09 2007-10-02 Cephalon, Inc. Dissolvable backing layer for use with a transmucosal delivery device
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TWI327915B (en) * 2003-06-12 2010-08-01 Organon Nv Pharmaceutical composition comprising antipsychotic agent and use of the antipsychotic agent for treating patients with overweight
BRPI0414321B8 (pt) * 2003-09-22 2021-06-22 Baxter Healthcare Sa esterilização à alta pressão para esterilização final de preparações farmacêuticas e produtos médicos
WO2005107808A2 (fr) * 2004-05-11 2005-11-17 Pfizer Products Inc. Combinaison d'antipsychotiques atypiques et d'antagonistes du recepteur de 5-ht1b
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US7872147B2 (en) 2005-04-07 2011-01-18 N. V. Organon Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
AU2006231281B2 (en) 2005-04-07 2011-04-28 Msd Oss B.V. Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
US7741358B2 (en) * 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
US7875729B2 (en) 2007-01-05 2011-01-25 Synthon Bv Process for making asenapine
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JP2011526881A (ja) * 2008-06-25 2011-10-20 ファイザー・インク ジアリール化合物およびそれらの使用
WO2010127674A1 (fr) * 2009-05-06 2010-11-11 Sunin K/S Compositions transdermiques à base d'asénapine pour le traitement de troubles psychiatriques
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WO2012123325A1 (fr) 2011-03-11 2012-09-20 Medichem S.A. Nouvelles formes cristallines du sel de trans-5-chloro-2-méthyl-2,3,3a,12b-tétrahydro-1h-dibenzo[2,3:6,7] oxépino[4,5-c]pyrrole avec l'acide maléique
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Also Published As

Publication number Publication date
NO308772B1 (no) 2000-10-30
BR1100625A (pt) 1999-12-28
BR9506924A (pt) 1997-09-30
HU9602383D0 (en) 1996-10-28
KR100330942B1 (ko) 2002-11-16
JPH09509674A (ja) 1997-09-30
MX9603713A (es) 1997-12-31
FI117923B (fi) 2007-04-30
PL180465B1 (pl) 2001-02-28
NO2010024I1 (no) 2011-01-03
WO1995023600A1 (fr) 1995-09-08
HU225051B1 (en) 2006-05-29
HUT76319A (en) 1997-08-28
EP0746317B1 (fr) 1998-06-10
NO2010024I2 (no) 2012-04-10
PL316080A1 (en) 1996-12-23
ES2118584T3 (es) 1998-09-16
DE122010000050I1 (de) 2011-05-05
FR10C0056I1 (fr) 2011-01-28
FR10C0056I2 (fr) 2011-11-25
JP4099224B2 (ja) 2008-06-11
FI963398A0 (fi) 1996-08-30
DE122010000050I2 (de) 2011-07-21
CA2182981C (fr) 2006-10-17
HK1008417A1 (en) 1999-05-07
NO963639L (no) 1996-10-30
AU1947895A (en) 1995-09-18
CN1079670C (zh) 2002-02-27
DK0746317T3 (da) 1999-03-22
CN1143320A (zh) 1997-02-19
DE69502939T2 (de) 1998-10-22
FI963398L (fi) 1996-08-30
AU692530B2 (en) 1998-06-11
US5763476A (en) 1998-06-09
DE69502939D1 (de) 1998-07-16
RU2139051C1 (ru) 1999-10-10
ATE167057T1 (de) 1998-06-15
JP4616810B2 (ja) 2011-01-19
CZ254196A3 (en) 1997-10-15
EP0746317A1 (fr) 1996-12-11
NZ282394A (en) 1997-12-19
NO963639D0 (no) 1996-08-30
JP2006342178A (ja) 2006-12-21
CA2182981A1 (fr) 1995-09-08
CZ284633B6 (cs) 1999-01-13

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