LU91751I2 - Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) - Google Patents

Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Info

Publication number
LU91751I2
LU91751I2 LU91751C LU91751C LU91751I2 LU 91751 I2 LU91751 I2 LU 91751I2 LU 91751 C LU91751 C LU 91751C LU 91751 C LU91751 C LU 91751C LU 91751 I2 LU91751 I2 LU 91751I2
Authority
LU
Luxembourg
Prior art keywords
pharmaceutically acceptable
pct
sublingual
asenapin
sycrest
Prior art date
Application number
LU91751C
Other languages
English (en)
Original Assignee
Organon Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU91751(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Nv filed Critical Organon Nv
Publication of LU91751I2 publication Critical patent/LU91751I2/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
LU91751C 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®) LU91751I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02
EP95912188A EP0746317B1 (fr) 1994-03-02 1995-03-01 Composition pharmaceutique sublinguale ou buccale
PCT/EP1995/000765 WO1995023600A1 (fr) 1994-03-02 1995-03-01 Composition pharmaceutique sublinguale ou buccale

Publications (1)

Publication Number Publication Date
LU91751I2 true LU91751I2 (fr) 2011-01-04

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
LU91751C LU91751I2 (fr) 1994-03-02 2010-11-04 Asenapin et ses dérivés pharmaceutiquement acceptables (SYCREST®)

Country Status (23)

Country Link
US (1) US5763476A (fr)
EP (1) EP0746317B1 (fr)
JP (2) JP4099224B2 (fr)
KR (1) KR100330942B1 (fr)
CN (1) CN1079670C (fr)
AT (1) ATE167057T1 (fr)
AU (1) AU692530B2 (fr)
BR (2) BR9506924A (fr)
CA (1) CA2182981C (fr)
CZ (1) CZ284633B6 (fr)
DE (2) DE69502939T2 (fr)
DK (1) DK0746317T3 (fr)
ES (1) ES2118584T3 (fr)
FI (1) FI117923B (fr)
FR (1) FR10C0056I2 (fr)
HK (1) HK1008417A1 (fr)
HU (1) HU225051B1 (fr)
LU (1) LU91751I2 (fr)
NO (2) NO308772B1 (fr)
NZ (1) NZ282394A (fr)
PL (1) PL180465B1 (fr)
RU (1) RU2139051C1 (fr)
WO (1) WO1995023600A1 (fr)

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TWI327915B (en) * 2003-06-12 2010-08-01 Organon Nv Pharmaceutical composition comprising antipsychotic agent and use of the antipsychotic agent for treating patients with overweight
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US7872147B2 (en) 2005-04-07 2011-01-18 N. V. Organon Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole
DK1710241T3 (da) 2005-04-07 2010-03-01 Organon Nv Intermediatforbindelser til fremstilling af trans-5-chlor-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrol
EP1710245B1 (fr) * 2005-04-07 2007-08-22 N.V. Organon Forme cristalline du maleate d`asenapine
US7741358B2 (en) 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
US7875729B2 (en) 2007-01-05 2011-01-25 Synthon Bv Process for making asenapine
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WO2010127674A1 (fr) * 2009-05-06 2010-11-11 Sunin K/S Compositions transdermiques à base d'asénapine pour le traitement de troubles psychiatriques
MX2012000061A (es) 2009-06-24 2012-06-01 Msd Oss Bv Formulaciones inyectables que contienen asenapina, y metodo de tratamiento usando las mismas.
AR077429A1 (es) 2009-07-29 2011-08-24 Organon Nv Compuestos hidroxiasenapina sus derivados y composiciones farmaceuticas que comprenden los mismos
EP2582704A4 (fr) 2010-06-18 2014-04-02 Reddys Lab Ltd Dr Maléate d'asénapine
WO2012013766A1 (fr) 2010-07-29 2012-02-02 Laboratorios Lesvi, S.L. Nouveau procédé de synthèse de l'asénapine
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EP3034079B1 (fr) 2010-11-15 2018-01-10 Agenebio, Inc. Dérivés de pyridazine, compositions et méthodes de traitement d'une déficience cognitive
WO2012066565A2 (fr) 2010-11-16 2012-05-24 Cadila Healthcare Limited Maléate d'asénapine amorphe et forme cristalline et procédé pour leur préparation
EP2468750A1 (fr) 2010-12-13 2012-06-27 Chemo Ibérica, S.A. Formes polymorphiques de maléate d'asénapine et procédés de préparation
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ITMI20121810A1 (it) 2012-10-24 2014-04-25 Chemo Iberica Sa Poliformi di maleato di asenapina e processo per la loro preparazione
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WO2019002204A1 (fr) 2017-06-26 2019-01-03 Lts Lohmann Therapie-Systeme Ag Système thérapeutique transdermique contenant de l'asénapine et un polymère hybride acrylique de type silicone
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CN112040940A (zh) 2018-03-23 2020-12-04 细胞内治疗公司 有机化合物
CN112601749B (zh) 2018-06-19 2024-03-26 艾吉因生物股份有限公司 用于治疗认知损害的苯并二氮杂环庚三烯衍生物，组合物和方法
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WO2020047408A1 (fr) 2018-08-31 2020-03-05 Intra-Cellular Therapies, Inc. Nouvelles méthodes
BR112021003655A2 (pt) 2018-08-31 2021-05-18 Intra-Cellular Therapies, Inc. métodos novos
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US12414948B2 (en) 2022-05-18 2025-09-16 Intra-Cellular Therapies, Inc. Methods
CN120584115A (zh) 2022-08-19 2025-09-02 艾吉因生物股份有限公司 苯并氮杂䓬衍生物、组合物和用于治疗认知损害的方法

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Also Published As

Publication number Publication date
JP4616810B2 (ja) 2011-01-19
WO1995023600A1 (fr) 1995-09-08
ATE167057T1 (de) 1998-06-15
CA2182981A1 (fr) 1995-09-08
RU2139051C1 (ru) 1999-10-10
NO308772B1 (no) 2000-10-30
NZ282394A (en) 1997-12-19
EP0746317B1 (fr) 1998-06-10
CN1079670C (zh) 2002-02-27
KR100330942B1 (ko) 2002-11-16
FI117923B (fi) 2007-04-30
JP2006342178A (ja) 2006-12-21
PL180465B1 (pl) 2001-02-28
BR1100625A (pt) 1999-12-28
PL316080A1 (en) 1996-12-23
CA2182981C (fr) 2006-10-17
HUT76319A (en) 1997-08-28
CN1143320A (zh) 1997-02-19
FI963398L (fi) 1996-08-30
DE69502939T2 (de) 1998-10-22
CZ284633B6 (cs) 1999-01-13
AU692530B2 (en) 1998-06-11
US5763476A (en) 1998-06-09
HU225051B1 (en) 2006-05-29
CZ254196A3 (en) 1997-10-15
JP4099224B2 (ja) 2008-06-11
FI963398A0 (fi) 1996-08-30
DE69502939D1 (de) 1998-07-16
JPH09509674A (ja) 1997-09-30
HU9602383D0 (en) 1996-10-28
DE122010000050I2 (de) 2011-07-21
DK0746317T3 (da) 1999-03-22
NO963639D0 (no) 1996-08-30
AU1947895A (en) 1995-09-18
HK1008417A1 (en) 1999-05-07
NO963639L (no) 1996-10-30
DE122010000050I1 (de) 2011-05-05
ES2118584T3 (es) 1998-09-16
FR10C0056I2 (fr) 2011-11-25
NO2010024I1 (no) 2011-01-03
BR9506924A (pt) 1997-09-30
EP0746317A1 (fr) 1996-12-11
FR10C0056I1 (fr) 2011-01-28
NO2010024I2 (no) 2012-04-10
MX9603713A (es) 1997-12-31

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