ATE175413T1 - Substituierte pyridopyrimidine als antihypertensiva - Google Patents

Substituierte pyridopyrimidine als antihypertensiva

Info

Publication number
ATE175413T1
ATE175413T1 AT94301881T AT94301881T ATE175413T1 AT E175413 T1 ATE175413 T1 AT E175413T1 AT 94301881 T AT94301881 T AT 94301881T AT 94301881 T AT94301881 T AT 94301881T AT E175413 T1 ATE175413 T1 AT E175413T1
Authority
AT
Austria
Prior art keywords
c6alkyl
hydroxy
carboxy
chem
compounds
Prior art date
Application number
AT94301881T
Other languages
English (en)
Inventor
John Watson Ellingboe
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/179,461 external-priority patent/US5466692A/en
Application filed by American Home Prod filed Critical American Home Prod
Application granted granted Critical
Publication of ATE175413T1 publication Critical patent/ATE175413T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT94301881T 1993-03-24 1994-03-16 Substituierte pyridopyrimidine als antihypertensiva ATE175413T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3661593A 1993-03-24 1993-03-24
US08/179,461 US5466692A (en) 1993-03-24 1994-01-10 Substituted pyridopyrimidines and antihypertensives

Publications (1)

Publication Number Publication Date
ATE175413T1 true ATE175413T1 (de) 1999-01-15

Family

ID=26713326

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94301881T ATE175413T1 (de) 1993-03-24 1994-03-16 Substituierte pyridopyrimidine als antihypertensiva

Country Status (16)

Country Link
EP (2) EP0618207B1 (de)
JP (1) JPH06321945A (de)
AT (1) ATE175413T1 (de)
AU (1) AU669966B2 (de)
BR (1) BR9401261A (de)
CA (1) CA2119692A1 (de)
DE (1) DE69415706T2 (de)
DK (1) DK0618207T3 (de)
ES (1) ES2126061T3 (de)
FI (1) FI108135B (de)
GR (1) GR3029879T3 (de)
HU (1) HU222240B1 (de)
LV (1) LV12261B (de)
NZ (1) NZ260164A (de)
PH (1) PH30373A (de)
SG (1) SG47714A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUP0104634A3 (en) 1998-07-06 2002-11-28 Bristol Myers Squibb Co Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
KR101530019B1 (ko) * 2007-06-07 2015-06-18 시그마타우 인두스트리에 파르마슈티케 리우니테 에스.피.에이. 혈관성형술 또는 동맥내막절제술 후 재협착 및 장기 섬유증으로 인한 질환의 치료에 유용한 5베타, 14베타-안드로스테인 유도체

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US521797A (en) * 1894-06-26 Half to john m
BG94957A (bg) * 1990-08-10 1993-12-24 Ciba - Geigy Ag Пиримидинови производни и средство за борба срещу вредители по растенията
US5290780A (en) * 1991-01-30 1994-03-01 American Cyanamid Co. Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
IL100917A0 (en) * 1991-02-16 1992-11-15 Fisons Plc Pyridinone and pyrimidinone derivatives,their preparation and pharmaceutical compositions containing them
IL101860A0 (en) * 1991-05-31 1992-12-30 Ici Plc Heterocyclic derivatives
TW226375B (de) * 1991-10-24 1994-07-11 American Home Prod
US5149699A (en) * 1991-10-24 1992-09-22 American Home Products Corporation Substituted pyridopyrimidines useful as antgiotensin II antagonists
GB9125842D0 (en) * 1991-12-04 1992-02-05 Ici Plc Heterocyclic derivatives

Also Published As

Publication number Publication date
GR3029879T3 (en) 1999-07-30
NZ260164A (en) 1996-02-27
AU669966B2 (en) 1996-06-27
LV12261B (en) 1999-09-20
HK1011358A1 (en) 1999-07-09
HU9400822D0 (en) 1994-06-28
EP0618207A1 (de) 1994-10-05
EP0618207B1 (de) 1999-01-07
FI941309A0 (fi) 1994-03-21
PH30373A (en) 1997-04-02
CA2119692A1 (en) 1994-09-25
ES2126061T3 (es) 1999-03-16
LV12261A (lv) 1999-04-20
DK0618207T3 (da) 1999-08-30
HUT66964A (en) 1995-01-30
DE69415706D1 (de) 1999-02-18
SG47714A1 (en) 1998-04-17
DE69415706T2 (de) 1999-05-20
FI108135B (fi) 2001-11-30
HU222240B1 (hu) 2003-05-28
FI941309L (fi) 1994-09-25
EP0863143A1 (de) 1998-09-09
JPH06321945A (ja) 1994-11-22
BR9401261A (pt) 1994-11-22
AU5799794A (en) 1994-09-29

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee