ATE197453T1 - Imidazol-, triazol- und tetrazolderivate - Google Patents

Imidazol-, triazol- und tetrazolderivate

Info

Publication number
ATE197453T1
ATE197453T1 AT93907945T AT93907945T ATE197453T1 AT E197453 T1 ATE197453 T1 AT E197453T1 AT 93907945 T AT93907945 T AT 93907945T AT 93907945 T AT93907945 T AT 93907945T AT E197453 T1 ATE197453 T1 AT E197453T1
Authority
AT
Austria
Prior art keywords
pct
triazole
imidazole
tetrazole derivatives
receptors
Prior art date
Application number
AT93907945T
Other languages
English (en)
Inventor
Pineiro Jose Luis Castro
Victor Giulio Matassa
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Application granted granted Critical
Publication of ATE197453T1 publication Critical patent/ATE197453T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Resins (AREA)
  • Paints Or Removers (AREA)
  • Lubricants (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
AT93907945T 1992-04-03 1993-03-29 Imidazol-, triazol- und tetrazolderivate ATE197453T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929207396A GB9207396D0 (en) 1992-04-03 1992-04-03 Therapeutic agents
PCT/GB1993/000652 WO1993020066A1 (en) 1992-04-03 1993-03-29 Imidazole, triazole and tetrazole derivatives

Publications (1)

Publication Number Publication Date
ATE197453T1 true ATE197453T1 (de) 2000-11-11

Family

ID=10713456

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93907945T ATE197453T1 (de) 1992-04-03 1993-03-29 Imidazol-, triazol- und tetrazolderivate

Country Status (10)

Country Link
US (1) US5607957A (de)
EP (1) EP0637307B1 (de)
JP (1) JP3285581B2 (de)
AT (1) ATE197453T1 (de)
AU (1) AU675641B2 (de)
CA (1) CA2133076A1 (de)
DE (1) DE69329645T2 (de)
ES (1) ES2152948T3 (de)
GB (1) GB9207396D0 (de)
WO (1) WO1993020066A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9420529D0 (en) 1994-10-12 1994-11-30 Pfizer Ltd Indoles
US5484763A (en) * 1995-02-10 1996-01-16 American Cyanamid Company Substituted benzisoxazole and benzisothiazole herbicidal agents
JP2003510359A (ja) 1999-10-01 2003-03-18 スミスクライン・ビーチャム・コーポレイション 化合物および方法
WO2001087845A2 (en) * 2000-05-15 2001-11-22 Fujisawa Pharmaceutical Co., Ltd. N-containing heterocyclic compounds and their use as 5-ht antagonists
CA2508290C (en) 2002-12-20 2017-02-28 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
KR20150087400A (ko) 2012-11-20 2015-07-29 버텍스 파마슈티칼스 인코포레이티드 인돌아민 2,3-디옥시게나제의 억제제로서 유용한 화합물
JP7189155B2 (ja) 2017-05-17 2022-12-13 アーカス バイオサイエンシズ インコーポレイティド 癌関連障害の治療のためのキナゾリン－ピラゾール誘導体
GB201801226D0 (en) 2018-01-25 2018-03-14 Redx Pharma Plc Modulators of Rho-associated protein kinase
MX2023009059A (es) 2021-02-02 2023-09-15 Liminal Biosciences Ltd Antagonistas de gpr84 y usos de estos.
JP2024527574A (ja) 2021-07-07 2024-07-25 テラン バイオサイエンシズ インコーポレイテッド Ｎ，ｎ－ジメチルトリプタミン及び関連する幻覚剤ならびにその使用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8505715L (sv) * 1984-12-04 1986-06-05 Glaxo Group Ltd Indolderivat
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
GB8724912D0 (en) * 1987-10-23 1987-11-25 Wellcome Found Indole derivatives
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions
IL96891A0 (en) * 1990-01-17 1992-03-29 Merck Sharp & Dohme Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
SI9111010B (sl) * 1990-06-07 2005-02-28 Astrazeneca Ab 3,5-disubstituirani indolni derivati kot "5-HT1-podobni" receptorski agonisti
EP0494774A1 (de) * 1991-01-11 1992-07-15 MERCK SHARP & DOHME LTD. Indazol-substituierte 5-Kettenglieder heteroaromatische Verbindungen
SK278998B6 (sk) * 1991-02-01 1998-05-06 Merck Sharp & Dohme Limited Deriváty imidazolu, triazolu a tetrazolu, spôsob i
CA2124206C (en) * 1991-11-25 2001-02-27 John Eugene Macor Indole derivatives

Also Published As

Publication number Publication date
AU3895693A (en) 1993-11-08
CA2133076A1 (en) 1993-10-14
DE69329645T2 (de) 2001-05-10
EP0637307B1 (de) 2000-11-08
WO1993020066A1 (en) 1993-10-14
DE69329645D1 (de) 2000-12-14
EP0637307A1 (de) 1995-02-08
JPH07505382A (ja) 1995-06-15
ES2152948T3 (es) 2001-02-16
AU675641B2 (en) 1997-02-13
JP3285581B2 (ja) 2002-05-27
US5607957A (en) 1997-03-04
GB9207396D0 (en) 1992-05-13

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties