ATE200223T1 - Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe - Google Patents

Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe

Info

Publication number: ATE200223T1
Authority: AT; Austria
Prior art keywords: sampangin; antimycobacterial; actives; antifungal; derivatives
Prior art date: 1991-06-14

Application number

AT92905142T

Other languages

English (en)

Inventor

Alice M Clark

Charles D Hufford

Shihchih Liu

Babajide O Oguntimein

John R Peterson

Jordan K Zjawiony

Original Assignee

Univ Mississippi

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-06-14

Filing date

1991-11-06

Publication date

2001-04-15

1991-11-06 Application filed by Univ Mississippi filed Critical Univ Mississippi

2001-04-15 Application granted granted Critical

2001-04-15 Publication of ATE200223T1 publication Critical patent/ATE200223T1/de

Links

BWQKHOMAOVUASZ-UHFFFAOYSA-N sampangine Chemical class C1=NC(C(=O)C=2C3=CC=CC=2)=C2C3=NC=CC2=C1 BWQKHOMAOVUASZ-UHFFFAOYSA-N 0.000 title abstract 3
230000000843 anti-fungal effect Effects 0.000 title 1
230000001355 anti-mycobacterial effect Effects 0.000 title 1
229940121375 antifungal agent Drugs 0.000 title 1
239000003926 antimycobacterial agent Substances 0.000 title 1
GVRYUHXXENMGEV-UHFFFAOYSA-N 4-methylbenzo[g]quinoline-5,10-dione Chemical compound O=C1C2=CC=CC=C2C(=O)C2=C1N=CC=C2C GVRYUHXXENMGEV-UHFFFAOYSA-N 0.000 abstract 2
206010017533 Fungal infection Diseases 0.000 abstract 1
206010062207 Mycobacterial infection Diseases 0.000 abstract 1
208000031888 Mycoses Diseases 0.000 abstract 1
230000002538 fungal effect Effects 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
208000027531 mycobacterial infectious disease Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/04—Ortho- or peri-condensed ring systems
- C07D221/06—Ring systems of three rings
- C07D221/08—Aza-anthracenes

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicines Containing Plant Substances (AREA)

AT92905142T 1991-06-14 1991-11-06 Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe ATE200223T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/715,776 US5227383A (en)	1991-06-14	1991-06-14	Compounds and compositions useful as antifungal and antimycobacterial agents
PCT/US1991/008319 WO1992022297A1 (en)	1991-06-14	1991-11-06	New compounds and compositions useful as antifungal and antimycobacterial agents

Publications (1)

Publication Number	Publication Date
ATE200223T1 true ATE200223T1 (de)	2001-04-15

Family

ID=24875436

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT92905142T ATE200223T1 (de)	1991-06-14	1991-11-06	Sampangin-derivate zur verwendung als antimykotische und antimykobakterielle wirkstoffe

Country Status (10)

Country	Link
US (2)	US5227383A (de)
EP (1)	EP0588796B1 (de)
JP (1)	JP3405540B2 (de)
AT (1)	ATE200223T1 (de)
CA (1)	CA2111338A1 (de)
DE (1)	DE69132575T2 (de)
DK (1)	DK0588796T3 (de)
ES (1)	ES2157899T3 (de)
GR (1)	GR3036159T3 (de)
WO (1)	WO1992022297A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4301424A1 (de) *	1993-01-20	1994-07-21	Basf Ag	Derivate des Azaanthrachinons und des Azaxanthons und diese enthaltende Herbizide und Pflanzenwachstumsregulatoren
US5476933A (en) *	1994-11-16	1995-12-19	State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University And The University Of Oregon	Azepine synthesis via a diels-alder reaction
US20040052868A1 (en)	2002-09-12	2004-03-18	William Asiedu	Composition treating for AIDS and associated conditions
AU2011219481B2 (en) *	2002-09-12	2012-09-20	Willfred-Ramix, Inc.	A composition for treating AIDS and associated conditions
JP4794136B2 (ja) *	2004-04-21	2011-10-19	阿蘇製薬株式会社	アクリジン誘導体
US7491721B2 (en) *	2004-05-12	2009-02-17	Lupin Limited	Antimycobacterial pharmaceutical composition
US20170112824A1 (en) *	2015-10-23	2017-04-27	Wright State University	Combination therapies for the treatment of fungal infections
CN106905317B (zh) *	2017-01-24	2019-03-22	广西师范大学	4-取代Sampangine生物碱衍生物及其合成方法和应用
KR20230010838A (ko) *	2018-06-18	2023-01-19	이엘씨 매니지먼트 엘엘씨	광안정화 화합물, 조성물, 및 방법
EP3806814A4 (de)	2018-06-18	2021-10-06	ELC Management LLC	Fotostabilierungsverbindungen, zusammensetzungen und verfahren
WO2019245877A1 (en)	2018-06-18	2019-12-26	Elc Management Llc	Photostabilizing compounds, compositions, and methods
KR102555304B1 (ko)	2018-06-18	2023-07-14	이엘씨 매니지먼트 엘엘씨	광안정화 화합물, 조성물, 및 방법
CN113461506A (zh) *	2021-06-23	2021-10-01	苏州求索生物科技有限公司	一种2-溴-1,4-萘并醌的制备工艺

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4080456A (en) *	1971-10-26	1978-03-21	Schering Aktiengesellschaft	Diacylapomorphines
AR204011A1 (es) *	1973-07-27	1975-11-12	Rhone Poulenc Sa	Procedimiento de preparacion de nuevos derivados de 7-h-indolizino(5,6,7-ij)isoquinoleina
JPS5337696A (en) *	1976-08-26	1978-04-06	Omnium Chimique Sa	Hexahydrocantinonee6 derivative
US4965272A (en) *	1988-07-14	1990-10-23	Hufford Charles D	Antimicrobial compound and compositions particularly effective against candida albicans
US5128344A (en) *	1990-11-06	1992-07-07	University Of Mississippi	Sampangine and derivatives useful as an antifungal agent

1991
- 1991-06-14 US US07/715,776 patent/US5227383A/en not_active Expired - Fee Related
- 1991-11-06 DK DK92905142T patent/DK0588796T3/da active
- 1991-11-06 WO PCT/US1991/008319 patent/WO1992022297A1/en not_active Ceased
- 1991-11-06 AT AT92905142T patent/ATE200223T1/de not_active IP Right Cessation
- 1991-11-06 JP JP50518192A patent/JP3405540B2/ja not_active Expired - Fee Related
- 1991-11-06 CA CA002111338A patent/CA2111338A1/en not_active Abandoned
- 1991-11-06 DE DE69132575T patent/DE69132575T2/de not_active Expired - Fee Related
- 1991-11-06 EP EP92905142A patent/EP0588796B1/de not_active Expired - Lifetime
- 1991-11-06 ES ES92905142T patent/ES2157899T3/es not_active Expired - Lifetime
1993
- 1993-07-12 US US08/090,594 patent/US5530004A/en not_active Expired - Lifetime
2001
- 2001-06-29 GR GR20010401010T patent/GR3036159T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
EP0588796A4 (en)	1994-09-14
GR3036159T3 (en)	2001-09-28
EP0588796A1 (de)	1994-03-30
JP3405540B2 (ja)	2003-05-12
EP0588796B1 (de)	2001-04-04
CA2111338A1 (en)	1992-12-23
ES2157899T3 (es)	2001-09-01
DE69132575T2 (de)	2001-10-18
US5530004A (en)	1996-06-25
DE69132575D1 (de)	2001-05-10
US5227383A (en)	1993-07-13
DK0588796T3 (da)	2001-05-07
WO1992022297A1 (en)	1992-12-23
JPH06508104A (ja)	1994-09-14

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Legal Events

Date	Code	Title	Description
2002-03-15	UEP	Publication of translation of european patent specification
2004-08-15	REN	Ceased due to non-payment of the annual fee