ATE203025T1 - Reverse-turnmimetika und damit zusammenhängendes verfahren - Google Patents

Reverse-turnmimetika und damit zusammenhängendes verfahren

Info

Publication number
ATE203025T1
ATE203025T1 AT96937733T AT96937733T ATE203025T1 AT E203025 T1 ATE203025 T1 AT E203025T1 AT 96937733 T AT96937733 T AT 96937733T AT 96937733 T AT96937733 T AT 96937733T AT E203025 T1 ATE203025 T1 AT E203025T1
Authority
AT
Austria
Prior art keywords
reverse
turn mimetics
related method
reverse turn
disclosed
Prior art date
Application number
AT96937733T
Other languages
English (en)
Inventor
Michael Kahn
Original Assignee
Molecumetics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Molecumetics Ltd filed Critical Molecumetics Ltd
Application granted granted Critical
Publication of ATE203025T1 publication Critical patent/ATE203025T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Peptides Or Proteins (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Toys (AREA)
  • Detergent Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT96937733T 1995-10-27 1996-10-24 Reverse-turnmimetika und damit zusammenhängendes verfahren ATE203025T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/549,007 US5929237A (en) 1995-10-27 1995-10-27 Reverse-turn mimetics and methods relating thereto
PCT/US1996/017053 WO1997015577A1 (en) 1995-10-27 1996-10-24 Reverse-turn mimetics and methods relating thereto

Publications (1)

Publication Number Publication Date
ATE203025T1 true ATE203025T1 (de) 2001-07-15

Family

ID=24191284

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96937733T ATE203025T1 (de) 1995-10-27 1996-10-24 Reverse-turnmimetika und damit zusammenhängendes verfahren

Country Status (10)

Country Link
US (1) US5929237A (de)
EP (1) EP0876371B1 (de)
JP (1) JPH11513986A (de)
KR (1) KR19990067102A (de)
AT (1) ATE203025T1 (de)
AU (1) AU719620B2 (de)
CA (1) CA2235138C (de)
DE (1) DE69613861T2 (de)
ES (1) ES2158360T3 (de)
WO (1) WO1997015577A1 (de)

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US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
EP2069791B1 (de) 2006-07-27 2012-01-25 University of Maryland, Baltimore Zellulärer rezeptor für antiproliferativen faktor
EP2155226A4 (de) * 2007-06-14 2010-07-28 Univ California Verbindungen zur hemmung der proteinaggregation und verfahren zu deren herstellung und verwendung
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US8343958B2 (en) 2008-02-29 2013-01-01 Mimetica Pty Ltd 3-aminoalkyl-1,4-diazepan-2-one melanocortin-5-receptor antagonists
US8377925B2 (en) 2008-02-29 2013-02-19 Mimetica Pty Ltd Methods of modulating the activity of the MC5 receptor and treatment of conditions related to this receptor
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WO2010033227A1 (en) * 2008-09-19 2010-03-25 Nektar Therapeutics Polymer conjugates of thymosin alpha 1 peptides
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WO2012115286A1 (en) 2011-02-25 2012-08-30 Prism Biolab Corporation Alpha helix mimetics and methods relating thereto
US9140698B2 (en) 2011-04-06 2015-09-22 The Board Of Regents Of The University Of Texas System Modulating bacterial MAM polypeptides in pathogenic disease
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US20130101664A1 (en) 2011-08-18 2013-04-25 Donald W. Kufe Muc1 ligand traps for use in treating cancers
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Also Published As

Publication number Publication date
AU719620B2 (en) 2000-05-11
DE69613861T2 (de) 2001-11-15
JPH11513986A (ja) 1999-11-30
AU7520596A (en) 1997-05-15
EP0876371A1 (de) 1998-11-11
US5929237A (en) 1999-07-27
DE69613861D1 (de) 2001-08-16
KR19990067102A (ko) 1999-08-16
EP0876371B1 (de) 2001-07-11
ES2158360T3 (es) 2001-09-01
WO1997015577A1 (en) 1997-05-01
CA2235138C (en) 2005-04-05
CA2235138A1 (en) 1997-05-01

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties