ATE207929T1 - Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene - Google Patents

Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Info

Publication number
ATE207929T1
ATE207929T1 AT95942689T AT95942689T ATE207929T1 AT E207929 T1 ATE207929 T1 AT E207929T1 AT 95942689 T AT95942689 T AT 95942689T AT 95942689 T AT95942689 T AT 95942689T AT E207929 T1 ATE207929 T1 AT E207929T1
Authority
AT
Austria
Prior art keywords
androan
antiandrogens
thioxo
aza
oxo
Prior art date
Application number
AT95942689T
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Ambrogio Magni
Vincenzo Olgiati
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of ATE207929T1 publication Critical patent/ATE207929T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT95942689T 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene ATE207929T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens

Publications (1)

Publication Number Publication Date
ATE207929T1 true ATE207929T1 (de) 2001-11-15

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95942689T ATE207929T1 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Country Status (10)

Country Link
US (1) US6147213A (de)
EP (1) EP0799239B1 (de)
AT (1) ATE207929T1 (de)
AU (1) AU4387296A (de)
DE (1) DE69523622T2 (de)
DK (1) DK0799239T3 (de)
ES (1) ES2163538T3 (de)
IT (1) IT1271325B (de)
PT (1) PT799239E (de)
WO (1) WO1996020210A2 (de)

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Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
JP2010510674A (ja) 2006-11-15 2010-04-02 エナジーツー・インコーポレイテッド 電気２重層キャパシタ装置
JP5456669B2 (ja) * 2007-05-03 2014-04-02 エール ユニヴァーシティ 局所活性「ソフト」抗アンドロゲン剤
KR101830879B1 (ko) 2009-07-01 2018-02-21 바스프 에스이 초고순도의 합성 탄소 물질
BR112012014092A2 (pt) * 2009-12-11 2016-07-05 Energ2 Technologies Inc materiais de carvão compreendendo um modificador eletroquímico.
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
WO2012045002A1 (en) 2010-09-30 2012-04-05 Energ2 Technologies, Inc. Enhanced packing of energy storage particles
EP2659498B1 (de) 2010-12-28 2020-07-22 Basf Se Kohlenstoffmaterialien mit verbessertem elektrochemischen eigenschaften
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
CN103947017B (zh) 2011-06-03 2017-11-17 巴斯福股份公司 用于混合能量存储装置中的碳‑铅共混物
US9409777B2 (en) 2012-02-09 2016-08-09 Basf Se Preparation of polymeric resins and carbon materials
CN105190948B (zh) 2013-03-14 2019-04-26 14族科技公司 包含锂合金化的电化学改性剂的复合碳材料
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
JP6665121B2 (ja) 2014-03-14 2020-03-13 グループ１４・テクノロジーズ・インコーポレイテッドＧｒｏｕｐ１４ Ｔｅｃｈｎｏｌｏｇｉｅｓ， Ｉｎｃ． 無溶媒中におけるゾル−ゲル重合のための新規方法、及びゾル−ゲル重合由来の可変炭素構造の作製
US20190097222A1 (en) 2015-08-14 2019-03-28 Energ2 Technologies, Inc. Composites of porous nano-featured silicon materials and carbon materials
EP4286355A3 (de) 2015-08-28 2024-05-01 Group14 Technologies, Inc. Neuartige materialien mit extrem langlebiger einlagerung von lithium und herstellungsverfahren dafür
US11611071B2 (en) 2017-03-09 2023-03-21 Group14 Technologies, Inc. Decomposition of silicon-containing precursors on porous scaffold materials
WO2022035879A1 (en) 2020-08-10 2022-02-17 Group14 Technologies, Inc. Vibro-thermally assisted chemical vapor infiltration
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
KR102600078B1 (ko) 2020-08-18 2023-11-08 그룹14 테크놀로지스, 인코포레이티드 규소-탄소 복합체 재료의 제조
CA3195890A1 (en) 2020-09-30 2022-04-07 Group14 Technologies, Inc. Methods of passivation to control oxygen content and reactivity of silicon-carbon composite materials

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
EP0799239A2 (de) 1997-10-08
PT799239E (pt) 2002-02-28
IT1271325B (it) 1997-05-27
US6147213A (en) 2000-11-14
DK0799239T3 (da) 2001-12-10
ITMI942626A1 (it) 1996-06-23
DE69523622D1 (de) 2001-12-06
EP0799239B1 (de) 2001-10-31
ITMI942626A0 (it) 1994-12-23
WO1996020210A2 (en) 1996-07-04
DE69523622T2 (de) 2002-05-29
ES2163538T3 (es) 2002-02-01
WO1996020210A3 (en) 1996-09-06
AU4387296A (en) 1996-07-19

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UEP Publication of translation of european patent specification