ATE207929T1 - Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene - Google Patents

Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Info

Publication number
ATE207929T1
ATE207929T1 AT95942689T AT95942689T ATE207929T1 AT E207929 T1 ATE207929 T1 AT E207929T1 AT 95942689 T AT95942689 T AT 95942689T AT 95942689 T AT95942689 T AT 95942689T AT E207929 T1 ATE207929 T1 AT E207929T1
Authority
AT
Austria
Prior art keywords
androan
antiandrogens
thioxo
aza
oxo
Prior art date
Application number
AT95942689T
Other languages
English (en)
Inventor
Stefano Poli
Roberto Girardello
Paride Grisenti
Ambrogio Magni
Vincenzo Olgiati
Original Assignee
Polichem Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Polichem Sa filed Critical Polichem Sa
Application granted granted Critical
Publication of ATE207929T1 publication Critical patent/ATE207929T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT95942689T 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene ATE207929T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI942626A IT1271325B (it) 1994-12-23 1994-12-23 Composti diastereomericamente puri derivati da 3-oxo e 3-tioxo-4-azaandrostani e loro uso come antiandrogeni
PCT/EP1995/005008 WO1996020210A2 (en) 1994-12-23 1995-12-18 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens

Publications (1)

Publication Number Publication Date
ATE207929T1 true ATE207929T1 (de) 2001-11-15

Family

ID=11370067

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95942689T ATE207929T1 (de) 1994-12-23 1995-12-18 Diastereomerenreine 3-oxo und 3-thioxo-4-aza- androstanderivate und ihre verwendung als antiandrogene

Country Status (10)

Country Link
US (1) US6147213A (de)
EP (1) EP0799239B1 (de)
AT (1) ATE207929T1 (de)
AU (1) AU4387296A (de)
DE (1) DE69523622T2 (de)
DK (1) DK0799239T3 (de)
ES (1) ES2163538T3 (de)
IT (1) IT1271325B (de)
PT (1) PT799239E (de)
WO (1) WO1996020210A2 (de)

Families Citing this family (23)

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Publication number Priority date Publication date Assignee Title
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
KR101496934B1 (ko) 2006-11-15 2015-03-03 유니버시티 오브 워싱톤 스루 이츠 센터 포 커머셜리제이션 전기 이중층 캐패시턴스 장치
PT2532648E (pt) * 2007-05-03 2014-04-24 Univ Yale Antiandrogénios «suaves» localmente activos
CN105226284B (zh) 2009-07-01 2017-11-28 巴斯夫欧洲公司 超纯合成碳材料
EP2510569B1 (de) * 2009-12-11 2020-07-22 Basf Se Kohlenstoffmaterialien mit einem elektrochemischen modifikator
US8916296B2 (en) 2010-03-12 2014-12-23 Energ2 Technologies, Inc. Mesoporous carbon materials comprising bifunctional catalysts
WO2012045002A1 (en) 2010-09-30 2012-04-05 Energ2 Technologies, Inc. Enhanced packing of energy storage particles
JP6324726B2 (ja) 2010-12-28 2018-05-16 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 電気化学特性が向上した炭素材料
US20120262127A1 (en) 2011-04-15 2012-10-18 Energ2 Technologies, Inc. Flow ultracapacitor
CN103947017B (zh) 2011-06-03 2017-11-17 巴斯福股份公司 用于混合能量存储装置中的碳‑铅共混物
WO2013120011A1 (en) 2012-02-09 2013-08-15 Energ2 Technologies, Inc. Preparation of polymeric resins and carbon materials
CN110112377A (zh) 2013-03-14 2019-08-09 14族科技公司 包含锂合金化的电化学改性剂的复合碳材料
US10195583B2 (en) 2013-11-05 2019-02-05 Group 14 Technologies, Inc. Carbon-based compositions with highly efficient volumetric gas sorption
KR102663138B1 (ko) 2014-03-14 2024-05-03 그룹14 테크놀로지스, 인코포레이티드 용매의 부재하의 졸-겔 중합을 위한 신규한 방법 및 그러한 방법으로부터의 가변형 탄소 구조의 생성
US20190097222A1 (en) 2015-08-14 2019-03-28 Energ2 Technologies, Inc. Composites of porous nano-featured silicon materials and carbon materials
CN119419246A (zh) 2015-08-28 2025-02-11 14集团技术公司 具有极其持久的锂嵌入的新型材料及其制造方法
EP3593369A4 (de) 2017-03-09 2021-03-03 Group14 Technologies, Inc. Zersetzung von siliciumhaltigen vorläufern auf porösen gerüstmaterialien
JP2023537954A (ja) 2020-08-10 2023-09-06 グループ１４・テクノロジーズ・インコーポレイテッド 振動熱補助化学気相浸透
EP4146595A1 (de) 2020-08-18 2023-03-15 Group14 Technologies, Inc. Herstellung von silicium-kohlenstoff-verbundwerkstoffen
US11639292B2 (en) 2020-08-18 2023-05-02 Group14 Technologies, Inc. Particulate composite materials
US11174167B1 (en) 2020-08-18 2021-11-16 Group14 Technologies, Inc. Silicon carbon composites comprising ultra low Z
US11335903B2 (en) 2020-08-18 2022-05-17 Group14 Technologies, Inc. Highly efficient manufacturing of silicon-carbon composites materials comprising ultra low z
CN116457309B (zh) 2020-09-30 2025-02-14 14集团技术公司 控制硅-碳复合材料的氧含量和反应性的钝化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4845104A (en) * 1986-11-20 1989-07-04 Merck & Co., Inc. Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
IE76452B1 (en) * 1990-10-29 1997-10-22 Sankyo Co Azasteroid compounds for the treatment of prostatic hypertrophy their preparation and use
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives

Also Published As

Publication number Publication date
PT799239E (pt) 2002-02-28
ITMI942626A1 (it) 1996-06-23
IT1271325B (it) 1997-05-27
EP0799239A2 (de) 1997-10-08
DK0799239T3 (da) 2001-12-10
US6147213A (en) 2000-11-14
DE69523622D1 (de) 2001-12-06
DE69523622T2 (de) 2002-05-29
ITMI942626A0 (it) 1994-12-23
AU4387296A (en) 1996-07-19
WO1996020210A3 (en) 1996-09-06
ES2163538T3 (es) 2002-02-01
EP0799239B1 (de) 2001-10-31
WO1996020210A2 (en) 1996-07-04

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