ATE212642T1 - Verfahren zur herstellung von aspartyl- cyclohexylalaninamid - Google Patents

Verfahren zur herstellung von aspartyl- cyclohexylalaninamid

Info

Publication number: ATE212642T1
Authority: AT; Austria
Prior art keywords: aspartyl; cyclohexylalaninamide; alpha; salt; optionally
Prior art date: 1998-06-05

Application number

AT99923656T

Other languages

English (en)

Inventor

Robert Stammler

Christophe Daubie

Michel Lavigne

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-06-05

Filing date

1999-06-03

Publication date

2002-02-15

1998-06-05 Priority claimed from FR9807069A external-priority patent/FR2779431B1/fr

1999-06-03 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2002-02-15 Application granted granted Critical

2002-02-15 Publication of ATE212642T1 publication Critical patent/ATE212642T1/de

Links

OWGNMFJENYYYAS-WPRPVWTQSA-N C[C@H](N(C1CCCCC1)C(=O)[C@@H](N)CC(O)=O)C(N)=O Chemical compound C[C@H](N(C1CCCCC1)C(=O)[C@@H](N)CC(O)=O)C(N)=O OWGNMFJENYYYAS-WPRPVWTQSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
150000003839 salts Chemical class 0.000 abstract 2
LRXLYISFSGZAEB-UWVGGRQHSA-N (3s)-3-amino-4-[[(2s)-1-amino-3-cyclohexyl-1-oxopropan-2-yl]amino]-4-oxobutanoic acid Chemical compound OC(=O)C[C@H](N)C(=O)N[C@H](C(N)=O)CC1CCCCC1 LRXLYISFSGZAEB-UWVGGRQHSA-N 0.000 abstract 1
241001502050 Acis Species 0.000 abstract 1
CREJAHXXJNVUCT-IYPAPVHQSA-N N[C@@H](CC(O)=O)C(NC([C@H](CC1=CC=CC=C1)N)=O)=O.N Chemical compound N[C@@H](CC(O)=O)C(NC([C@H](CC1=CC=CC=C1)N)=O)=O.N CREJAHXXJNVUCT-IYPAPVHQSA-N 0.000 abstract 1
-1 alpha-aspartyl phenylamine ester Chemical class 0.000 abstract 1
238000010640 amide synthesis reaction Methods 0.000 abstract 1
238000009903 catalytic hydrogenation reaction Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
230000001131 transforming effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06104—Dipeptides with the first amino acid being acidic
- C07K5/06113—Asp- or Asn-amino acid

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Biochemistry (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Peptides Or Proteins (AREA)

AT99923656T 1998-06-05 1999-06-03 Verfahren zur herstellung von aspartyl- cyclohexylalaninamid ATE212642T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR9807069A FR2779431B1 (fr)	1998-06-05	1998-06-05	Procede de preparation de l'aspartyl cyclohexylalaninamide
US10441798P	1998-10-15	1998-10-15
PCT/FR1999/001300 WO1999064443A1 (fr)	1998-06-05	1999-06-03	Procede de preparation de l'aspartyl cyclohexylalaninamide

Publications (1)

Publication Number	Publication Date
ATE212642T1 true ATE212642T1 (de)	2002-02-15

Family

ID=26234363

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99923656T ATE212642T1 (de)	1998-06-05	1999-06-03	Verfahren zur herstellung von aspartyl- cyclohexylalaninamid

Country Status (10)

Country	Link
US (1)	US6384272B2 (de)
EP (1)	EP1084138B1 (de)
JP (1)	JP4317326B2 (de)
AT (1)	ATE212642T1 (de)
AU (1)	AU4044699A (de)
DE (1)	DE69900850T2 (de)
DK (1)	DK1084138T3 (de)
ES (1)	ES2170581T3 (de)
PT (1)	PT1084138E (de)
WO (1)	WO1999064443A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HRP20040784A2 (en) *	2002-01-29	2005-04-30	Wyeth	Compositions and methods for modulating connexin hemichannels

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE902238A1 (en) *	1989-06-30	1991-01-16	Abbott Lab	Tetrapeptide type-b cck receptor ligands
US5340802A (en)	1989-06-30	1994-08-23	Abbott Laboratories	Peptide analog type-B CCK receptor ligands
NL1005808C2 (nl) *	1997-04-14	1998-10-19	Dsm Nv	Hexahydro-aspartaamamiden en werkwijze voor de bereiding ervan.

1999
- 1999-06-03 AT AT99923656T patent/ATE212642T1/de active
- 1999-06-03 WO PCT/FR1999/001300 patent/WO1999064443A1/fr not_active Ceased
- 1999-06-03 JP JP2000553451A patent/JP4317326B2/ja not_active Expired - Fee Related
- 1999-06-03 PT PT99923656T patent/PT1084138E/pt unknown
- 1999-06-03 DK DK99923656T patent/DK1084138T3/da active
- 1999-06-03 DE DE69900850T patent/DE69900850T2/de not_active Expired - Lifetime
- 1999-06-03 AU AU40446/99A patent/AU4044699A/en not_active Abandoned
- 1999-06-03 ES ES99923656T patent/ES2170581T3/es not_active Expired - Lifetime
- 1999-06-03 EP EP99923656A patent/EP1084138B1/de not_active Expired - Lifetime
2000
- 2000-12-04 US US09/729,011 patent/US6384272B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
WO1999064443A1 (fr)	1999-12-16
US20010034460A1 (en)	2001-10-25
AU4044699A (en)	1999-12-30
DE69900850T2 (de)	2002-08-29
DK1084138T3 (da)	2002-04-22
EP1084138B1 (de)	2002-01-30
US6384272B2 (en)	2002-05-07
JP2002517509A (ja)	2002-06-18
DE69900850D1 (de)	2002-03-14
EP1084138A1 (de)	2001-03-21
JP4317326B2 (ja)	2009-08-19
ES2170581T3 (es)	2002-08-01
PT1084138E (pt)	2002-07-31

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Legal Events

Date	Code	Title	Description
2002-06-15	UEP	Publication of translation of european patent specification