ATE222255T1 - 14-substituierte marcfortine und derivate als antiparasitäre mittel - Google Patents

14-substituierte marcfortine und derivate als antiparasitäre mittel

Info

Publication number
ATE222255T1
ATE222255T1 AT94920689T AT94920689T ATE222255T1 AT E222255 T1 ATE222255 T1 AT E222255T1 AT 94920689 T AT94920689 T AT 94920689T AT 94920689 T AT94920689 T AT 94920689T AT E222255 T1 ATE222255 T1 AT E222255T1
Authority
AT
Austria
Prior art keywords
derivatives
antiparasic
agents
marcfortine
substituted
Prior art date
Application number
AT94920689T
Other languages
English (en)
Inventor
Byung H Lee
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of ATE222255T1 publication Critical patent/ATE222255T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Curing Cements, Concrete, And Artificial Stone (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Enzymes And Modification Thereof (AREA)
AT94920689T 1993-06-16 1994-06-07 14-substituierte marcfortine und derivate als antiparasitäre mittel ATE222255T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7807693A 1993-06-16 1993-06-16
PCT/US1994/006037 WO1994029319A1 (en) 1993-06-16 1994-06-07 14-substituted marcfortines and derivatives useful as antiparasitic agents

Publications (1)

Publication Number Publication Date
ATE222255T1 true ATE222255T1 (de) 2002-08-15

Family

ID=22141768

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94920689T ATE222255T1 (de) 1993-06-16 1994-06-07 14-substituierte marcfortine und derivate als antiparasitäre mittel

Country Status (25)

Country Link
US (1) US5750533A (de)
EP (1) EP0703916B1 (de)
JP (2) JP3747059B2 (de)
KR (1) KR100332192B1 (de)
CN (1) CN1058266C (de)
AT (1) ATE222255T1 (de)
AU (1) AU686188B2 (de)
CA (1) CA2161960A1 (de)
CZ (1) CZ289684B6 (de)
DE (1) DE69431187T2 (de)
DK (1) DK0703916T3 (de)
ES (1) ES2181722T3 (de)
FI (1) FI956045L (de)
HU (1) HU223768B1 (de)
IL (1) IL109958A0 (de)
MY (1) MY111601A (de)
NO (1) NO313803B1 (de)
NZ (1) NZ268476A (de)
PL (1) PL180406B1 (de)
PT (1) PT703916E (de)
RU (1) RU2131877C1 (de)
SK (1) SK283594B6 (de)
TW (1) TW410227B (de)
WO (1) WO1994029319A1 (de)
ZA (1) ZA943959B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY113806A (en) * 1995-07-21 2002-05-31 Upjohn Co Antiparasitic marcfortines and paraherquamides
ZA976761B (en) * 1996-09-09 1999-01-29 Upjohn Co 25 Methylene and 24,25-epoxy marcfortines and paraherquamides
WO1998021211A1 (en) * 1996-11-15 1998-05-22 Pharmacia & Upjohn Company 1- and 2-substituted marcfortines and paraherquamides as antiparasitic agents

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US390532A (en) * 1888-10-02 titscher
US5075307A (en) * 1987-07-28 1991-12-24 Merck & Co., Inc. Paraherquamide and dihydroparaherquamide as antihelminthic agents
US4873247A (en) * 1987-11-27 1989-10-10 Goegelman Robert T Derivatives of paraherquamide isolated from a fermentation broth active as antiparasitic agents
US4978656A (en) * 1988-08-12 1990-12-18 Merck & Co., Inc. Synthetic derivatives of paraherquamide
US4923867A (en) * 1988-08-24 1990-05-08 Merck & Co., Inc. Synthetic marcfortine derivatives useful as antiparasitic agents
DE3831839A1 (de) * 1988-09-20 1990-03-29 Standard Elektrik Lorenz Ag Optischer sende- und/oder empfangsbaustein
NZ233043A (en) * 1989-03-30 1992-09-25 Merck & Co Inc Anthelmintic heterocyclic compounds prepared by action of cunninghamella blakesleeana on (dihydro)paraherquamide
US5032595A (en) * 1989-11-24 1991-07-16 Fidia-Georgetown Institute For The Neurosciences Method of stimulating steroidogenesis with alpidem
IE904606A1 (en) * 1989-12-21 1991-07-03 Beecham Group Plc Novel products
GB9014194D0 (en) * 1990-06-26 1990-08-15 Pfizer Ltd Antiparasitic agents
GB2247026B (en) * 1990-06-26 1994-09-28 Amoco Corp Purification of a dialkylated transalkylation product
WO1992022555A1 (en) * 1991-06-17 1992-12-23 Beecham Group Plc Paraherquamide derivatives, precursor thereof, processes for their preparation, microorganism used and their use as antiparasitic agents
JPH07501693A (ja) * 1991-11-22 1995-02-23 ジ・アップジョン・カンパニー 抗寄生虫病剤として有用なマークフォルティン／パラハークアミド誘導体

Also Published As

Publication number Publication date
EP0703916B1 (de) 2002-08-14
CA2161960A1 (en) 1994-12-22
CN1125448A (zh) 1996-06-26
PL180406B1 (pl) 2001-01-31
US5750533A (en) 1998-05-12
ES2181722T3 (es) 2003-03-01
JPH08511529A (ja) 1996-12-03
EP0703916A1 (de) 1996-04-03
SK283594B6 (sk) 2003-10-07
JP2005162766A (ja) 2005-06-23
NO955093L (no) 1996-02-15
DE69431187D1 (de) 2002-09-19
AU686188B2 (en) 1998-02-05
RU2131877C1 (ru) 1999-06-20
DK0703916T3 (da) 2002-12-02
HU9503594D0 (en) 1996-02-28
PL312258A1 (en) 1996-04-15
TW410227B (en) 2000-11-01
WO1994029319A1 (en) 1994-12-22
KR960703127A (ko) 1996-06-19
AU7138994A (en) 1995-01-03
SK152595A3 (en) 1997-06-04
CZ289684B6 (cs) 2002-03-13
CZ316495A3 (en) 1996-03-13
NO955093D0 (no) 1995-12-15
JP3747059B2 (ja) 2006-02-22
FI956045A7 (fi) 1995-12-15
CN1058266C (zh) 2000-11-08
FI956045A0 (fi) 1995-12-15
HU223768B1 (hu) 2005-01-28
HUT74680A (en) 1997-01-28
KR100332192B1 (ko) 2002-11-27
MY111601A (en) 2000-09-27
ZA943959B (en) 1995-12-06
PT703916E (pt) 2002-12-31
NO313803B1 (no) 2002-12-02
DE69431187T2 (de) 2003-04-10
IL109958A0 (en) 1994-10-07
NZ268476A (en) 1997-11-24
FI956045L (fi) 1995-12-15

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee