ATE235486T1 - Verfahren zu herstellung von o-fluorierten tetrahydrothiopyran carbamaten - Google Patents

Verfahren zu herstellung von o-fluorierten tetrahydrothiopyran carbamaten

Info

Publication number: ATE235486T1
Authority: AT; Austria
Prior art keywords: tetrahydrothiopyran; fluorinated; carbamates; producing; cyclic
Prior art date: 1999-02-01

Application number

AT00909891T

Other languages

English (en)

Inventor

James R Gage

Original Assignee

Upjohn Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-02-01

Filing date

2000-01-31

Publication date

2003-04-15

2000-01-31 Application filed by Upjohn Co filed Critical Upjohn Co

2003-04-15 Application granted granted Critical

2003-04-15 Publication of ATE235486T1 publication Critical patent/ATE235486T1/de

Links

KXDHJXZQYSOELW-UHFFFAOYSA-M Carbamate Chemical compound NC([O-])=O KXDHJXZQYSOELW-UHFFFAOYSA-M 0.000 title 1
YPWFISCTZQNZAU-UHFFFAOYSA-N Thiane Chemical class C1CCSCC1 YPWFISCTZQNZAU-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical compound O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 abstract 1
YCKRFDGAMUMZLT-UHFFFAOYSA-N Fluorine atom Chemical compound [F] YCKRFDGAMUMZLT-UHFFFAOYSA-N 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
150000004657 carbamic acid derivatives Chemical class 0.000 abstract 1
229910052731 fluorine Inorganic materials 0.000 abstract 1
239000011737 fluorine Substances 0.000 abstract 1
229910052717 sulfur Inorganic materials 0.000 abstract 1
239000011593 sulfur Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
- C07D335/02—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Plural Heterocyclic Compounds (AREA)

AT00909891T 1999-02-01 2000-01-31 Verfahren zu herstellung von o-fluorierten tetrahydrothiopyran carbamaten ATE235486T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US11815099P	1999-02-01	1999-02-01
PCT/US2000/000506 WO2000044741A2 (en)	1999-02-01	2000-01-31	Process to prepare cyclic-sulfur fluorine containing oxazolidinones

Publications (1)

Publication Number	Publication Date
ATE235486T1 true ATE235486T1 (de)	2003-04-15

Family

ID=22376779

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AT02009273T ATE293616T1 (de)	1999-02-01	2000-01-31	2-fluoro-(oxido-thiopyran-4-yl)benzol derivate
AT00909891T ATE235486T1 (de)	1999-02-01	2000-01-31	Verfahren zu herstellung von o-fluorierten tetrahydrothiopyran carbamaten

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AT02009273T ATE293616T1 (de)	1999-02-01	2000-01-31	2-fluoro-(oxido-thiopyran-4-yl)benzol derivate

Country Status (20)

Country	Link
US (1)	US6239283B1 (de)
EP (1)	EP1149089B1 (de)
JP (1)	JP2002535400A (de)
KR (1)	KR20010101890A (de)
CN (2)	CN1495181A (de)
AT (2)	ATE293616T1 (de)
AU (1)	AU767579B2 (de)
BR (1)	BR0007918A (de)
CA (1)	CA2359711A1 (de)
DE (2)	DE60001807T2 (de)
DK (1)	DK1149089T3 (de)
ES (2)	ES2241920T3 (de)
HK (1)	HK1042697B (de)
HU (1)	HUP0200003A3 (de)
IL (1)	IL144669A0 (de)
NZ (1)	NZ513292A (de)
PL (1)	PL349911A1 (de)
PT (1)	PT1149089E (de)
WO (1)	WO2000044741A2 (de)
ZA (1)	ZA200105844B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN1072222C (zh) *	1995-09-01	2001-10-03	法玛西雅厄普约翰公司	以c－c键连接于4－8元杂环环的苯基噁唑烷酮
GB9928568D0 (en)	1999-12-03	2000-02-02	Zeneca Ltd	Chemical compounds
GB0009803D0 (en)	2000-04-25	2000-06-07	Astrazeneca Ab	Chemical compounds
WO2002002095A2 (en)	2000-06-30	2002-01-10	Pharmacia & Upjohn Company	Compositions for treating bacterial infections containing oxazolidinone compound, sulbactam and an ampicillin
AR038536A1 (es)	2002-02-25	2005-01-19	Upjohn Co	N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
US7141588B2 (en) *	2002-02-25	2006-11-28	Pfizer, Inc.	N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
JP2006516989A (ja) *	2003-02-07	2006-07-13	ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー	抗菌剤として使用するための二環式環によりｎ−置換されたオキサゾリジノン誘導体
JP2006516991A (ja) *	2003-02-07	2006-07-13	ワーナー−ランバート・カンパニー、リミテッド、ライアビリティ、カンパニー	抗菌剤
US7304050B2 (en)	2003-09-16	2007-12-04	Pfizer Inc.	Antibacterial agents
BRPI0513083A (pt) *	2004-08-06	2008-04-22	Pharmacia & Upjohn Co Llc	oxazolidinonas contendo oxindóis como agentes antibacterianos

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CN1072222C (zh) *	1995-09-01	2001-10-03	法玛西雅厄普约翰公司	以c－c键连接于4－8元杂环环的苯基噁唑烷酮
GB9702213D0 (en)	1996-02-24	1997-03-26	Zeneca Ltd	Chemical compounds
ATE209193T1 (de)	1996-04-11	2001-12-15	Upjohn Co	Verfahren zur herstellung von oxazolidinonen

2000
- 2000-01-31 ES ES02009273T patent/ES2241920T3/es not_active Expired - Lifetime
- 2000-01-31 US US09/495,017 patent/US6239283B1/en not_active Expired - Fee Related
- 2000-01-31 DE DE60001807T patent/DE60001807T2/de not_active Expired - Fee Related
- 2000-01-31 WO PCT/US2000/000506 patent/WO2000044741A2/en not_active Ceased
- 2000-01-31 NZ NZ513292A patent/NZ513292A/en unknown
- 2000-01-31 EP EP00909891A patent/EP1149089B1/de not_active Expired - Lifetime
- 2000-01-31 DE DE60019630T patent/DE60019630T2/de not_active Expired - Fee Related
- 2000-01-31 CN CNA200310102715XA patent/CN1495181A/zh active Pending
- 2000-01-31 AT AT02009273T patent/ATE293616T1/de not_active IP Right Cessation
- 2000-01-31 DK DK00909891T patent/DK1149089T3/da active
- 2000-01-31 AU AU32076/00A patent/AU767579B2/en not_active Ceased
- 2000-01-31 PL PL00349911A patent/PL349911A1/xx not_active Application Discontinuation
- 2000-01-31 IL IL14466900A patent/IL144669A0/xx unknown
- 2000-01-31 HK HK02104073.0A patent/HK1042697B/zh not_active IP Right Cessation
- 2000-01-31 CA CA002359711A patent/CA2359711A1/en not_active Abandoned
- 2000-01-31 AT AT00909891T patent/ATE235486T1/de not_active IP Right Cessation
- 2000-01-31 PT PT00909891T patent/PT1149089E/pt unknown
- 2000-01-31 JP JP2000595997A patent/JP2002535400A/ja active Pending
- 2000-01-31 KR KR1020017009639A patent/KR20010101890A/ko not_active Ceased
- 2000-01-31 BR BR0007918-9A patent/BR0007918A/pt not_active IP Right Cessation
- 2000-01-31 HU HU0200003A patent/HUP0200003A3/hu unknown
- 2000-01-31 ES ES00909891T patent/ES2194709T3/es not_active Expired - Lifetime
- 2000-01-31 CN CNB008025738A patent/CN1142158C/zh not_active Expired - Fee Related
2001
- 2001-07-16 ZA ZA200105844A patent/ZA200105844B/en unknown

Also Published As

Publication number	Publication date
HK1042697A1 (en)	2002-08-23
ATE293616T1 (de)	2005-05-15
HUP0200003A2 (en)	2002-06-29
NZ513292A (en)	2003-08-29
ES2241920T3 (es)	2005-11-01
IL144669A0 (en)	2002-05-23
US6239283B1 (en)	2001-05-29
KR20010101890A (ko)	2001-11-15
HUP0200003A3 (en)	2002-11-28
CA2359711A1 (en)	2000-08-03
PT1149089E (pt)	2003-07-31
JP2002535400A (ja)	2002-10-22
EP1149089A2 (de)	2001-10-31
WO2000044741A2 (en)	2000-08-03
CN1142158C (zh)	2004-03-17
WO2000044741A3 (en)	2000-12-07
DE60019630T2 (de)	2006-03-16
ES2194709T3 (es)	2003-12-01
DE60019630D1 (de)	2005-05-25
DE60001807D1 (de)	2003-04-30
DK1149089T3 (da)	2003-07-21
AU767579B2 (en)	2003-11-20
CN1495181A (zh)	2004-05-12
PL349911A1 (en)	2002-10-07
HK1042697B (zh)	2004-08-20
BR0007918A (pt)	2001-10-23
CN1335842A (zh)	2002-02-13
EP1149089B1 (de)	2003-03-26
DE60001807T2 (de)	2003-11-06
ZA200105844B (en)	2002-07-16
AU3207600A (en)	2000-08-18

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Legal Events

Date

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2003-07-15

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Publication of translation of european patent specification

Ref document number: 1149089

Country of ref document: EP

2006-10-15

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