ATE244706T1 - Enantiomere von mercaptolactonen und verfahren zu ihrer herstellung - Google Patents
Enantiomere von mercaptolactonen und verfahren zu ihrer herstellungInfo
- Publication number
- ATE244706T1 ATE244706T1 AT00917002T AT00917002T ATE244706T1 AT E244706 T1 ATE244706 T1 AT E244706T1 AT 00917002 T AT00917002 T AT 00917002T AT 00917002 T AT00917002 T AT 00917002T AT E244706 T1 ATE244706 T1 AT E244706T1
- Authority
- AT
- Austria
- Prior art keywords
- enantiomers
- mercaptolactones
- production
- processes
- formula
- Prior art date
Links
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical compound C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 title abstract 2
- 239000000543 intermediate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/26—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D307/30—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/32—Oxygen atoms
- C07D307/33—Oxygen atoms in position 2, the oxygen atom being in its keto or unsubstituted enol form
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/0026—Oxygen-containing hetero ring cyclic ketals
- C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9909229.8A GB9909229D0 (en) | 1999-04-23 | 1999-04-23 | Enantiomers of mercapto lactones and processes for their synthesis |
| PCT/EP2000/002705 WO2000064882A2 (en) | 1999-04-23 | 2000-03-28 | Enantiomers of mercapto lactones and processes for their synthesis |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE244706T1 true ATE244706T1 (de) | 2003-07-15 |
Family
ID=10852031
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00917002T ATE244706T1 (de) | 1999-04-23 | 2000-03-28 | Enantiomere von mercaptolactonen und verfahren zu ihrer herstellung |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP1173430B1 (de) |
| JP (1) | JP2002543069A (de) |
| AT (1) | ATE244706T1 (de) |
| AU (1) | AU3814800A (de) |
| DE (1) | DE60003807T2 (de) |
| ES (1) | ES2202090T3 (de) |
| GB (1) | GB9909229D0 (de) |
| WO (1) | WO2000064882A2 (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003255851B2 (en) | 2002-07-08 | 2009-07-23 | Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. | New compounds, compositions and methods for treatment of inflammatory diseases and conditions |
| NZ537716A (en) | 2002-07-08 | 2007-05-31 | Glaxosmithkline Zagreb | Novel nonsteroidal anti-inflammatory substances, compositions and methods for their use |
| EP1551865B1 (de) | 2002-07-08 | 2009-04-22 | GlaxoSmithKline istrazivacki centar Zagreb d.o.o. | Hybridmoleküle von makroliden mit steroidalen/nicht-steroidalen antientzündlich aktiven molekülen |
| JP5192730B2 (ja) * | 2006-05-29 | 2013-05-08 | 昭和電工株式会社 | メルカプト複素環化合物の製造方法 |
| ES2385848T3 (es) | 2006-05-29 | 2012-08-01 | Showa Denko K.K. | Procedimiento de producción de un compuesto mercapto heterocíclico |
| EP2443134A2 (de) | 2009-06-16 | 2012-04-25 | Schering Corporation | Neue [3,2-c]heteroarylsteroide als glucocorticoidrezeptoragonisten, zusammensetzungen und verwendung |
| EP4635969A1 (de) * | 2022-12-16 | 2025-10-22 | Tianjin Pharmaceutical Biotechnology Co., Ltd. | Neues glucocorticoid, verfahren zu seiner herstellung und seine verwendung |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SK89198A3 (en) * | 1995-12-29 | 1999-03-12 | Glaxo Group Ltd | Lactone derivatives of 17.beta.-carboxy, carbothio and amide androstane derivatives |
-
1999
- 1999-04-23 GB GBGB9909229.8A patent/GB9909229D0/en not_active Ceased
-
2000
- 2000-03-28 ES ES00917002T patent/ES2202090T3/es not_active Expired - Lifetime
- 2000-03-28 AU AU38148/00A patent/AU3814800A/en not_active Abandoned
- 2000-03-28 DE DE60003807T patent/DE60003807T2/de not_active Expired - Fee Related
- 2000-03-28 AT AT00917002T patent/ATE244706T1/de not_active IP Right Cessation
- 2000-03-28 WO PCT/EP2000/002705 patent/WO2000064882A2/en not_active Ceased
- 2000-03-28 JP JP2000613835A patent/JP2002543069A/ja active Pending
- 2000-03-28 EP EP00917002A patent/EP1173430B1/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| WO2000064882A2 (en) | 2000-11-02 |
| GB9909229D0 (en) | 1999-06-16 |
| DE60003807D1 (de) | 2003-08-14 |
| WO2000064882A3 (en) | 2001-02-22 |
| EP1173430B1 (de) | 2003-07-09 |
| EP1173430A1 (de) | 2002-01-23 |
| ES2202090T3 (es) | 2004-04-01 |
| DE60003807T2 (de) | 2004-05-27 |
| AU3814800A (en) | 2000-11-10 |
| JP2002543069A (ja) | 2002-12-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |