ATE248606T1 - Kombinationen einem ibat inhibitor und einem mtp inhibitor für kardiovaskuläre indikationen - Google Patents

Kombinationen einem ibat inhibitor und einem mtp inhibitor für kardiovaskuläre indikationen

Info

Publication number
ATE248606T1
ATE248606T1 AT99965901T AT99965901T ATE248606T1 AT E248606 T1 ATE248606 T1 AT E248606T1 AT 99965901 T AT99965901 T AT 99965901T AT 99965901 T AT99965901 T AT 99965901T AT E248606 T1 ATE248606 T1 AT E248606T1
Authority
AT
Austria
Prior art keywords
inhibitor
combinations
ibat
mtp
cardiovascular indications
Prior art date
Application number
AT99965901T
Other languages
English (en)
Inventor
Bradley T Keller
David B Reitz
Joseph R Schuh
James A Sikorski
Samuel J Tremont
Rodney W Lappe
Original Assignee
Searle Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22352512&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE248606(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Searle Llc filed Critical Searle Llc
Application granted granted Critical
Publication of ATE248606T1 publication Critical patent/ATE248606T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT99965901T 1998-12-23 1999-12-17 Kombinationen einem ibat inhibitor und einem mtp inhibitor für kardiovaskuläre indikationen ATE248606T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11395598P 1998-12-23 1998-12-23
PCT/US1999/027946 WO2000038725A1 (en) 1998-12-23 1999-12-17 Combinations for cardiovascular indications

Publications (1)

Publication Number Publication Date
ATE248606T1 true ATE248606T1 (de) 2003-09-15

Family

ID=22352512

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99965901T ATE248606T1 (de) 1998-12-23 1999-12-17 Kombinationen einem ibat inhibitor und einem mtp inhibitor für kardiovaskuläre indikationen

Country Status (23)

Country Link
US (1) US20040058908A1 (de)
EP (2) EP1354604A1 (de)
JP (1) JP2002533411A (de)
KR (1) KR20020002367A (de)
CN (1) CN1342091A (de)
AR (1) AR037482A1 (de)
AT (1) ATE248606T1 (de)
AU (1) AU779264B2 (de)
BR (1) BR9916564A (de)
CA (1) CA2356515A1 (de)
CZ (1) CZ20012344A3 (de)
DE (1) DE69911058T2 (de)
DK (1) DK1140187T3 (de)
EA (1) EA200100704A1 (de)
ES (1) ES2207330T3 (de)
HU (1) HUP0104655A2 (de)
IL (1) IL143944A0 (de)
MX (1) MXPA01006468A (de)
NO (1) NO20013157L (de)
NZ (1) NZ512532A (de)
PT (1) PT1140187E (de)
WO (1) WO2000038725A1 (de)
ZA (5) ZA200105056B (de)

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ZA200105062B (en) 2002-08-28
CN1342091A (zh) 2002-03-27
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HUP0104655A2 (hu) 2002-04-29
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AU779264B2 (en) 2005-01-13
DE69911058D1 (de) 2003-10-09
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EP1140187A1 (de) 2001-10-10
PT1140187E (pt) 2004-01-30
ZA200105056B (en) 2002-06-20
EP1140187B1 (de) 2003-09-03
CZ20012344A3 (cs) 2002-01-16
DE69911058T2 (de) 2004-06-03
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