ATE260928T1 - Ketolidantibiotika - Google Patents

Ketolidantibiotika

Info

Publication number
ATE260928T1
ATE260928T1 AT01301966T AT01301966T ATE260928T1 AT E260928 T1 ATE260928 T1 AT E260928T1 AT 01301966 T AT01301966 T AT 01301966T AT 01301966 T AT01301966 T AT 01301966T AT E260928 T1 ATE260928 T1 AT E260928T1
Authority
AT
Austria
Prior art keywords
compounds
formula
infections
relates
ketolide antibiotics
Prior art date
Application number
AT01301966T
Other languages
English (en)
Inventor
Takushi Kaneko
William Thomas Mcmillen
Wei-Guo Su
Hongjuan Zhao
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE260928T1 publication Critical patent/ATE260928T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Cephalosporin Compounds (AREA)
AT01301966T 2000-03-06 2001-03-05 Ketolidantibiotika ATE260928T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18697000P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
ATE260928T1 true ATE260928T1 (de) 2004-03-15

Family

ID=22687057

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01301966T ATE260928T1 (de) 2000-03-06 2001-03-05 Ketolidantibiotika

Country Status (11)

Country Link
US (1) US6555524B2 (de)
EP (1) EP1132392B1 (de)
JP (1) JP2001261694A (de)
AT (1) ATE260928T1 (de)
BR (1) BR0100850A (de)
CA (1) CA2339051A1 (de)
DE (1) DE60102171T2 (de)
DK (1) DK1132392T3 (de)
ES (1) ES2214385T3 (de)
PT (1) PT1132392E (de)
TR (1) TR200400630T4 (de)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5413293A (en) * 1992-12-22 1995-05-09 Hughes Aircraft Company Magnetic torque attitude control systems
US6555581B1 (en) 2001-02-15 2003-04-29 Jones Pharma, Inc. Levothyroxine compositions and methods
US7067148B2 (en) 2001-02-15 2006-06-27 King Pharmaceutical Research & Development, Inc. Stabilized pharmaceutical and thyroid hormone compositions and method of preparation
US7101569B2 (en) 2001-08-14 2006-09-05 Franz G Andrew Methods of administering levothyroxine pharmaceutical compositions
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
TW200420573A (en) 2002-09-26 2004-10-16 Rib X Pharmaceuticals Inc Bifunctional heterocyclic compounds and methods of making and using same
EP1638549A4 (de) 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc Neue antibakterielle mittel
EP1723159B1 (de) 2004-02-27 2019-06-12 Melinta Therapeutics, Inc. Makrozyklische verbindungen, deren herstellung und verwendung
UA85937C2 (uk) 2004-12-21 2009-03-10 Пфайзер Продактс Інк. Макроліди
US7387972B2 (en) * 2006-03-01 2008-06-17 Promos Technologies Pte. Ltd. Reducing nitrogen concentration with in-situ steam generation
EP2214484A4 (de) 2007-10-25 2013-01-02 Cempra Pharmaceuticals Inc Verfahren zur herstellung von antibakteriellen makrolid-wirkstoffen
JP5711135B2 (ja) 2008-10-24 2015-04-30 センプラ ファーマシューティカルズ,インコーポレイテッド 胃腸疾患を治療するための方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
ES2608285T3 (es) * 2009-09-10 2017-04-07 Cempra Pharmaceuticals, Inc. Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC
MX361413B (es) 2010-03-22 2018-12-05 Cempra Pharmaceuticals Inc Star Formas cristalinas de un macrólido y usos para las mismas.
CN102917708B (zh) 2010-05-20 2015-11-25 森普拉制药公司 制备大环内酯和酮内酯及其中间体的方法
EP2613630A4 (de) 2010-09-10 2014-01-15 Cempra Pharmaceuticals Inc Wasserstoffbindung zur formung von fluorketoliden zur behandlung von krankheiten
NZ700182A (en) 2012-03-27 2017-02-24 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
AU2014239959A1 (en) 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
CN105188712A (zh) 2013-03-15 2015-12-23 森普拉制药公司 用于制备大环内酯抗菌剂的收敛方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CO4990960A1 (es) 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
FR2777282B1 (fr) 1998-04-08 2001-04-20 Hoechst Marion Roussel Inc Nouveaux derives de la 2-fluoro 3-de((2,6-dideoxy 3-c-methyl 3-0-methyl-alpha-l-ribohexopyranosyl) oxyl) 6-o-methyl 3-oxo erythromycine, leur procede de preparation et leur application a la synthese de principes actifs de medicaments

Also Published As

Publication number Publication date
EP1132392B1 (de) 2004-03-03
EP1132392A1 (de) 2001-09-12
DK1132392T3 (da) 2004-06-07
DE60102171T2 (de) 2005-03-03
ES2214385T3 (es) 2004-09-16
US20020065235A1 (en) 2002-05-30
PT1132392E (pt) 2004-06-30
US6555524B2 (en) 2003-04-29
DE60102171D1 (de) 2004-04-08
CA2339051A1 (en) 2001-09-06
TR200400630T4 (tr) 2004-05-21
BR0100850A (pt) 2001-11-27
JP2001261694A (ja) 2001-09-26

Similar Documents

Publication Publication Date Title
DK1132392T3 (da) Ketolid-antibiotika
EA200100623A1 (ru) Кетолидные антибиотики
ATE344269T1 (de) Carbamat und carbazat ketolid antibiotika
BG105543A (en) Novel macrolide antibiotics
DE69917717D1 (de) C11-Carbamate von antibakteriellen Makroliden
DK1167376T3 (da) Makrolidantibiotika
YU66900A (sh) Derivati higromicina a
WO2002018353A3 (en) Oxazolidinone chemotherapeutic agents
YU64300A (sh) Derivati 2"-deoksi higromicina
AP2001002154A0 (en) Hygromycin a derivatives (changed by the ISA to read hygromycin a derivatives as antibacterial agents.
EA200201167A1 (ru) Производные гигромицина а для лечения бактериальных и протозойных инфекций
AP2002002492A0 (en) Hygromycin a prodrugs.

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification

Ref document number: 1132392

Country of ref document: EP

REN Ceased due to non-payment of the annual fee