ATE276252T1 - Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe - Google Patents

Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe

Info

Publication number
ATE276252T1
ATE276252T1 AT00993258T AT00993258T ATE276252T1 AT E276252 T1 ATE276252 T1 AT E276252T1 AT 00993258 T AT00993258 T AT 00993258T AT 00993258 T AT00993258 T AT 00993258T AT E276252 T1 ATE276252 T1 AT E276252T1
Authority
AT
Austria
Prior art keywords
substituents
c6alkyl
c6alkoxy
halogen
phenyl
Prior art date
Application number
AT00993258T
Other languages
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Maurizio Schwarzenbach
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE276252T1 publication Critical patent/ATE276252T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D275/00Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/44Acylated amino or imino radicals
    • C07D277/46Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT00993258T 1999-12-02 2000-11-30 Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe ATE276252T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH220799 1999-12-02
PCT/EP2000/012064 WO2001040223A2 (en) 1999-12-02 2000-11-30 Aminoheterocyclylamides as pesticides and antiparasitic agents

Publications (1)

Publication Number Publication Date
ATE276252T1 true ATE276252T1 (de) 2004-10-15

Family

ID=4228396

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00993258T ATE276252T1 (de) 1999-12-02 2000-11-30 Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe

Country Status (18)

Country Link
US (1) US6673820B2 (de)
EP (1) EP1254135B1 (de)
JP (1) JP2003515608A (de)
KR (1) KR100479137B1 (de)
CN (1) CN1196700C (de)
AT (1) ATE276252T1 (de)
AU (1) AU765618B2 (de)
BR (1) BR0016034A (de)
CA (1) CA2390113A1 (de)
DE (1) DE60013910T2 (de)
DK (1) DK1254135T3 (de)
ES (1) ES2228664T3 (de)
MX (1) MXPA02005428A (de)
NZ (1) NZ518931A (de)
PT (1) PT1254135E (de)
RU (1) RU2002117428A (de)
WO (1) WO2001040223A2 (de)
ZA (1) ZA200204337B (de)

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US7196106B2 (en) 2002-11-05 2007-03-27 Merck & Co., Inc Cyanothiophene derivatives, compositions containing such compounds and methods of use
JP2004269515A (ja) * 2003-02-18 2004-09-30 Nippon Nohyaku Co Ltd 置換複素環アミド誘導体、その中間体及び農園芸用薬剤並びにその使用方法
US20050085531A1 (en) * 2003-10-03 2005-04-21 Hodge Carl N. Thiophene-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof
NL2000351C2 (nl) 2005-12-22 2007-09-11 Pfizer Prod Inc Estrogeen-modulatoren.
US20100200021A1 (en) * 2006-02-17 2010-08-12 Nils Adey Slide Conditioning Systems and Methods
WO2008005764A2 (en) * 2006-06-30 2008-01-10 Fmc Corporation Novel zeta-cypermethrin composition
EP2560966B1 (de) 2010-03-30 2021-01-06 Verseon International Corporation Mehrfach substituierte aromatische verbindungen als thrombinhemmer
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
WO2011133920A1 (en) 2010-04-23 2011-10-27 Cytokinetics, Inc. Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use
AR081626A1 (es) 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
CN102067845B (zh) * 2011-01-31 2013-07-17 湖南大学 5-苄基-4-烷基-2-芳氨基噻唑作为制备杀虫剂的应用
US8759380B2 (en) 2011-04-22 2014-06-24 Cytokinetics, Inc. Certain heterocycles, compositions thereof, and methods for their use
JP6126115B2 (ja) * 2011-11-25 2017-05-10 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺内部寄生生物剤としてのアリールカルボキサミド類及びヘタリールカルボキサミド類の使用
EP2970141B1 (de) 2013-03-15 2020-02-26 Verseon Corporation Halogenpyrazole als thrombinhemmer
ES2853483T3 (es) 2013-03-15 2021-09-16 Verseon Int Corporation Compuestos aromáticos multisustituidos como inhibidores de la serina proteasa
BR112017004704A2 (pt) 2014-09-17 2018-01-23 Verseon Corp composto, composição farmacêutica, e, método para tratar uma doença ou distúrbio em um indivíduo
US10532995B2 (en) 2015-02-27 2020-01-14 Verseon Corporation Substituted pyrazole compounds as serine protease inhibitors
WO2017005717A1 (en) 2015-07-06 2017-01-12 Bayer Cropscience Aktiengesellschaft Heterocyclic compounds as pesticides
JP2020502168A (ja) * 2016-12-16 2020-01-23 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺有害生物剤としてのチアジアゾール誘導体
EP3558986A1 (de) 2016-12-22 2019-10-30 Bayer CropScience Aktiengesellschaft Substituierte 1,2,4-thiadiazolylpyrrolone und 1,2,4-thiadiazolylhydantoine sowie deren salze und ihre verwendung als herbizide wirkstoffe
BR112019012584A2 (pt) * 2016-12-22 2019-11-19 Bayer Ag heteroarilpirrolonas substituídas e sais das mesmas e uso das mesmas como substâncias ativas herbicidas
WO2019105875A1 (en) 2017-11-28 2019-06-06 Bayer Aktiengesellschaft Heterocyclic compounds as pesticides
US12030875B2 (en) 2018-09-07 2024-07-09 PIC Therapeutics, Inc. EIF4E inhibitors and uses thereof
AU2021230289A1 (en) 2020-03-03 2022-09-29 PIC Therapeutics, Inc. eIF4E inhibitors and uses thereof
WO2022194841A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194842A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194843A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2023020962A1 (en) 2021-08-17 2023-02-23 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
CN117794928A (zh) 2021-08-17 2024-03-29 拜耳公司 取代的1,2,4-噻二唑基烟酰胺、其盐或n-氧化物及其作为除草活性物质的用途
CN118159536A (zh) 2021-08-17 2024-06-07 拜耳公司 取代的1,2,4-噻二唑基烟酰胺、其盐或n-氧化物及其作为除草活性物质的用途
CN118019739A (zh) 2021-08-25 2024-05-10 皮克医疗公司 Eif4e抑制剂及其用途
JP2024534127A (ja) 2021-08-25 2024-09-18 ピク セラピューティクス, インコーポレイテッド eIF4E阻害剤及びその使用
EP4238972A1 (de) 2022-03-04 2023-09-06 Bayer AG Substituierte 1,2,4-thiadiazolyl-picolinamide, salze oder n-oxide davon und ihre verwendung als herbizide wirkstoffe
EP4238973A1 (de) 2022-03-04 2023-09-06 Bayer AG Substituierte 1,2,4-thiadiazolyl-nicotinamide, salze oder n-oxide davon und ihre verwendung als herbizide wirkstoffe

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DE1924830A1 (de) * 1968-07-06 1970-11-19 Merck Patent Gmbh Neues Verfahren zur Herstellung von 5-Acylamino-isothiazolderivaten
AU7103974A (en) * 1973-07-19 1976-01-15 Fmc Corp Herbicidal isothiazolylureas
US4966908A (en) * 1988-03-21 1990-10-30 Ciba-Geigy Corporation Isonicotinic acid amides for protecting plants against disease
EP0623282A1 (de) 1993-05-05 1994-11-09 Shell Internationale Researchmaatschappij B.V. Pestizide Verfahren und Verbindungen
GB9725298D0 (en) * 1997-11-28 1998-01-28 Zeneca Ltd Insecticidal thiazole derivatives
JP2000226389A (ja) * 1998-11-30 2000-08-15 Mitsubishi Chemicals Corp N−チアジアゾリルピラゾールカルボキサミド誘導体およびこれを有効成分とする殺虫、殺ダニ剤

Also Published As

Publication number Publication date
DK1254135T3 (da) 2005-01-17
CN1468235A (zh) 2004-01-14
WO2001040223A3 (en) 2001-12-20
AU765618B2 (en) 2003-09-25
CA2390113A1 (en) 2001-06-07
WO2001040223A2 (en) 2001-06-07
WO2001040223B1 (en) 2002-05-30
AU2838901A (en) 2001-06-12
JP2003515608A (ja) 2003-05-07
RU2002117428A (ru) 2003-12-20
NZ518931A (en) 2004-02-27
MXPA02005428A (es) 2002-11-29
EP1254135A2 (de) 2002-11-06
US20030148890A1 (en) 2003-08-07
ES2228664T3 (es) 2005-04-16
DE60013910T2 (de) 2005-09-29
BR0016034A (pt) 2002-07-30
PT1254135E (pt) 2005-03-31
DE60013910D1 (de) 2004-10-21
CN1196700C (zh) 2005-04-13
ZA200204337B (en) 2003-06-03
KR100479137B1 (ko) 2005-03-31
US6673820B2 (en) 2004-01-06
KR20020058064A (ko) 2002-07-12
EP1254135B1 (de) 2004-09-15

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