ATE279192T1 - Die verwendung eines benzimidazoles zur herstellung eines medikamentes zur krebsvorbeugung - Google Patents

Die verwendung eines benzimidazoles zur herstellung eines medikamentes zur krebsvorbeugung

Info

Publication number
ATE279192T1
ATE279192T1 AT00952534T AT00952534T ATE279192T1 AT E279192 T1 ATE279192 T1 AT E279192T1 AT 00952534 T AT00952534 T AT 00952534T AT 00952534 T AT00952534 T AT 00952534T AT E279192 T1 ATE279192 T1 AT E279192T1
Authority
AT
Austria
Prior art keywords
sub
carbon atoms
less
hydrogen
benzimidazole
Prior art date
Application number
AT00952534T
Other languages
English (en)
Inventor
James Berger Camden
Original Assignee
Uaf Technologies And Res Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Uaf Technologies And Res Llc filed Critical Uaf Technologies And Res Llc
Application granted granted Critical
Publication of ATE279192T1 publication Critical patent/ATE279192T1/de

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
AT00952534T 1999-08-13 2000-08-04 Die verwendung eines benzimidazoles zur herstellung eines medikamentes zur krebsvorbeugung ATE279192T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/374,717 US6423734B1 (en) 1999-08-13 1999-08-13 Method of preventing cancer
PCT/US2000/021381 WO2001012169A2 (en) 1999-08-13 2000-08-04 Method of cancer treatment

Publications (1)

Publication Number Publication Date
ATE279192T1 true ATE279192T1 (de) 2004-10-15

Family

ID=23477934

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00952534T ATE279192T1 (de) 1999-08-13 2000-08-04 Die verwendung eines benzimidazoles zur herstellung eines medikamentes zur krebsvorbeugung

Country Status (12)

Country Link
US (2) US6423734B1 (de)
EP (1) EP1202735B1 (de)
JP (1) JP2003506482A (de)
AT (1) ATE279192T1 (de)
AU (1) AU763311B2 (de)
CA (1) CA2380414C (de)
CO (1) CO5200778A1 (de)
DE (1) DE60014916T2 (de)
MX (1) MXPA02001571A (de)
NZ (1) NZ516766A (de)
PE (1) PE20010541A1 (de)
WO (1) WO2001012169A2 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6479526B1 (en) 1995-04-12 2002-11-12 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of viruses and cancers
US6506783B1 (en) * 1997-05-16 2003-01-14 The Procter & Gamble Company Cancer treatments and pharmaceutical compositions therefor
US6423734B1 (en) * 1999-08-13 2002-07-23 The Procter & Gamble Company Method of preventing cancer
DE60115069T2 (de) 2000-09-11 2006-08-03 Chiron Corp., Emeryville Chinolinonderivate als tyrosin-kinase inhibitoren
US6462062B1 (en) * 2000-09-26 2002-10-08 The Procter & Gamble Company Compounds and methods for use thereof in the treatment of cancer or viral infections
US6608096B1 (en) * 2000-09-26 2003-08-19 University Of Arizona Foundation Compounds and methods for use thereof in the treatment of cancer or viral infections
US6380232B1 (en) 2000-09-26 2002-04-30 The Procter & Gamble Company Benzimidazole urea derivatives, and pharmaceutical compositions and unit dosages thereof
AU2002239395A1 (en) * 2000-11-01 2002-06-03 The Procter And Gamble Company Hiv treatment with benzimidazoles
CZ20032691A3 (en) 2001-03-12 2004-04-14 Avanir Pharmaceuticals Benzimidazole compounds for modulating ige and inhibiting cellular proliferation
US20050038022A1 (en) * 2001-03-26 2005-02-17 Unisearch Limited Method for treatment of cancer and compositions for use therein
AU2002245927B2 (en) * 2001-03-26 2005-11-17 Pitney Pharmaceuticals Pty Limited Method for treatment of cancer and compositions for use therein
US20030158118A1 (en) * 2001-11-26 2003-08-21 Weidner Morten Sloth Combination of cimetidine and cysteine derivatives for treating cancer
AU2003220585A1 (en) * 2002-03-26 2003-10-13 Arizona Board of Regents on behalf of the University of Arizone Solubilization of weak bases
EP1539754A4 (de) 2002-08-23 2009-02-25 Novartis Vaccines & Diagnostic Benzimidazolchinolinone und deren verwendung
WO2004024655A2 (en) 2002-09-12 2004-03-25 Avanir Pharmaceuticals Phenyl-indole compounds for modulating ige and inhibiting cellular proliferation
TWI276631B (en) 2002-09-12 2007-03-21 Avanir Pharmaceuticals Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
MXPA05009564A (es) * 2003-03-12 2005-11-17 Univ Arizona Sales de bases debiles.
US20090286838A1 (en) * 2004-12-06 2009-11-19 Newsouth Innovations Pty Limited Treatment for cancer
US20060257317A1 (en) * 2005-05-04 2006-11-16 Duke University Combination therapy in the treatment of cancer
EP2465857B1 (de) 2005-05-17 2014-06-04 Novartis AG Verfahren zum Synthetisieren heterocyclischer Verbindungen
EP2432451A2 (de) * 2009-05-20 2012-03-28 Children's Medical Center Corporation Zusammensetzungen für die behandlung von metastasierendem krebs und anwendungsverfahren dafür

Family Cites Families (85)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2933502A (en) 1958-02-12 1960-04-19 Du Pont Benzimidazolone derivatives
US3010968A (en) 1959-11-25 1961-11-28 Du Pont Process for manufacture of certain alkyl esters of benzimidazole carbamic acids
NL134354C (de) 1963-05-23
US3499761A (en) 1964-07-20 1970-03-10 Gaf Corp Silver halide emulsions containing alkyl esters of benzimidazole carbamic acid antifogging agents
BE666795A (de) * 1964-08-04 1966-01-13
USRE28403E (en) 1964-08-04 1975-04-29 Butyl and n-propoxy-z-carbo- methoxyaminobenzimidazoles
US3541213A (en) 1966-05-06 1970-11-17 Du Pont Fungicidal and mite ovicidal substituted 2-aminobenzimidazoles
US3399212A (en) 1966-05-16 1968-08-27 Smith Kline French Lab Benzimidazole ureas
US3480642A (en) 1967-03-22 1969-11-25 Smithkline Corp Process for producing 2-carbalkoxyaminobenzimidazoles
US3881014A (en) 1968-11-05 1975-04-29 Bayer Ag N-tritylimidazoles for treating fungal infections
BE744970A (fr) 1969-01-28 1970-07-27 Lilly Co Eli Agents antiviraux et immuno-depresseurs
BE759337A (fr) 1969-11-24 1971-05-24 Lilly Co Eli Benzimidazol (2,1-b)-quinazolin (6h) ones qui sont des immuno-depresseurs, et nouvelles benzimidazo (2,1-b) quinazolin-12-(6h) ones
FR2046114A5 (en) 1970-01-30 1971-03-05 Dynachim Sarl Benzimidazole derivs anthelmintic, antifung - al bactericidal, aericidal, insecticidal, nema
US3956262A (en) 1970-12-09 1976-05-11 Beecham Group Limited Triazenoimidazoles
US3738995A (en) 1971-05-14 1973-06-12 Du Pont Solvent process for the preparation of 1 - carbamoyl-substituted 2 - benzimidazolecarbamates
DE2144505A1 (de) 1971-09-06 1973-03-15 Boehringer Sohn Ingelheim S-triazino- eckige klammer auf 1,2-a eckige klammer zu-benzimidazole
FR2155888A1 (en) 1971-10-13 1973-05-25 Agot Aime Solid anthelmintic composn - for more economical treatment of ruminants
DE2227919C2 (de) 1972-06-08 1982-12-23 Bayer Ag, 5090 Leverkusen Verfahren zur Herstellung von Benzimidazol-2-yl-carbaminsäure-methylester
DE2253324A1 (de) 1972-10-31 1974-05-09 Bayer Ag 1-alkoxycarbonyl-2- eckige klammer auf bis-(alkoxycarbonyl)-amino eckige klammer zu -benzimidazole, verfahren zu ihrer herstellung, sowie ihre verwendung als fungizide
US4046906A (en) 1973-04-21 1977-09-06 Hoechst Aktiengesellschaft Salts of alkyl 2-benzimidazole-carbamate
JPS5134161A (en) 1974-09-18 1976-03-23 Yoshitomi Pharmaceutical 22 benzuimidazoorukarubaminsanesuteru no seizoho
JPS5142565A (en) 1974-10-09 1976-04-10 Copal Co Ltd onnoff taimaa
US4001423A (en) 1975-06-20 1977-01-04 Dodds Dale I 2-(2-ethoxy)ethoxyethyl benzimidazolecarbamate
DE2527677A1 (de) 1975-06-21 1977-01-20 Bayer Ag Verfahren zur herstellung von 2,4- dioxo-1,2,3,4-tetrahydro-s-triazino- eckige klammer auf 1,2-a eckige klammer zu -benzimidazolen
US4086235A (en) 1976-04-12 1978-04-25 Syntex (U.S.A.) Inc. 5 (6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
IN159210B (de) 1982-01-11 1987-04-11 Council Scient Ind Res
IN158878B (de) 1982-07-15 1987-02-07 Council Scient Ind Res
HU193951B (en) 1985-03-11 1987-12-28 Richter Gedeon Vegyeszet Process for producing new sulfur-containing 5-substituted benzimidazol derivatives and pharmaceutical compositions containing them
JPS6323274A (ja) 1986-07-16 1988-01-30 Sony Corp デ−タ伝送方法
US4731366A (en) 1986-08-05 1988-03-15 Harbor Branch Oceanographic Institution, Inc. Discorhabdin compositions and their methods of use
GB2210875B (en) 1987-10-09 1991-05-29 Farmos Oy Aromatase inhibiting 4(5)-imidazoles
US5329012A (en) 1987-10-29 1994-07-12 The Research Foundation Of State University Of New York Bis(acyloxmethyl)imidazole compounds
US5114951A (en) 1989-04-11 1992-05-19 Burroughs Wellcome Company Agents for combating multiple drug resistance
US5149527A (en) 1990-09-18 1992-09-22 Oncotech, Inc. Immunopotentiating protocol for chemotherapy-responsive tumors
US5284662A (en) 1990-10-01 1994-02-08 Ciba-Geigy Corp. Oral osmotic system for slightly soluble active agents
GB9106278D0 (en) 1991-03-25 1991-05-08 Smithkline Beecham Plc Method of treatment
US5364875A (en) 1992-05-11 1994-11-15 The Du Pont Merck Pharmaceutical Company Imidazoles linked to bicyclic heterocyclic groups for the treatment of atherosclerosis
US5310748A (en) 1992-05-11 1994-05-10 The Du Pont Merck Pharmaceutical Company Imidazoles for the treatment of atherosclerosis
US5290801A (en) 1992-05-29 1994-03-01 The Du Pont Merck Pharmaceutical Company Benzimidazoles for the treatment of atherosclerosis
CA2140653A1 (en) 1992-08-12 1994-03-03 Irene Abraham Protein kinase inhibitors and related compounds combined with taxol
FR2703057B1 (fr) 1993-03-24 1995-06-16 Elysees Balzac Financiere Matériau alvéolaire cellulosique renfermant un agent biocide et procédé pour sa préparation.
RO118000B1 (ro) 1993-03-31 2002-12-30 Merck & Co Inc Metoda pentru tratamentul sida, prevenirea si tratamentul infectiei cu hiv sau inhibarea proteazei hiv si compozitie farmaceutica pentru aplicarea metodei
US5434163A (en) 1993-05-14 1995-07-18 The Medical College Of Pennsylvania Treatment of Cryptococcus neoformans infection
US5554373A (en) 1993-11-05 1996-09-10 Seabrook; Samuel G. Compositions containing anti-microbial agents and methods for making and using same
JP3213471B2 (ja) 1994-04-13 2001-10-02 ポーラ化成工業株式会社 薬効成分含有リポソーム製剤の製造方法
NZ305784A (en) 1995-04-12 2001-03-30 Procter & Gamble Benzimidazole containing medicaments for treating cancers, tumors and viral infections
US5656615A (en) 1995-04-12 1997-08-12 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of cancers and viruses in mammals
ZA962880B (en) 1995-04-12 1997-03-17 Procter & Gamble A pharmaceutical composition for inhibiting the growth of viruses and cancers
US6262093B1 (en) * 1995-04-12 2001-07-17 The Proctor & Gamble Company Methods of treating cancer with benzimidazoles
ZA962879B (en) * 1995-04-12 1997-03-17 Procter & Gamble A pharmaceutical composition for inhibiting the growth of viruses and cancers
US6177460B1 (en) * 1995-04-12 2001-01-23 The Procter & Gamble Company Method of treatment for cancer or viral infections
AU714056B2 (en) * 1995-04-12 1999-12-16 Uaf Technologies And Research Llc A pharmaceutical composition containing N-chlorophenylcarbamates and N-chlorophenylthiocarbamates for inhibiting the growth of viruses and cancers
US5665713A (en) 1995-04-12 1997-09-09 Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of viruses and cancers
US5629341A (en) 1995-04-12 1997-05-13 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of viruses and cancers
US5665751A (en) 1995-06-07 1997-09-09 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of cancers
MX9707809A (es) 1995-06-07 1998-01-31 Procter & Gamble Una composicion farmaceutica que contiene bencimidazol para inhibir el crecimiento de canceres.
US5770616A (en) * 1995-06-07 1998-06-23 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of cancers
US20010039291A1 (en) * 1995-06-07 2001-11-08 The Procter & Gamble Company Compositions and methods of treatment for cancer or viral infections
US6265427B1 (en) * 1995-06-07 2001-07-24 The Proctor & Gamble Company Pharmaceutical composition for the method of treating leukemia
CN1186433A (zh) 1995-06-07 1998-07-01 普罗克特和甘保尔公司 苯并咪唑类在制备白血病治疗药物上的应用
US6200992B1 (en) * 1995-06-07 2001-03-13 The Procter & Gamble Company Pharmaceutical composition for inhibiting the growth of cancers
KR19990036137A (ko) 1995-08-03 1999-05-25 데이비드 엠 모이어 암 성장을 억제하기 위한 그리세오풀빈의 용도
MX9707808A (es) * 1995-08-04 1998-01-31 Procter & Gamble Una composicion farmaceutica que contiene n-clorofenilcarbamatos y n-clorofiniltiocarbamatos para inhibir el crecimiento de virus y canceres.
US6686391B2 (en) * 1995-08-04 2004-02-03 University Of Arizona Foundation N-chlorophenylcarbamate and N-chlorophenylthiocarbamate compositions
US5908855A (en) 1996-07-16 1999-06-01 The Procter & Gamble Company Compositions for treating viral infections
EP0841921A2 (de) 1995-08-04 1998-05-20 The Procter & Gamble Company Verwendung von fluoconazol zur hemmung des krebswachtums
AU6966696A (en) 1995-10-05 1997-04-28 Warner-Lambert Company Method for treating and preventing inflammation and atherosclerosis
US5900429A (en) * 1997-01-28 1999-05-04 The Procter & Gamble Company Method for inhibiting the growth of cancers
PE11499A1 (es) 1997-05-16 1999-03-01 Procter & Gamble Tratamiento del hiv y cancer
US6506783B1 (en) 1997-05-16 2003-01-14 The Procter & Gamble Company Cancer treatments and pharmaceutical compositions therefor
US6245789B1 (en) 1998-05-19 2001-06-12 The Procter & Gamble Company HIV and viral treatment
ATE429813T1 (de) 1998-10-09 2009-05-15 Gen Mills Inc Verkapselung empfindlicher flüssiger komponenten in eine matrix zur gewinnung diskreter lagerbeständiger partikel
US6211177B1 (en) 1998-11-24 2001-04-03 Cell Pathways, Inc. Method for treating neoplasia by exposure to substituted 2-aryl-benzimidazole derivatives
US20010053773A1 (en) * 1998-12-22 2001-12-20 The Procter & Gamble Company Method for inhibiting the growth of cancers
US6294192B1 (en) 1999-02-26 2001-09-25 Lipocine, Inc. Triglyceride-free compositions and methods for improved delivery of hydrophobic therapeutic agents
US6136835A (en) * 1999-05-17 2000-10-24 The Procter & Gamble Company Methods of treatment for viral infections
US6423734B1 (en) 1999-08-13 2002-07-23 The Procter & Gamble Company Method of preventing cancer
US20010047021A1 (en) 2000-04-28 2001-11-29 The Procter & Gamble Company Cancer treatment
US6384049B1 (en) * 2000-05-25 2002-05-07 The Procter & Gamble Company Cancer treatment
US6290929B1 (en) * 2000-07-28 2001-09-18 The Procter & Gamble Company Cancer treatment
US6518269B1 (en) 2000-07-28 2003-02-11 University Of Arizona Foundation Cancer treatment
US6407105B1 (en) * 2000-09-26 2002-06-18 The Procter & Gamble Company Compounds and methods for use thereof in the treatment of cancer or viral infections
AU2001292796B2 (en) 2000-09-26 2005-12-22 Uaf Technologies And Research Llc Benzimidazoles and methods for use thereof in the treatment of cancer or viral infections
US6380232B1 (en) * 2000-09-26 2002-04-30 The Procter & Gamble Company Benzimidazole urea derivatives, and pharmaceutical compositions and unit dosages thereof
AU2002239395A1 (en) 2000-11-01 2002-06-03 The Procter And Gamble Company Hiv treatment with benzimidazoles

Also Published As

Publication number Publication date
DE60014916T2 (de) 2005-04-07
US6906091B2 (en) 2005-06-14
US6423734B1 (en) 2002-07-23
EP1202735A2 (de) 2002-05-08
AU6521000A (en) 2001-03-13
CA2380414C (en) 2006-06-13
AU763311B2 (en) 2003-07-17
CA2380414A1 (en) 2001-02-22
EP1202735B1 (de) 2004-10-13
JP2003506482A (ja) 2003-02-18
PE20010541A1 (es) 2001-05-16
DE60014916D1 (de) 2004-11-18
NZ516766A (en) 2003-11-28
US20030032664A1 (en) 2003-02-13
WO2001012169A2 (en) 2001-02-22
MXPA02001571A (es) 2003-10-14
WO2001012169A3 (en) 2002-02-14
CO5200778A1 (es) 2002-09-27

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