ATE287714T1 - Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen - Google Patents

Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen

Info

Publication number
ATE287714T1
ATE287714T1 AT00917940T AT00917940T ATE287714T1 AT E287714 T1 ATE287714 T1 AT E287714T1 AT 00917940 T AT00917940 T AT 00917940T AT 00917940 T AT00917940 T AT 00917940T AT E287714 T1 ATE287714 T1 AT E287714T1
Authority
AT
Austria
Prior art keywords
inhibiting compounds
retroviral protease
protease inhibiting
pharmaceutical emulsions
emulsions
Prior art date
Application number
AT00917940T
Other languages
English (en)
Inventor
Youmin Wang
Walter Morozowich
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of ATE287714T1 publication Critical patent/ATE287714T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT00917940T 1999-03-31 2000-03-22 Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen ATE287714T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12702699P 1999-03-31 1999-03-31
PCT/US2000/006681 WO2000057885A1 (en) 1999-03-31 2000-03-22 Pharmaceutical emulsions for retroviral protease inhibitors

Publications (1)

Publication Number Publication Date
ATE287714T1 true ATE287714T1 (de) 2005-02-15

Family

ID=22427949

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00917940T ATE287714T1 (de) 1999-03-31 2000-03-22 Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen

Country Status (8)

Country Link
EP (1) EP1165091B1 (de)
JP (1) JP4638053B2 (de)
AT (1) ATE287714T1 (de)
AU (1) AU3883700A (de)
DE (1) DE60017720T2 (de)
ES (1) ES2234582T3 (de)
PT (1) PT1165091E (de)
WO (1) WO2000057885A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0000774D0 (sv) 2000-03-08 2000-03-08 Astrazeneca Ab New formulation
SE0102993D0 (sv) * 2001-09-07 2001-09-07 Astrazeneca Ab New self emulsifying drug delivery system
CA3108961C (en) 2008-08-01 2024-07-02 Hospira, Inc. Pharmaceutical compositions comprising clevidipine and methods for producing low concentrations of impurities thereof
CN102627654B (zh) * 2012-05-08 2013-11-27 山东大学 含异山梨醇结构单元的hiv-1蛋白酶抑制剂及其制备方法与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0999838T3 (da) * 1997-07-29 2002-07-08 Upjohn Co Selv-emulgerende formulering for lipofile forbindelser
JP4524367B2 (ja) * 1997-07-29 2010-08-18 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 自己乳化性処方形態の酸性親油性化合物用の医薬組成物

Also Published As

Publication number Publication date
DE60017720T2 (de) 2006-01-12
JP2002540158A (ja) 2002-11-26
JP4638053B2 (ja) 2011-02-23
WO2000057885A1 (en) 2000-10-05
AU3883700A (en) 2000-10-16
ES2234582T3 (es) 2005-07-01
PT1165091E (pt) 2005-05-31
EP1165091B1 (de) 2005-01-26
EP1165091A1 (de) 2002-01-02
DE60017720D1 (de) 2005-03-03

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