ATE287714T1 - Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen - Google Patents

Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen

Info

Publication number
ATE287714T1
ATE287714T1 AT00917940T AT00917940T ATE287714T1 AT E287714 T1 ATE287714 T1 AT E287714T1 AT 00917940 T AT00917940 T AT 00917940T AT 00917940 T AT00917940 T AT 00917940T AT E287714 T1 ATE287714 T1 AT E287714T1
Authority
AT
Austria
Prior art keywords
inhibiting compounds
retroviral protease
protease inhibiting
pharmaceutical emulsions
emulsions
Prior art date
Application number
AT00917940T
Other languages
English (en)
Inventor
Youmin Wang
Walter Morozowich
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of ATE287714T1 publication Critical patent/ATE287714T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT00917940T 1999-03-31 2000-03-22 Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen ATE287714T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12702699P 1999-03-31 1999-03-31
PCT/US2000/006681 WO2000057885A1 (en) 1999-03-31 2000-03-22 Pharmaceutical emulsions for retroviral protease inhibitors

Publications (1)

Publication Number Publication Date
ATE287714T1 true ATE287714T1 (de) 2005-02-15

Family

ID=22427949

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00917940T ATE287714T1 (de) 1999-03-31 2000-03-22 Pharmazeutische emulsionen für retroviral- protease hemmende verbindungen

Country Status (8)

Country Link
EP (1) EP1165091B1 (de)
JP (1) JP4638053B2 (de)
AT (1) ATE287714T1 (de)
AU (1) AU3883700A (de)
DE (1) DE60017720T2 (de)
ES (1) ES2234582T3 (de)
PT (1) PT1165091E (de)
WO (1) WO2000057885A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0000774D0 (sv) 2000-03-08 2000-03-08 Astrazeneca Ab New formulation
SE0102993D0 (sv) * 2001-09-07 2001-09-07 Astrazeneca Ab New self emulsifying drug delivery system
EP2320740B1 (de) * 2008-08-01 2014-03-26 The Medicines Company Pharmazeutische zusammensetzungen von clividipine und verfahren zur herstellung von konzentrationen daraus mit geringem verunreinigungsgrad
CN102627654B (zh) * 2012-05-08 2013-11-27 山东大学 含异山梨醇结构单元的hiv-1蛋白酶抑制剂及其制备方法与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1112927C (zh) * 1997-07-29 2003-07-02 法玛西雅厄普约翰美国公司 自体乳化剂形式的酸性亲脂性化合物的药物组合物
KR100509130B1 (ko) * 1997-07-29 2005-08-18 파마시아 앤드 업존 캄파니 엘엘씨 친지성 화합물의 자가유화 제제

Also Published As

Publication number Publication date
JP2002540158A (ja) 2002-11-26
EP1165091B1 (de) 2005-01-26
WO2000057885A1 (en) 2000-10-05
ES2234582T3 (es) 2005-07-01
DE60017720T2 (de) 2006-01-12
EP1165091A1 (de) 2002-01-02
PT1165091E (pt) 2005-05-31
DE60017720D1 (de) 2005-03-03
JP4638053B2 (ja) 2011-02-23
AU3883700A (en) 2000-10-16

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