ATE296827T1 - Heteropolycyclische inhibitoren - Google Patents

Heteropolycyclische inhibitoren

Info

Publication number
ATE296827T1
ATE296827T1 AT01955500T AT01955500T ATE296827T1 AT E296827 T1 ATE296827 T1 AT E296827T1 AT 01955500 T AT01955500 T AT 01955500T AT 01955500 T AT01955500 T AT 01955500T AT E296827 T1 ATE296827 T1 AT E296827T1
Authority
AT
Austria
Prior art keywords
heteropolycyclic
inhibitors
administering
compound
formula
Prior art date
Application number
AT01955500T
Other languages
English (en)
Inventor
Zaihui Zhang
Xinyao Du
Greg Chopiuk
Serguei Sviridov
Original Assignee
Quadra Logic Tech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Quadra Logic Tech Inc filed Critical Quadra Logic Tech Inc
Application granted granted Critical
Publication of ATE296827T1 publication Critical patent/ATE296827T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT01955500T 2000-07-06 2001-07-06 Heteropolycyclische inhibitoren ATE296827T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US61103800A 2000-07-06 2000-07-06
PCT/IB2001/001519 WO2002002562A2 (en) 2000-07-06 2001-07-06 Heteropolycyclic inhibitors

Publications (1)

Publication Number Publication Date
ATE296827T1 true ATE296827T1 (de) 2005-06-15

Family

ID=24447360

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01955500T ATE296827T1 (de) 2000-07-06 2001-07-06 Heteropolycyclische inhibitoren

Country Status (8)

Country Link
US (2) US6514972B2 (de)
EP (1) EP1296985B1 (de)
AT (1) ATE296827T1 (de)
AU (1) AU2001277659A1 (de)
CA (1) CA2414885A1 (de)
DE (1) DE60111228T2 (de)
ES (1) ES2243527T3 (de)
WO (1) WO2002002562A2 (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002002562A2 (en) * 2000-07-06 2002-01-10 Kinetek Pharmaceuticals, Inc. Heteropolycyclic inhibitors
US8715708B2 (en) * 2005-08-31 2014-05-06 University Of Maryland Cyclic acetal biomaterials
US7462615B2 (en) * 2005-12-08 2008-12-09 Hybrigenics Sa Inhibitors of cysteine proteases, the pharmaceutical compositions thereof and their therapeutic applications
MX2008007195A (es) * 2005-12-08 2008-09-10 Hybrigenics Sa Inhibidores de proteasas de cisteina, composiciones farmaceuticas de las mismas y sus aplicaciones terapeuticas.
EP1798232A1 (de) * 2005-12-08 2007-06-20 Hybrigenics S.A. Cysteine Proteasehemmer, deren pharmazeutische Zusammensetzungen und therapeutische Anwendungen
US7875613B2 (en) * 2006-10-30 2011-01-25 Hybrigenics Sa Tetracyclic inhibitors of cysteine proteases, the pharmaceutical compositions thereof and their therapeutic applications
EP1918292A1 (de) * 2006-10-30 2008-05-07 Hybrigenics S.A. Tetrazyklische Inhibitoren für Cysteinproteasen, pharmazeutische Zubereitungen und therapeutische Anwendungen
MX2009004517A (es) * 2006-10-30 2009-05-13 Hybrigenics Sa Nuevos inhibidores tetraciclicos de las proteasas de cisteina, las composiciones farmaceuticas de las mismas y sus aplicaciones terapeuticas.
WO2012006104A2 (en) * 2010-06-28 2012-01-12 Academia Sinica, Taiwan Compounds and methods for treating tuberculosis infection
CN103520165A (zh) * 2013-10-31 2014-01-22 华东理工大学 茚并三嗪类化合物作为依赖nad(p)h的醌氧化还原酶底物的用途
WO2016187046A1 (en) * 2015-05-15 2016-11-24 Indiana University Research & Technology Corporation Survivin-targeting anti-tumor agents and uses thereof
CN105061360B (zh) * 2015-07-28 2018-06-19 首都师范大学 一种3,4-二氨基-1,2,5-噻二唑的提纯方法
AU2019351124A1 (en) * 2018-09-28 2021-05-20 Acucela Inc. Inhibitors of VAP-1
EP3856176A4 (de) 2018-09-28 2022-05-04 Acucela Inc. Inhibitoren von vap-1
CN113368080B (zh) * 2020-02-25 2023-11-17 香港中文大学 稳定的、生物粘附的、扩散限制性团聚体
WO2022103827A1 (en) * 2020-11-10 2022-05-19 New Mexico Tech University Research Park Corporation Kp372-1-induced dna damage as a chemotherapeutic approach to treat cancer

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4159375A (en) * 1978-08-24 1979-06-26 American Cyanamid Company 6- AND 7-Aryl-1,2,4-triazolo[4,3-b]-1,2,4-triazines
US4405619A (en) * 1981-09-02 1983-09-20 Diamond Shamrock Corporation Antiinflammatory substituted-1,2,4-triazolo[4,3-b]-1,2,4-triazines
GB8826237D0 (en) 1988-11-09 1988-12-14 Univ Belfast Fingerprint reagent
WO1995024190A2 (en) 1994-03-07 1995-09-14 Sugen, Inc. Receptor tyrosine kinase inhibitors for inhibiting cell proliferative disorders and compositions thereof
WO2001079209A2 (en) * 2000-04-13 2001-10-25 Millennium Pharmaceuticals, Inc. Diazafluorenone il-8 antagonists
WO2002002562A2 (en) * 2000-07-06 2002-01-10 Kinetek Pharmaceuticals, Inc. Heteropolycyclic inhibitors

Also Published As

Publication number Publication date
AU2001277659A1 (en) 2002-01-14
US20030144294A1 (en) 2003-07-31
EP1296985A2 (de) 2003-04-02
WO2002002562A2 (en) 2002-01-10
EP1296985B1 (de) 2005-06-01
US7196083B2 (en) 2007-03-27
US20020035251A1 (en) 2002-03-21
WO2002002562A3 (en) 2002-05-02
DE60111228T2 (de) 2006-03-16
DE60111228D1 (de) 2005-07-07
ES2243527T3 (es) 2005-12-01
CA2414885A1 (en) 2002-01-10
US6514972B2 (en) 2003-02-04

Similar Documents

Publication Publication Date Title
DE60111228D1 (de) Heteropolycyclische inhibitoren
DK1223980T3 (da) Anvendelse af CSF-1-inhibitorer
CY1108738T1 (el) Θεραπευτικοι παραγοντες χρησιμοι για την αγωγη του πονου
SE0000540D0 (sv) New compounds
DE60317198D1 (de) Proteinkinaseinhibitoren
DE60331187D1 (de) Kinaseinhibitoren
DE60335359D1 (de) Phthalazinonderivate
EA200300906A1 (ru) Новые спиротрициклические производные и их применение в качестве ингибиторов фосфодиэстеразы-7
GB9801690D0 (en) Therapeutic agents
BG106585A (en) Kinase inhibitors as therapeutic agents
CY1107634T1 (el) Φαρμακευτικη συνθεση
EA200200769A1 (ru) Ингибиторы гиразы и их применение
CY1111396T1 (el) Ρινικη χορηγηση μετοκλοπραμιδης για την αγωγη της γαστροπαρεσης
SE0104248D0 (sv) Method of treatment
DK1458393T3 (da) Substituerede diketopiperaziner som oxytocinantagonister
HRP20090159T1 (en) Use of glucosidase inhibitors for therapy of mucovisidosis
GB9903403D0 (en) Substituted stilbene compounds with vascular damaging activity
MY143245A (en) 4- 2-(cycloalkylamino)pyrimidin-4-yl-(phenyl)-imidazolin-2-one derivatives as p38 map-kinase inhibitors for the treatment of inflammatory diseases
SE0004827D0 (sv) Therapeutic compounds
MXPA03000337A (es) Inhibidores de trombina que comprenden un grupo aminoisoquinolina.
MXPA05003909A (es) Compuestos de benzopiranona, composiciones de los mismos, y metodos para el tratamiento o prevencion del cancer.
DE60117783D1 (de) Naphthamidin-urokinasinhibitoren
AU2002211217A1 (en) Method of treating stroke
DE60108873D1 (de) Nicht-antibakterielle tetrazykline als anti-pilz medikamente
DK1553938T3 (da) Anvendelse af epothilonderivater til behandling af hyperparathyroidisme

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification

Ref document number: 1296985

Country of ref document: EP

REN Ceased due to non-payment of the annual fee