ATE308343T1 - Trägerhilfstoff - Google Patents

Trägerhilfstoff

Info

Publication number: ATE308343T1
Authority: AT; Austria
Prior art keywords: carrier aid; aid; carrier; whiteness; trehalose
Prior art date: 1998-07-15

Application number

AT99929812T

Other languages

English (en)

Inventor

Kazuhiro Oobae

Etsuo Kamada

Shun Ichi Gomi

Original Assignee

Asahi Kasei Chemicals Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-07-15

Filing date

1999-07-13

Publication date

2005-11-15

1999-07-13 Application filed by Asahi Kasei Chemicals Corp filed Critical Asahi Kasei Chemicals Corp

2005-11-15 Application granted granted Critical

2005-11-15 Publication of ATE308343T1 publication Critical patent/ATE308343T1/de

Links

239000002245 particle Substances 0.000 abstract 2
HDTRYLNUVZCQOY-UHFFFAOYSA-N α-D-glucopyranosyl-α-D-glucopyranoside Natural products OC1C(O)C(O)C(CO)OC1OC1C(O)C(O)C(O)C(CO)O1 HDTRYLNUVZCQOY-UHFFFAOYSA-N 0.000 abstract 1
HDTRYLNUVZCQOY-WSWWMNSNSA-N Trehalose Natural products O[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@@H]1O[C@@H]1[C@H](O)[C@@H](O)[C@@H](O)[C@@H](CO)O1 HDTRYLNUVZCQOY-WSWWMNSNSA-N 0.000 abstract 1
HDTRYLNUVZCQOY-LIZSDCNHSA-N alpha,alpha-trehalose Chemical compound O[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@@H]1O[C@@H]1[C@H](O)[C@@H](O)[C@H](O)[C@@H](CO)O1 HDTRYLNUVZCQOY-LIZSDCNHSA-N 0.000 abstract 1
239000000546 pharmaceutical excipient Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
Oil, Petroleum & Natural Gas (AREA)
General Chemical & Material Sciences (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Detergent Compositions (AREA)
Crystals, And After-Treatments Of Crystals (AREA)
Control And Other Processes For Unpacking Of Materials (AREA)
Glass Compositions (AREA)

AT99929812T 1998-07-15 1999-07-13 Trägerhilfstoff ATE308343T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP20029598		1998-07-15
JP32356098		1998-11-13
PCT/JP1999/003775 WO2000003735A1 (fr)	1998-07-15	1999-07-13	Excipient

Publications (1)

Publication Number	Publication Date
ATE308343T1 true ATE308343T1 (de)	2005-11-15

Family

ID=26512084

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99929812T ATE308343T1 (de)	1998-07-15	1999-07-13	Trägerhilfstoff

Country Status (10)

Country	Link
US (1)	US6699845B2 (de)
EP (1)	EP1097722B1 (de)
JP (1)	JP4748627B2 (de)
KR (1)	KR100421264B1 (de)
CN (1)	CN1185013C (de)
AT (1)	ATE308343T1 (de)
AU (1)	AU743109B2 (de)
CA (1)	CA2337015C (de)
DE (1)	DE69928110T2 (de)
WO (1)	WO2000003735A1 (de)

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US7407955B2 (en)	2002-08-21	2008-08-05	Boehringer Ingelheim Pharma Gmbh & Co., Kg	8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US20040131672A1 (en) *	2003-01-07	2004-07-08	Nilobon Podhipleux	Direct compression pharmaceutical composition containing a pharmaceutically active ingredient with poor flowing properties
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AU2004224492B2 (en) *	2003-03-26	2008-10-09	Kabushiki Kaisha Hayashibara Seibutsu Kagaku Kenkyujo	Method of powdering nonsugar component and powdering base
DE102004054054A1 (de)	2004-11-05	2006-05-11	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
JP2007131587A (ja) *	2005-11-11	2007-05-31	Activas Pharma:Kk	キノリノン誘導体を有効成分とする医薬組成物、及びその製造方法
EA015035B1 (ru) *	2005-12-07	2011-04-29	Никомед Фарма Ас	Предварительно уплотненные кальцийсодержащие композиции
CN100391541C (zh) *	2006-03-16	2008-06-04	南台科技大学	以胶质类食材制造赋形剂的方法
CA2650498A1 (en) *	2006-03-31	2007-10-11	Rubicon Research Private Limited	Orally disintegrating tablets
PE20080251A1 (es)	2006-05-04	2008-04-25	Boehringer Ingelheim Int	Usos de inhibidores de dpp iv
BRPI0711558A2 (pt)	2006-05-04	2011-11-08	Boeringer Ingelheim Internat Gmbh	polimorfos
EP1852108A1 (de)	2006-05-04	2007-11-07	Boehringer Ingelheim Pharma GmbH & Co.KG	Zusammensetzungen von DPP-IV-Inhibitoren
WO2008001734A1 (en) *	2006-06-27	2008-01-03	Daiichi Sankyo Company, Limited	Compressed preparation
WO2008079342A2 (en) *	2006-12-21	2008-07-03	Mallinckrodt Inc.	Composition of and method for preparing orally disintegrating tablets
PE20140960A1 (es)	2008-04-03	2014-08-15	Boehringer Ingelheim Int	Formulaciones que comprenden un inhibidor de dpp4
BRPI0916997A2 (pt)	2008-08-06	2020-12-15	Boehringer Ingelheim International Gmbh	Inibidor de dpp-4 e seu uso
US20200155558A1 (en)	2018-11-20	2020-05-21	Boehringer Ingelheim International Gmbh	Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
JP5344938B2 (ja) *	2009-01-29	2013-11-20	旭化成ケミカルズ株式会社	崩壊性固形製剤
EA034869B1 (ru)	2009-11-27	2020-03-31	Бёрингер Ингельхайм Интернациональ Гмбх	Лечение генотипированных пациентов с диабетом ингибиторами дпп-4, такими как линаглиптин
MX341025B (es)	2010-05-05	2016-08-04	Boehringer Ingelheim Int Gmbh *	Terapia de combinacion.
US9034883B2 (en)	2010-11-15	2015-05-19	Boehringer Ingelheim International Gmbh	Vasoprotective and cardioprotective antidiabetic therapy
AU2012310757B2 (en) *	2011-09-21	2016-05-12	Nagase Viita Co., Ltd.	Production method for powder containing crystalline alpha, alpha-trehalose dihydrate
US9522964B2 (en) *	2012-04-03	2016-12-20	Development, Inc.	Micronized starch and methods for manufacturing same
US20130303554A1 (en)	2012-05-14	2013-11-14	Boehringer Ingelheim International Gmbh	Use of a dpp-4 inhibitor in sirs and/or sepsis
JP6224084B2 (ja)	2012-05-14	2017-11-01	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	糸球体上皮細胞関連障害及び／又はネフローゼ症候群の治療に用いるｄｐｐ−４阻害薬としてのキサンチン誘導体
CN109310697A (zh)	2016-06-10	2019-02-05	勃林格殷格翰国际有限公司	利格列汀和二甲双胍的组合
AU2018344621B8 (en)	2017-10-03	2020-07-23	Mizkan Holdings Co., Ltd.	Composition containing fine food particulate complexes, and method for producing same
KR20210052281A (ko)	2019-10-29	2021-05-10	신에쓰 가가꾸 고교 가부시끼가이샤	캡슐 충전용 조성물 및 이것을 사용한 캡슐 제제의 제조 방법 그리고 캡슐 제제
KR102848723B1 (ko)	2025-04-18	2025-08-21	주식회사 탑시스템	축전부의 방열을 위한 대면적 히트싱크를 갖는 태양광 발전부가 구비된 가로등

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US4678812A (en)	1986-05-30	1987-07-07	E. I. Du Pont De Nemours And Company	Trehalose as stabilizer and tableting excipient
US4762857A (en)	1986-05-30	1988-08-09	E. I. Du Pont De Nemours And Company	Trehalose as stabilizer and tableting excipient
JP3069458B2 (ja)	1992-01-29	2000-07-24	武田薬品工業株式会社	口腔内崩壊型錠剤およびその製造法
EP0627218B1 (de)	1992-02-18	2001-12-19	Nippon Shinyaku Company, Limited	Verfahren zur Herstellung von schnelllöslicher Tabletten und schnelllöslichen Tablette beinhaltend Xylitol
JPH069382A (ja) *	1992-04-17	1994-01-18	Takeda Chem Ind Ltd	安定化された固型製剤およびその製造方法
DK0606753T3 (da)	1992-12-28	2000-02-21	Hayashibara Biochem Lab	Ikke-reducerende saccharid-dannende enzym og fremstilling og anvendelser deraf
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JP3534130B2 (ja) *	1994-03-01	2004-06-07	旭化成ケミカルズ株式会社	医薬品組成物
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JP3616166B2 (ja)	1994-07-19	2005-02-02	株式会社林原生物化学研究所	トレハロースとその製造方法並びに用途
JP2919771B2 (ja)	1995-04-17	1999-07-19	佐藤製薬株式会社	速溶解性錠剤の製造方法及び該製造方法により製造した速溶解性錠剤
JP3418274B2 (ja)	1995-06-05	2003-06-16	日本化薬株式会社	口腔内感触の良好な錠剤
JPH0948726A (ja)	1995-08-07	1997-02-18	Tanabe Seiyaku Co Ltd	口腔内速崩壊性製剤およびその製法
WO1997009037A1 (fr)	1995-09-07	1997-03-13	Otsuka Pharmaceutical Co., Ltd.	Preparation effervescente se presentant sous forme de comprimes produits a basse pression
JP3624038B2 (ja) *	1995-12-11	2005-02-23	株式会社林原生物化学研究所	糖衣固形物及びその製造方法
BR9714509A (pt) *	1996-02-09	2000-03-21	Quadrant Holdings Cambridge	Formulações sólidas contendo trealose
JPH09316006A (ja)	1996-05-29	1997-12-09	Yatsuken:Kk	口腔内溶解性固形製剤
PT914818E (pt)	1996-06-14	2005-08-31	Kyowa Hakko Kogyo Kk	Comprimido de desintegracao rapida por via intraoral
GB9616536D0 (en) *	1996-08-06	1996-09-25	Quadrant Holdings Cambridge	Co-amoxiclav dosage form
TW527195B (en) *	1997-10-09	2003-04-11	Ssp Co Ltd	Fast-soluble solid pharmaceutical combinations
JPH11116464A (ja)	1997-10-09	1999-04-27	Ss Pharmaceut Co Ltd	迅速溶解性固形製剤およびその製造法

1999
- 1999-07-13 CN CNB998086274A patent/CN1185013C/zh not_active Expired - Lifetime
- 1999-07-13 JP JP2000559869A patent/JP4748627B2/ja not_active Expired - Lifetime
- 1999-07-13 EP EP99929812A patent/EP1097722B1/de not_active Expired - Lifetime
- 1999-07-13 KR KR10-2001-7000538A patent/KR100421264B1/ko not_active Expired - Lifetime
- 1999-07-13 AU AU46516/99A patent/AU743109B2/en not_active Expired
- 1999-07-13 CA CA002337015A patent/CA2337015C/en not_active Expired - Lifetime
- 1999-07-13 DE DE69928110T patent/DE69928110T2/de not_active Expired - Lifetime
- 1999-07-13 AT AT99929812T patent/ATE308343T1/de not_active IP Right Cessation
- 1999-07-13 WO PCT/JP1999/003775 patent/WO2000003735A1/ja not_active Ceased
2001
- 2001-01-12 US US09/759,104 patent/US6699845B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
DE69928110D1 (de)	2005-12-08
AU743109B2 (en)	2002-01-17
CA2337015A1 (en)	2000-01-27
US20020042393A1 (en)	2002-04-11
EP1097722B1 (de)	2005-11-02
CN1309570A (zh)	2001-08-22
DE69928110T2 (de)	2006-07-27
WO2000003735A1 (fr)	2000-01-27
JP4748627B2 (ja)	2011-08-17
US6699845B2 (en)	2004-03-02
EP1097722A1 (de)	2001-05-09
KR20010071883A (ko)	2001-07-31
KR100421264B1 (ko)	2004-03-18
CA2337015C (en)	2004-09-07
AU4651699A (en)	2000-02-07
CN1185013C (zh)	2005-01-19
EP1097722A4 (de)	2002-03-20

Legal Events

Date	Code	Title	Description
2006-05-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
EP1097722A4 (de)	2002-03-20	Trägerhilfstoff
ATE419653T1 (de)	2009-01-15	Elektrolumineszierende anordnungen
EA199900318A1 (ru)	1999-12-29	Способ производства гранул цеолита х с низким содержанием двуокиси кремния с низким содержанием инертного связующего
MY111172A (en)	1999-09-30	Perfume particles.
MY121397A (en)	2006-01-28	Ziprasidone formulations
BG101893A (en)	1999-01-29	Nodulosporic acid derivatives
IL132238A0 (en)	2001-03-19	Fungicidal trifluromethylalkylamino - triazolopyrimidines
GR3025639T3 (en)	1998-03-31	Porous inorganic ultrasound contrast agents
ATE504562T1 (de)	2011-04-15	7-, 8- und 9-substitutierte tetracyclinverbindungen
AU5792690A (en)	1991-02-07	Aqeous pharmaceutical suspension for substantially water insoluble pharmaceutical actives
EP1435395A4 (de)	2005-04-20	Eisenmetallgranulat
DK1083151T3 (da)	2002-05-06	Pyrogent fremstillet aluminiumoxid
MY103969A (en)	1993-10-30	Detergent composition containing perfume
ZA963392B (en)	1996-09-06	Triggered active packagig material
HUT73158A (en)	1996-06-28	Insecticidal and acaricidal suspension concentrate containing arylpyrrole derivatives
WO1996019686A3 (en)	1996-10-17	Ferrofluid having oxidation resistance
HRP20030002A2 (en)	2005-10-31	STABLE GABAPENTIN HAVING pH WITHIN A CONTROLLED RANGE
SG63757A1 (en)	1999-03-30	Adding impurities to improve the efficiency of allngan quantum well led's
AR016099A1 (es)	2001-06-20	Composiciones detergentes liquidas no acuosas que contienen particulas enzimaticas que tienen densidad reducida
NO952138D0 (no)	1995-05-30	Cefiximpreparat
AU591525B2 (en)	1989-12-07	Stabilization of interferons
TR200003413A2 (tr)	2001-06-21	Granüler organosilan hazır ürün, bunun üretimi için bir işlem ve kullanımı
ES2153637T3 (es)	2001-03-01	Percarbonato de sodio y su procedimiento de obtencion.
ATE297457T1 (de)	2005-06-15	Alkylbenzolsulfonat-granulate
AU3856595A (en)	1996-06-06	Hydrate for drug use