ATE319702T1 - Verfahren zur herstellung von benzothiophen- derivaten - Google Patents

Verfahren zur herstellung von benzothiophen- derivaten

Info

Publication number: ATE319702T1
Authority: AT; Austria
Prior art keywords: formula; benzothiophene derivatives; chem; compound; producing
Prior art date: 1999-08-02

Application number

AT00115890T

Other languages

English (en)

Inventor

Bernd Junghans

Michelangelo Scalone

Thomas Albert Zeibig

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-08-02

Filing date

2000-07-25

Publication date

2006-03-15

2000-07-25 Application filed filed Critical

2006-03-15 Application granted granted Critical

2006-03-15 Publication of ATE319702T1 publication Critical patent/ATE319702T1/de

Links

FCEHBMOGCRZNNI-UHFFFAOYSA-N 1-benzothiophene Chemical class C1=CC=C2SC=CC2=C1 FCEHBMOGCRZNNI-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
ZEXIVBYDDCIOKA-UHFFFAOYSA-N 1-benzothiophen-2-ol Chemical compound C1=CC=C2SC(O)=CC2=C1 ZEXIVBYDDCIOKA-UHFFFAOYSA-N 0.000 abstract 1
239000013543 active substance Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
238000007282 cyclocarbonylation reaction Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
238000007127 saponification reaction Methods 0.000 abstract 1
159000000000 sodium salts Chemical class 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Catalysts (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT00115890T 1999-08-02 2000-07-25 Verfahren zur herstellung von benzothiophen- derivaten ATE319702T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP99115222		1999-08-02

Publications (1)

Publication Number	Publication Date
ATE319702T1 true ATE319702T1 (de)	2006-03-15

Family

ID=8238708

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00115890T ATE319702T1 (de)	1999-08-02	2000-07-25	Verfahren zur herstellung von benzothiophen- derivaten

Country Status (13)

Country	Link
US (3)	US6291685B1 (de)
EP (1)	EP1078923B1 (de)
JP (2)	JP3278649B2 (de)
KR (1)	KR100440102B1 (de)
CN (1)	CN1123570C (de)
AT (1)	ATE319702T1 (de)
CA (1)	CA2314699A1 (de)
CY (1)	CY1106096T1 (de)
DE (1)	DE60026404T2 (de)
DK (1)	DK1078923T3 (de)
ES (1)	ES2258431T3 (de)
JO (1)	JO2239B1 (de)
PT (1)	PT1078923E (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6531609B2 (en) *	2000-04-14	2003-03-11	Hoffmann-La Roche Inc.	Process for the preparation of thiazolidinedione derivatives
AU2002230409A1 (en) *	2000-11-27	2002-06-03	Eli Lilly And Company	Process for preparing 3-aryl-benzo(b)thiophenes
EP1355880A2 (de) *	2001-01-25	2003-10-29	F. Hoffmann-La Roche Ag	Verfahren zur herstellung von heterocyclischen inden-analogen
SK11322003A3 (en)	2001-02-12	2004-10-05	Hoffmann La Roche	6-Substituted pyrido-pyrimidines
EP1792614A1 (de) *	2001-02-22	2007-06-06	Teijin Pharma Limited	Benzo[b]thiophenderivate
SE0100903D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
SE0100902D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
RU2278859C2 (ru)	2001-05-15	2006-06-27	Ф.Хоффманн-Ля Рош Аг	Замещенные карбоновыми кислотами оксазоловые производные в качестве ppar-альфа и гамма-активаторов при лечении диабета
PL374818A1 (en)	2002-07-03	2005-10-31	F.Hoffmann-La Roche Ag	Oxazole derivatives and their use as insulin sensitizers
SE0202539D0 (sv) *	2002-08-27	2002-08-27	Astrazeneca Ab	Compounds
ATE483699T1 (de)	2002-08-30	2010-10-15	Hoffmann La Roche	Neue 2-arylthiazolverbindungen als ppar-alpha und gamma agonisten
WO2004024726A1 (en)	2002-09-12	2004-03-25	F. Hoffmann-La Roche Ag	N-substituted-1h-indol-5-propionic acid compounds as ppar agonists useful for the treatment of diabetes
DE60323130D1 (de)	2002-11-25	2008-10-02	Hoffmann La Roche	Indolderivaten
GB0311092D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
GB0311091D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
SE0401762D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Novel compounds
US7648992B2 (en)	2004-07-05	2010-01-19	Astrazeneca Ab	Hydantoin derivatives for the treatment of obstructive airway diseases
SE0401763D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Compounds
SE0403086D0 (sv)	2004-12-17	2004-12-17	Astrazeneca Ab	Compounds
SE0403085D0 (sv) *	2004-12-17	2004-12-17	Astrazeneca Ab	Novel componds
DE102005017216A1 (de) *	2005-04-14	2006-10-19	Deutsches Zentrum für Luft- und Raumfahrttechnik e.V.	Thermische Wasserstoffherstellung in einer Gas-Festphasenreaktion
TW200831488A (en) *	2006-11-29	2008-08-01	Astrazeneca Ab	Novel compounds
EP3479334A4 (de)	2016-06-30	2020-03-04	Cutaneous Information Technologies, LLC	System und verfahren für pflegeübergänge
CN115805103B (zh) *	2021-09-14	2024-04-09	万华化学集团股份有限公司	一种失活钛硅分子筛的再生方法
CN116459873B (zh) *	2022-01-12	2025-02-18	万华化学集团股份有限公司	一种烯属不饱和化合物羰基化催化剂及其制备方法、应用
CN117019118B (zh) *	2023-10-08	2024-01-05	西安金沃泰环保科技有限公司	一种用于苯系废气的过滤材料及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5330998A (en) *	1988-03-08	1994-07-19	Pfizer Inc.	Thiazolidinedione derivatives as hypoglycemic agents
CA2245055C (en)	1989-02-28	2003-03-25	F. Hoffmann-La Roche Ag	Amidation of pyridines
DE4317320A1 (de) *	1993-05-25	1994-12-01	Boehringer Mannheim Gmbh	Neue Thiazolidindione und diese enthaltende Arzneimittel
US6133279A (en) *	1996-06-26	2000-10-17	Chugai Seiyaku Kabushiki Kaisha	Therapeutic agents for renal diseases and organ preservatives
CA2259487A1 (en) *	1996-07-01	1998-01-08	Margaret Mary Faul	Hypoglycemic and hypolipidemic compounds
DE19711616A1 (de)	1997-03-20	1998-09-24	Boehringer Mannheim Gmbh	Verbessertes Verfahren zur Herstellung von Thiazolidindionen

2000
- 2000-07-25 EP EP00115890A patent/EP1078923B1/de not_active Expired - Lifetime
- 2000-07-25 DE DE60026404T patent/DE60026404T2/de not_active Expired - Fee Related
- 2000-07-25 AT AT00115890T patent/ATE319702T1/de not_active IP Right Cessation
- 2000-07-25 DK DK00115890T patent/DK1078923T3/da active
- 2000-07-25 PT PT00115890T patent/PT1078923E/pt unknown
- 2000-07-25 ES ES00115890T patent/ES2258431T3/es not_active Expired - Lifetime
- 2000-07-26 US US09/625,887 patent/US6291685B1/en not_active Expired - Fee Related
- 2000-07-27 JO JO2000128A patent/JO2239B1/en active
- 2000-07-28 CN CN00121170A patent/CN1123570C/zh not_active Expired - Fee Related
- 2000-07-28 CA CA002314699A patent/CA2314699A1/en not_active Abandoned
- 2000-07-31 KR KR10-2000-0044225A patent/KR100440102B1/ko not_active Expired - Fee Related
- 2000-08-01 JP JP2000232565A patent/JP3278649B2/ja not_active Expired - Fee Related
2001
- 2001-05-08 US US09/851,352 patent/US6437144B2/en not_active Expired - Fee Related
- 2001-11-08 US US10/008,877 patent/US6482958B2/en not_active Expired - Fee Related
- 2001-11-09 JP JP2001344469A patent/JP2002155079A/ja active Pending
2006
- 2006-06-07 CY CY20061100759T patent/CY1106096T1/el unknown

Also Published As

Publication number	Publication date
US6437144B2 (en)	2002-08-20
CY1106096T1 (el)	2011-06-08
EP1078923B1 (de)	2006-03-08
JP2001048876A (ja)	2001-02-20
CN1123570C (zh)	2003-10-08
CN1282741A (zh)	2001-02-07
JP2002155079A (ja)	2002-05-28
US6291685B1 (en)	2001-09-18
ES2258431T3 (es)	2006-09-01
EP1078923A3 (de)	2001-07-11
KR100440102B1 (ko)	2004-07-15
KR20010049948A (ko)	2001-06-15
DE60026404D1 (de)	2006-05-04
US6482958B2 (en)	2002-11-19
JO2239B1 (en)	2004-10-07
JP3278649B2 (ja)	2002-04-30
EP1078923A2 (de)	2001-02-28
US20020010345A1 (en)	2002-01-24
US20020077488A1 (en)	2002-06-20
DK1078923T3 (da)	2006-07-10
DE60026404T2 (de)	2006-10-19
CA2314699A1 (en)	2001-02-02
PT1078923E (pt)	2006-07-31

Legal Events

Date

Code

Title

Description

2006-12-15

UEP

Publication of translation of european patent specification

Ref document number: 1078923

Country of ref document: EP

2009-04-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
DE60026404D1 (de)	2006-05-04	Verfahren zur Herstellung von Benzothiophen-Derivaten
EE200200572A (et)	2004-04-15	Pertsükvinniin, selle valmistamismeetod, kandseene liik ja farmatseutiline kompositsioon
DK1159279T3 (da)	2003-02-17	4-Oxo-4,7-dihydro-thieno[2,3-b]pyridin-5-carboxamider som antivirale midler
PT87163A (pt)	1988-05-01	Process for preparing 1-phenyl-3-naphthalenyloxipropanamines
PT992509E (pt)	2004-12-31	Novos derivados macrolidos
KR940002249A (ko)	1994-02-17	치환된 아미노티에노피리딘, 이의 제조방법 및 약제로서의 이의 용도
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NO982927L (no)	1998-06-23	Biologisk aktive benzotiazolon etanaminer
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ATE298336T1 (de)	2005-07-15	Verfahren zur herstellung von thiazolidinedion- derivaten und zwischenprodukte
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CA2378002A1 (en)	2001-01-18	Method for preparing 2-(2-arylmorpholin-2-yl)ethanol derivatives and intermediates
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