ATE319702T1 - Verfahren zur herstellung von benzothiophen- derivaten - Google Patents

Verfahren zur herstellung von benzothiophen- derivaten

Info

Publication number: ATE319702T1
Authority: AT; Austria
Prior art keywords: formula; benzothiophene derivatives; chem; compound; producing
Prior art date: 1999-08-02

Application number

AT00115890T

Other languages

English (en)

Inventor

Bernd Junghans

Michelangelo Scalone

Thomas Albert Zeibig

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-08-02

Filing date

2000-07-25

Publication date

2006-03-15

2000-07-25 Application filed filed Critical

2006-03-15 Application granted granted Critical

2006-03-15 Publication of ATE319702T1 publication Critical patent/ATE319702T1/de

Links

FCEHBMOGCRZNNI-UHFFFAOYSA-N 1-benzothiophene Chemical class C1=CC=C2SC=CC2=C1 FCEHBMOGCRZNNI-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
ZEXIVBYDDCIOKA-UHFFFAOYSA-N 1-benzothiophen-2-ol Chemical compound C1=CC=C2SC(O)=CC2=C1 ZEXIVBYDDCIOKA-UHFFFAOYSA-N 0.000 abstract 1
239000013543 active substance Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
238000007282 cyclocarbonylation reaction Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
238000007127 saponification reaction Methods 0.000 abstract 1
159000000000 sodium salts Chemical class 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Catalysts (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT00115890T 1999-08-02 2000-07-25 Verfahren zur herstellung von benzothiophen- derivaten ATE319702T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP99115222		1999-08-02

Publications (1)

Publication Number	Publication Date
ATE319702T1 true ATE319702T1 (de)	2006-03-15

Family

ID=8238708

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00115890T ATE319702T1 (de)	1999-08-02	2000-07-25	Verfahren zur herstellung von benzothiophen- derivaten

Country Status (13)

Country	Link
US (3)	US6291685B1 (de)
EP (1)	EP1078923B1 (de)
JP (2)	JP3278649B2 (de)
KR (1)	KR100440102B1 (de)
CN (1)	CN1123570C (de)
AT (1)	ATE319702T1 (de)
CA (1)	CA2314699A1 (de)
CY (1)	CY1106096T1 (de)
DE (1)	DE60026404T2 (de)
DK (1)	DK1078923T3 (de)
ES (1)	ES2258431T3 (de)
JO (1)	JO2239B1 (de)
PT (1)	PT1078923E (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6531609B2 (en)	2000-04-14	2003-03-11	Hoffmann-La Roche Inc.	Process for the preparation of thiazolidinedione derivatives
AU2002230409A1 (en) *	2000-11-27	2002-06-03	Eli Lilly And Company	Process for preparing 3-aryl-benzo(b)thiophenes
MXPA03006606A (es) *	2001-01-25	2003-09-22	Hoffmann La Roche	Proceso para preparacion de analogos de indeno heterociclico.
CZ20032416A3 (cs)	2001-02-12	2004-07-14	F. Hoffmann-La Roche Ag	6-Substituované pyridopyrimidiny
AU2002233698B2 (en) *	2001-02-22	2007-11-08	Teijin Limited	Benzo(b)thiophene derivative and process for producing the same
SE0100902D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
SE0100903D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
DE60211891T2 (de)	2001-05-15	2007-05-24	F. Hoffmann-La Roche Ag	Carbonsäure-substituierte oxazol-derivate zur verwendung als ppar-alpha und -gamma aktivatoren zur behandlung von diabetes
JP4290648B2 (ja)	2002-07-03	2009-07-08	エフ．ホフマン−ラロシュアーゲー	オキサゾール誘導体及びインスリン感作物質としてのそれらの使用
SE0202539D0 (sv) *	2002-08-27	2002-08-27	Astrazeneca Ab	Compounds
PL375779A1 (en)	2002-08-30	2005-12-12	F.Hoffmann-La Roche Ag	Novel 2-arylthiazole compounds as pparalpha and ppargamma agonists
EP1539746B1 (de)	2002-09-12	2006-11-15	F. Hoffmann-La Roche Ag	N-substituierte-1h-indol-5-propansäure verbindungen als ppar-agonisten zur behandlung von diabetis
MXPA05005445A (es)	2002-11-25	2005-08-26	Hoffmann La Roche	Derivados de indolilo.
GB0311091D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
GB0311092D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
SE0401762D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Novel compounds
SE0401763D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Compounds
US7648992B2 (en)	2004-07-05	2010-01-19	Astrazeneca Ab	Hydantoin derivatives for the treatment of obstructive airway diseases
SE0403085D0 (sv) *	2004-12-17	2004-12-17	Astrazeneca Ab	Novel componds
SE0403086D0 (sv)	2004-12-17	2004-12-17	Astrazeneca Ab	Compounds
DE102005017216A1 (de) *	2005-04-14	2006-10-19	Deutsches Zentrum für Luft- und Raumfahrttechnik e.V.	Thermische Wasserstoffherstellung in einer Gas-Festphasenreaktion
TW200831488A (en) *	2006-11-29	2008-08-01	Astrazeneca Ab	Novel compounds
EP3479334A4 (de)	2016-06-30	2020-03-04	Cutaneous Information Technologies, LLC	System und verfahren für pflegeübergänge
CN115805103B (zh) *	2021-09-14	2024-04-09	万华化学集团股份有限公司	一种失活钛硅分子筛的再生方法
CN116459873B (zh) *	2022-01-12	2025-02-18	万华化学集团股份有限公司	一种烯属不饱和化合物羰基化催化剂及其制备方法、应用
CN117019118B (zh) *	2023-10-08	2024-01-05	西安金沃泰环保科技有限公司	一种用于苯系废气的过滤材料及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5330998A (en) *	1988-03-08	1994-07-19	Pfizer Inc.	Thiazolidinedione derivatives as hypoglycemic agents
CA2245055C (en)	1989-02-28	2003-03-25	F. Hoffmann-La Roche Ag	Amidation of pyridines
DE4317320A1 (de) *	1993-05-25	1994-12-01	Boehringer Mannheim Gmbh	Neue Thiazolidindione und diese enthaltende Arzneimittel
US6133279A (en) *	1996-06-26	2000-10-17	Chugai Seiyaku Kabushiki Kaisha	Therapeutic agents for renal diseases and organ preservatives
EP0925063A4 (de) *	1996-07-01	2000-12-27	Lilly Co Eli	Blutzuckersenkende und lipidsenkende verbindungen
DE19711616A1 (de)	1997-03-20	1998-09-24	Boehringer Mannheim Gmbh	Verbessertes Verfahren zur Herstellung von Thiazolidindionen

2000
- 2000-07-25 PT PT00115890T patent/PT1078923E/pt unknown
- 2000-07-25 EP EP00115890A patent/EP1078923B1/de not_active Expired - Lifetime
- 2000-07-25 DK DK00115890T patent/DK1078923T3/da active
- 2000-07-25 AT AT00115890T patent/ATE319702T1/de not_active IP Right Cessation
- 2000-07-25 DE DE60026404T patent/DE60026404T2/de not_active Expired - Fee Related
- 2000-07-25 ES ES00115890T patent/ES2258431T3/es not_active Expired - Lifetime
- 2000-07-26 US US09/625,887 patent/US6291685B1/en not_active Expired - Fee Related
- 2000-07-27 JO JO2000128A patent/JO2239B1/en active
- 2000-07-28 CA CA002314699A patent/CA2314699A1/en not_active Abandoned
- 2000-07-28 CN CN00121170A patent/CN1123570C/zh not_active Expired - Fee Related
- 2000-07-31 KR KR10-2000-0044225A patent/KR100440102B1/ko not_active Expired - Fee Related
- 2000-08-01 JP JP2000232565A patent/JP3278649B2/ja not_active Expired - Fee Related
2001
- 2001-05-08 US US09/851,352 patent/US6437144B2/en not_active Expired - Fee Related
- 2001-11-08 US US10/008,877 patent/US6482958B2/en not_active Expired - Fee Related
- 2001-11-09 JP JP2001344469A patent/JP2002155079A/ja active Pending
2006
- 2006-06-07 CY CY20061100759T patent/CY1106096T1/el unknown

Also Published As

Publication number	Publication date
US6437144B2 (en)	2002-08-20
CA2314699A1 (en)	2001-02-02
EP1078923A3 (de)	2001-07-11
PT1078923E (pt)	2006-07-31
DK1078923T3 (da)	2006-07-10
US6291685B1 (en)	2001-09-18
CY1106096T1 (el)	2011-06-08
JP2001048876A (ja)	2001-02-20
DE60026404D1 (de)	2006-05-04
KR100440102B1 (ko)	2004-07-15
EP1078923A2 (de)	2001-02-28
EP1078923B1 (de)	2006-03-08
KR20010049948A (ko)	2001-06-15
CN1123570C (zh)	2003-10-08
JO2239B1 (en)	2004-10-07
CN1282741A (zh)	2001-02-07
ES2258431T3 (es)	2006-09-01
US20020010345A1 (en)	2002-01-24
JP3278649B2 (ja)	2002-04-30
DE60026404T2 (de)	2006-10-19
US6482958B2 (en)	2002-11-19
US20020077488A1 (en)	2002-06-20
JP2002155079A (ja)	2002-05-28

Legal Events

Date

Code

Title

Description

2006-12-15

UEP

Publication of translation of european patent specification

Ref document number: 1078923

Country of ref document: EP

2009-04-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
ATE319702T1 (de)	2006-03-15	Verfahren zur herstellung von benzothiophen- derivaten
EE200200572A (et)	2004-04-15	Pertsükvinniin, selle valmistamismeetod, kandseene liik ja farmatseutiline kompositsioon
DK1159279T3 (da)	2003-02-17	4-Oxo-4,7-dihydro-thieno[2,3-b]pyridin-5-carboxamider som antivirale midler
BG108426A (bg)	2005-01-31	Нови производни на сулфоновата киселина
PT992509E (pt)	2004-12-31	Novos derivados macrolidos
KR940002249A (ko)	1994-02-17	치환된 아미노티에노피리딘, 이의 제조방법 및 약제로서의 이의 용도
ATE298747T1 (de)	2005-07-15	Verfahren zur herstellung von 5- hydroxybenzo(b)thiophen-3-carbonsäure
PT1204658E (pt)	2003-08-29	Agonistas benzofurilpiperazina de serotonina
DE60237388D1 (de)	2010-09-30	Verfahren zur herstellung von zusammensetzungen mit erhöhtem gehalt von salzen pharmazeutisch aktiver rotamere
DE60010682D1 (de)	2004-06-17	Verfahren zur herstellung von zwischenprodukten für pestizide
ATE295368T1 (de)	2005-05-15	Verfahren zur herstellung 3-amino-gallensaurer derivate
ATE318825T1 (de)	2006-03-15	Herstellung von cephalosporin
EP1227081A4 (de)	2004-08-11	Verfahren zur herstellung von oxyiminoalkansäure-derivaten
EA200101170A1 (ru)	2002-04-25	Галоидпроизводные 9-деоксо-9а-аза-9а-гомоэритромицина а
NO20021727D0 (no)	2002-04-12	Fremgangsmåte for fremstilling av 3,4-metylen-dioksy- mandelisk syre
DE60111634D1 (de)	2005-07-28	Verfahren zur herstellung von thiazolidinedion-derivaten und zwischenprodukte
DK1392672T3 (da)	2005-08-29	Chlormethylering af thiopen
DE60233307D1 (de)	2009-09-24	Verfahren zur herstellung optisch aktiver propoxyanilinderivate
AU686104B2 (en)	1998-02-05	Substituted amidinonaphthyl ester derivatives
DE69928610D1 (de)	2006-01-05	Verfahren zur Herstellung von 2-Carbamoyl-Pyridinen
DE60335960D1 (de)	2011-03-17	1,2,4-triazolderivat, verfahren zu dessenherstellung, und dieses enthaltende pharmazeutische zusammensetzung
ATE247963T1 (de)	2003-09-15	Medikament zur behandlung von glaukoma und ischämischer retinopathie
CA2378002A1 (en)	2001-01-18	Method for preparing 2-(2-arylmorpholin-2-yl)ethanol derivatives and intermediates
BR9902049A (pt)	2000-05-02	Derivados 9a,11b-desidro de 9-oxima-3-ceto-6-o-metileritromicina.
DE50107619D1 (de)	2006-02-16	Verfahren zur herstellung von 4-brom-anilin-derivaten