ATE319702T1 - Verfahren zur herstellung von benzothiophen- derivaten - Google Patents

Verfahren zur herstellung von benzothiophen- derivaten

Info

Publication number: ATE319702T1
Authority: AT; Austria
Prior art keywords: formula; benzothiophene derivatives; chem; compound; producing
Prior art date: 1999-08-02

Application number

AT00115890T

Other languages

English (en)

Inventor

Bernd Junghans

Michelangelo Scalone

Thomas Albert Zeibig

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-08-02

Filing date

2000-07-25

Publication date

2006-03-15

2000-07-25 Application filed filed Critical

2006-03-15 Application granted granted Critical

2006-03-15 Publication of ATE319702T1 publication Critical patent/ATE319702T1/de

Links

FCEHBMOGCRZNNI-UHFFFAOYSA-N 1-benzothiophene Chemical class C1=CC=C2SC=CC2=C1 FCEHBMOGCRZNNI-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
ZEXIVBYDDCIOKA-UHFFFAOYSA-N 1-benzothiophen-2-ol Chemical compound C1=CC=C2SC(O)=CC2=C1 ZEXIVBYDDCIOKA-UHFFFAOYSA-N 0.000 abstract 1
239000013543 active substance Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
238000007282 cyclocarbonylation reaction Methods 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
238000007127 saponification reaction Methods 0.000 abstract 1
159000000000 sodium salts Chemical class 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Catalysts (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT00115890T 1999-08-02 2000-07-25 Verfahren zur herstellung von benzothiophen- derivaten ATE319702T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP99115222		1999-08-02

Publications (1)

Publication Number	Publication Date
ATE319702T1 true ATE319702T1 (de)	2006-03-15

Family

ID=8238708

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00115890T ATE319702T1 (de)	1999-08-02	2000-07-25	Verfahren zur herstellung von benzothiophen- derivaten

Country Status (13)

Country	Link
US (3)	US6291685B1 (de)
EP (1)	EP1078923B1 (de)
JP (2)	JP3278649B2 (de)
KR (1)	KR100440102B1 (de)
CN (1)	CN1123570C (de)
AT (1)	ATE319702T1 (de)
CA (1)	CA2314699A1 (de)
CY (1)	CY1106096T1 (de)
DE (1)	DE60026404T2 (de)
DK (1)	DK1078923T3 (de)
ES (1)	ES2258431T3 (de)
JO (1)	JO2239B1 (de)
PT (1)	PT1078923E (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6531609B2 (en) *	2000-04-14	2003-03-11	Hoffmann-La Roche Inc.	Process for the preparation of thiazolidinedione derivatives
WO2002042289A2 (en) *	2000-11-27	2002-05-30	Eli Lilly And Company	Process for preparing 3-aryl-benzo[b]thiophenes
KR100559019B1 (ko)	2001-01-25	2006-03-10	에프. 호프만-라 로슈 아게	헤테로사이클릭 인덴 유사체의 제조 방법
HU229604B1 (en)	2001-02-12	2014-02-28	Hoffmann La Roche	6-substituted pyrido-pyrimidines, process for their preparation and pharmaceutical compositions containing them
NZ522150A (en) *	2001-02-22	2006-03-31	Teijin Ltd	Benzo[b]thiophene derivatives and processes for preparing the same
SE0100903D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
SE0100902D0 (sv) *	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
ME01310B (me)	2001-05-15	2011-10-10	Hoffmann La Roche	Derivati oksazola koji su supstituisani karboksilnom kiselinom za primenu kao ppar-alfa-1-gama aktivatori u lečenju dijabetesa
ATE372990T1 (de)	2002-07-03	2007-09-15	Hoffmann La Roche	Oxazolderivat und deren verwendung als insulinsensibilisatoren
SE0202539D0 (sv) *	2002-08-27	2002-08-27	Astrazeneca Ab	Compounds
CN100475810C (zh)	2002-08-30	2009-04-08	霍夫曼-拉罗奇有限公司	作为PPARα和PPARγ激动剂的新型2-芳基噻唑化合物
NZ537979A (en)	2002-09-12	2007-08-31	Hoffmann La Roche	N-substituted-1H-indol-5-propionic acid compounds as PPAR agonists useful for the treatment of diabetes
MXPA05005445A (es)	2002-11-25	2005-08-26	Hoffmann La Roche	Derivados de indolilo.
GB0311091D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
GB0311092D0 (en) *	2003-05-14	2003-06-18	Bp Chem Int Ltd	Process
SE0401763D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Compounds
SE0401762D0 (sv) *	2004-07-05	2004-07-05	Astrazeneca Ab	Novel compounds
US7648992B2 (en)	2004-07-05	2010-01-19	Astrazeneca Ab	Hydantoin derivatives for the treatment of obstructive airway diseases
SE0403085D0 (sv) *	2004-12-17	2004-12-17	Astrazeneca Ab	Novel componds
SE0403086D0 (sv)	2004-12-17	2004-12-17	Astrazeneca Ab	Compounds
DE102005017216A1 (de) *	2005-04-14	2006-10-19	Deutsches Zentrum für Luft- und Raumfahrttechnik e.V.	Thermische Wasserstoffherstellung in einer Gas-Festphasenreaktion
TW200831488A (en) *	2006-11-29	2008-08-01	Astrazeneca Ab	Novel compounds
WO2018005828A1 (en)	2016-06-30	2018-01-04	Cutaneous Information Technologies, Llc	System and method for transitions of care
CN115805103B (zh) *	2021-09-14	2024-04-09	万华化学集团股份有限公司	一种失活钛硅分子筛的再生方法
CN116459873B (zh) *	2022-01-12	2025-02-18	万华化学集团股份有限公司	一种烯属不饱和化合物羰基化催化剂及其制备方法、应用
CN117019118B (zh) *	2023-10-08	2024-01-05	西安金沃泰环保科技有限公司	一种用于苯系废气的过滤材料及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5330998A (en) *	1988-03-08	1994-07-19	Pfizer Inc.	Thiazolidinedione derivatives as hypoglycemic agents
CA2008878C (en)	1989-02-28	2003-01-21	Michelangelo Scalone	Process for preparing pyridine-2-carboxamides
DE4317320A1 (de) *	1993-05-25	1994-12-01	Boehringer Mannheim Gmbh	Neue Thiazolidindione und diese enthaltende Arzneimittel
WO1997049388A1 (en) *	1996-06-26	1997-12-31	Chugai Seiyaku Kabushiki Kaisha	Remedies for renal diseases and organ-preserving agents
IL121202A (en) *	1996-07-01	2001-08-26	Lilly Co Eli	Hypoglycemic and hypolipidemic compounds, process for their preparation, pharmaceutial compositions comprising same, and uses thereof
DE19711616A1 (de)	1997-03-20	1998-09-24	Boehringer Mannheim Gmbh	Verbessertes Verfahren zur Herstellung von Thiazolidindionen

2000
- 2000-07-25 DK DK00115890T patent/DK1078923T3/da active
- 2000-07-25 ES ES00115890T patent/ES2258431T3/es not_active Expired - Lifetime
- 2000-07-25 PT PT00115890T patent/PT1078923E/pt unknown
- 2000-07-25 EP EP00115890A patent/EP1078923B1/de not_active Expired - Lifetime
- 2000-07-25 DE DE60026404T patent/DE60026404T2/de not_active Expired - Fee Related
- 2000-07-25 AT AT00115890T patent/ATE319702T1/de not_active IP Right Cessation
- 2000-07-26 US US09/625,887 patent/US6291685B1/en not_active Expired - Fee Related
- 2000-07-27 JO JO2000128A patent/JO2239B1/en active
- 2000-07-28 CA CA002314699A patent/CA2314699A1/en not_active Abandoned
- 2000-07-28 CN CN00121170A patent/CN1123570C/zh not_active Expired - Fee Related
- 2000-07-31 KR KR10-2000-0044225A patent/KR100440102B1/ko not_active Expired - Fee Related
- 2000-08-01 JP JP2000232565A patent/JP3278649B2/ja not_active Expired - Fee Related
2001
- 2001-05-08 US US09/851,352 patent/US6437144B2/en not_active Expired - Fee Related
- 2001-11-08 US US10/008,877 patent/US6482958B2/en not_active Expired - Fee Related
- 2001-11-09 JP JP2001344469A patent/JP2002155079A/ja active Pending
2006
- 2006-06-07 CY CY20061100759T patent/CY1106096T1/el unknown

Also Published As

Publication number	Publication date
US6291685B1 (en)	2001-09-18
JP3278649B2 (ja)	2002-04-30
DE60026404T2 (de)	2006-10-19
CA2314699A1 (en)	2001-02-02
CN1123570C (zh)	2003-10-08
US20020010345A1 (en)	2002-01-24
US20020077488A1 (en)	2002-06-20
EP1078923A3 (de)	2001-07-11
DE60026404D1 (de)	2006-05-04
CN1282741A (zh)	2001-02-07
KR20010049948A (ko)	2001-06-15
KR100440102B1 (ko)	2004-07-15
JP2002155079A (ja)	2002-05-28
CY1106096T1 (el)	2011-06-08
JO2239B1 (en)	2004-10-07
EP1078923B1 (de)	2006-03-08
ES2258431T3 (es)	2006-09-01
DK1078923T3 (da)	2006-07-10
PT1078923E (pt)	2006-07-31
EP1078923A2 (de)	2001-02-28
JP2001048876A (ja)	2001-02-20
US6437144B2 (en)	2002-08-20
US6482958B2 (en)	2002-11-19

Legal Events

Date

Code

Title

Description

2006-12-15

UEP

Publication of translation of european patent specification

Ref document number: 1078923

Country of ref document: EP

2009-04-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
DE60026404D1 (de)	2006-05-04	Verfahren zur Herstellung von Benzothiophen-Derivaten
EE200200572A (et)	2004-04-15	Pertsükvinniin, selle valmistamismeetod, kandseene liik ja farmatseutiline kompositsioon
DK1159279T3 (da)	2003-02-17	4-Oxo-4,7-dihydro-thieno[2,3-b]pyridin-5-carboxamider som antivirale midler
PT87163A (pt)	1988-05-01	Process for preparing 1-phenyl-3-naphthalenyloxipropanamines
PT992509E (pt)	2004-12-31	Novos derivados macrolidos
KR940002249A (ko)	1994-02-17	치환된 아미노티에노피리딘, 이의 제조방법 및 약제로서의 이의 용도
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