ATE319706T1 - Pyridinon und pyridinethion-derivate mit hiv- hemmenden eigenschaften - Google Patents

Pyridinon und pyridinethion-derivate mit hiv- hemmenden eigenschaften

Info

Publication number: ATE319706T1
Authority: AT; Austria
Prior art keywords: sub; sup; inhibiting properties; pyridinethone; pyridinone
Prior art date: 2000-09-19

Application number

AT01980812T

Other languages

English (en)

Inventor

Jerome Guillemont

Abdellah Benjahad

Dominique Mabire

Guyen Chi Hung N

David Grierson

Claude Monneret

Emile Bisagni

Gerard Sanz

Laurence Decrane

Original Assignee

Centre Nat Rech Scient

Inst Curie

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-09-19

Filing date

2001-09-18

Publication date

2006-03-15

2001-09-18 Application filed by Centre Nat Rech Scient, Inst Curie filed Critical Centre Nat Rech Scient

2006-03-15 Application granted granted Critical

2006-03-15 Publication of ATE319706T1 publication Critical patent/ATE319706T1/de

Links

UBQKCCHYAOITMY-UHFFFAOYSA-N pyridin-2-ol Chemical compound OC1=CC=CC=N1 UBQKCCHYAOITMY-UHFFFAOYSA-N 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 4
125000002485 formyl group Chemical group [H]C(*)=O 0.000 abstract 2
125000001475 halogen functional group Chemical group 0.000 abstract 2
150000001204 N-oxides Chemical class 0.000 abstract 1
125000003342 alkenyl group Chemical group 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
125000004414 alkyl thio group Chemical group 0.000 abstract 1
150000001412 amines Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
230000002401 inhibitory effect Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000001424 substituent group Chemical group 0.000 abstract 1

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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D213/63—One oxygen atom
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems

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Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Virology (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Tropical Medicine & Parasitology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
AIDS & HIV (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Molecular Biology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Quinoline Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AT01980812T 2000-09-19 2001-09-18 Pyridinon und pyridinethion-derivate mit hiv- hemmenden eigenschaften ATE319706T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP00402583		2000-09-19

Publications (1)

Publication Number	Publication Date
ATE319706T1 true ATE319706T1 (de)	2006-03-15

Family

ID=8173871

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01980812T ATE319706T1 (de)	2000-09-19	2001-09-18	Pyridinon und pyridinethion-derivate mit hiv- hemmenden eigenschaften

Country Status (7)

Country	Link
US (1)	US7115608B2 (de)
EP (1)	EP1318995B1 (de)
JP (1)	JP2004509867A (de)
AT (1)	ATE319706T1 (de)
AU (1)	AU2002212598A1 (de)
DE (1)	DE60117839T2 (de)
WO (1)	WO2002024650A2 (de)

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EP3331876B1 (de)	2015-08-05	2020-10-07	Vitae Pharmaceuticals, LLC	Modulatoren von ror-gamma
EP3868750A1 (de)	2015-11-20	2021-08-25	Vitae Pharmaceuticals, LLC	Modulatoren von ror-gamma
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2001
- 2001-09-18 AT AT01980812T patent/ATE319706T1/de not_active IP Right Cessation
- 2001-09-18 WO PCT/IB2001/002082 patent/WO2002024650A2/en not_active Ceased
- 2001-09-18 AU AU2002212598A patent/AU2002212598A1/en not_active Abandoned
- 2001-09-18 US US10/380,784 patent/US7115608B2/en not_active Expired - Fee Related
- 2001-09-18 JP JP2002529063A patent/JP2004509867A/ja active Pending
- 2001-09-18 DE DE60117839T patent/DE60117839T2/de not_active Expired - Lifetime
- 2001-09-18 EP EP01980812A patent/EP1318995B1/de not_active Expired - Lifetime

Also Published As

Publication number	Publication date
JP2004509867A (ja)	2004-04-02
WO2002024650A2 (en)	2002-03-28
WO2002024650B1 (en)	2002-11-14
EP1318995B1 (de)	2006-03-08
AU2002212598A1 (en)	2002-04-02
WO2002024650A3 (en)	2002-08-08
EP1318995A2 (de)	2003-06-18
DE60117839D1 (de)	2006-05-04
US7115608B2 (en)	2006-10-03
US20040229847A1 (en)	2004-11-18
DE60117839T2 (de)	2006-11-23

Legal Events

Date	Code	Title	Description
2006-09-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
DE60117839D1 (de)	2006-05-04	Pyridinon und pyridinethion-derivate mit hiv-hemmenden eigenschaften
NO20023823D0 (no)	2002-08-13	Fremgangsmåte for tilvirkning og bruk av pyrrolopyrimidinon- derivater
DK0870768T3 (da)	2002-07-01	Azaindol-ethylaminderivater som nikotinacetylcholinreceptor-bindingsmidler
MX9700883A (es)	1997-08-30	Derivados sustituidos de la quinazolina.
IS6565A (is)	2002-09-24	Trópan afleiður nytsamlegar í meðferð
DK1382604T3 (da)	2006-04-18	Quinolinderivater med en azolylgruppe og quinazolinderivater
HUP0204429A2 (hu)	2003-04-28	Aril-amin-származékok és alkalmazásuk antitelomeráz hatású szerként
DK1442019T3 (da)	2008-01-14	Amidderivater som glycogensynthasekinase 3- beta-inhibitorer
NZ333382A (en)	2000-05-26	N-[4-(heteroarylmethyl)phenyl]-heteroarylamines
DK0862562T3 (da)	2001-09-24	Benzoxazepinforbindelser, fremstilling deraf og anvendelse deraf som lipidniveauformindskende midler
TR200000918T2 (tr)	2000-07-21	Halojen ikameli tetrasiklik tetrahidrofuran türevleri.
CS142891A3 (en)	1992-02-19	Application of substituted 1,2,4-triazinediones
ATE346067T1 (de)	2006-12-15	Carbolinderivate
TR200001950T2 (tr)	2000-11-21	İkameli 2-benzilamino-2-fenil-asetamid bileşikler.
DE69814563D1 (de)	2003-06-18	Pyrrolo-(3,2-b)pyridine und ihre Verwendung als 5-HT1F Agonisten
ES8802302A1 (es)	1988-05-01	Procedimiento para la obtencion de 1-aril-4-nitropirazoles.
MXPA03000887A (es)	2004-04-05	Derivados heterociclicos fusionados como inhibidores de fosfodiesterasa.
ATE203537T1 (de)	2001-08-15	Pyrazol(1,5-a)pyrimidin derivate
BG103395A (en)	2000-02-29	Derivatives of benzenesulphonamide and medicaments containing them
DK0558104T3 (da)	1999-04-26	1,5-Benzodiazepinderivater og deres anvendelse i lægemidler
FR2838124B1 (fr)	2004-05-28	Derives de 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino [4,5-b]indole-1-acetamide, leur preparation et leur application en therapeutique
GR1001123B (el)	1993-04-28	Μεθοδος παρασκευης 1,4-διυδροπυριδινων.