ATE332295T1 - Verfahren zur herstellung von 5-substituierten oxazolverbindungen und 1,5-disubstituierten imidazolverbindungen - Google Patents
Verfahren zur herstellung von 5-substituierten oxazolverbindungen und 1,5-disubstituierten imidazolverbindungenInfo
- Publication number
- ATE332295T1 ATE332295T1 AT02705404T AT02705404T ATE332295T1 AT E332295 T1 ATE332295 T1 AT E332295T1 AT 02705404 T AT02705404 T AT 02705404T AT 02705404 T AT02705404 T AT 02705404T AT E332295 T1 ATE332295 T1 AT E332295T1
- Authority
- AT
- Austria
- Prior art keywords
- compounds
- producing
- substituted oxazole
- tosmic
- base
- Prior art date
Links
- -1 5-SUBSTITUTED OXAZOLE COMPOUNDS Chemical class 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 title 1
- CFOAUYCPAUGDFF-UHFFFAOYSA-N tosmic Chemical compound CC1=CC=C(S(=O)(=O)C[N+]#[C-])C=C1 CFOAUYCPAUGDFF-UHFFFAOYSA-N 0.000 abstract 2
- 239000000010 aprotic solvent Substances 0.000 abstract 1
- 238000000354 decomposition reaction Methods 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 125000002485 formyl group Chemical class [H]C(*)=O 0.000 abstract 1
- 150000002391 heterocyclic compounds Chemical class 0.000 abstract 1
- 150000007529 inorganic bases Chemical class 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000008204 material by function Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 150000007530 organic bases Chemical class 0.000 abstract 1
- 239000000575 pesticide Substances 0.000 abstract 1
- 239000003444 phase transfer catalyst Substances 0.000 abstract 1
- 239000003586 protic polar solvent Substances 0.000 abstract 1
- 239000011877 solvent mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/32—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001084092 | 2001-03-23 | ||
| JP2001084183 | 2001-03-23 | ||
| JP2001084184 | 2001-03-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE332295T1 true ATE332295T1 (de) | 2006-07-15 |
Family
ID=27346333
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02705404T ATE332295T1 (de) | 2001-03-23 | 2002-03-20 | Verfahren zur herstellung von 5-substituierten oxazolverbindungen und 1,5-disubstituierten imidazolverbindungen |
Country Status (9)
| Country | Link |
|---|---|
| US (3) | USRE40795E1 (de) |
| EP (1) | EP1371649B1 (de) |
| JP (1) | JP4161367B2 (de) |
| KR (1) | KR100586671B1 (de) |
| CN (1) | CN100506805C (de) |
| AT (1) | ATE332295T1 (de) |
| DE (1) | DE60212947T2 (de) |
| IL (2) | IL157724A0 (de) |
| WO (1) | WO2002076958A1 (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5112621B2 (ja) * | 2005-06-02 | 2013-01-09 | 日本曹達株式会社 | 5−置換オキサゾール化合物の精製方法及び製造方法 |
| KR101008187B1 (ko) * | 2008-06-16 | 2011-01-14 | 오토스테크 주식회사 | 기능성 가스켓을 갖는 용접 마스크 |
| CN104387301B (zh) * | 2014-11-11 | 2016-05-04 | 常州大学 | 一种2-氟-4-甲基苯磺酰甲基异腈的合成方法 |
| CN107095868B (zh) * | 2017-06-01 | 2019-06-11 | 深圳碳希生物科技有限公司 | 3-(5-噁唑基)苯酚在美白方面的应用及其制备方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH064600B2 (ja) * | 1984-03-26 | 1994-01-19 | ア−ス製薬株式会社 | 1−シトロネリ−ル−5−置換イミダゾ−ル類 |
| JPH0755931B2 (ja) * | 1986-03-24 | 1995-06-14 | アース製薬株式会社 | 1,5−ジ置換イミダゾ−ル |
| US4958030A (en) * | 1988-12-12 | 1990-09-18 | Ciba-Geigy Corporation | Process for the preparation of 3-phenylpyrrole derivatives |
| JP3065336B2 (ja) * | 1990-09-21 | 2000-07-17 | 日本合成化学工業株式会社 | 5―置換オキサゾールの製造法 |
| AU3087195A (en) | 1994-08-02 | 1996-03-04 | Nippon Soda Co., Ltd. | Oxazole derivative, process for producing the same, and herbicide |
| DE19633390A1 (de) * | 1996-08-19 | 1998-02-26 | Basf Ag | Verfahren zur Herstellung substituierter Imidazole |
-
2002
- 2002-03-20 US US11/825,114 patent/USRE40795E1/en not_active Expired - Lifetime
- 2002-03-20 US US10/471,434 patent/US7102010B2/en not_active Expired - Lifetime
- 2002-03-20 DE DE60212947T patent/DE60212947T2/de not_active Expired - Lifetime
- 2002-03-20 JP JP2002576218A patent/JP4161367B2/ja not_active Expired - Fee Related
- 2002-03-20 WO PCT/JP2002/002704 patent/WO2002076958A1/ja not_active Ceased
- 2002-03-20 AT AT02705404T patent/ATE332295T1/de not_active IP Right Cessation
- 2002-03-20 EP EP02705404A patent/EP1371649B1/de not_active Expired - Lifetime
- 2002-03-20 KR KR1020037012334A patent/KR100586671B1/ko not_active Expired - Fee Related
- 2002-03-20 IL IL15772402A patent/IL157724A0/xx active IP Right Grant
- 2002-03-20 CN CNB028068394A patent/CN100506805C/zh not_active Expired - Fee Related
-
2003
- 2003-09-03 IL IL157724A patent/IL157724A/en unknown
-
2006
- 2006-07-25 US US11/492,302 patent/US20070027324A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002076958A1 (en) | 2002-10-03 |
| DE60212947D1 (de) | 2006-08-17 |
| EP1371649B1 (de) | 2006-07-05 |
| CN100506805C (zh) | 2009-07-01 |
| JP4161367B2 (ja) | 2008-10-08 |
| EP1371649A1 (de) | 2003-12-17 |
| IL157724A (en) | 2008-06-05 |
| EP1371649A4 (de) | 2005-05-25 |
| IL157724A0 (en) | 2004-03-28 |
| JPWO2002076958A1 (ja) | 2004-10-21 |
| US20070027324A1 (en) | 2007-02-01 |
| US20040116711A1 (en) | 2004-06-17 |
| US7102010B2 (en) | 2006-09-05 |
| USRE40795E1 (en) | 2009-06-23 |
| KR100586671B1 (ko) | 2006-06-07 |
| KR20030083007A (ko) | 2003-10-23 |
| DE60212947T2 (de) | 2007-01-11 |
| CN1500084A (zh) | 2004-05-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |