ATE341343T1 - Medizinische zusammensetzungen mit diuretischem und die insulinresistenz verbesserndem mittel - Google Patents
Medizinische zusammensetzungen mit diuretischem und die insulinresistenz verbesserndem mittelInfo
- Publication number
- ATE341343T1 ATE341343T1 AT01271867T AT01271867T ATE341343T1 AT E341343 T1 ATE341343 T1 AT E341343T1 AT 01271867 T AT01271867 T AT 01271867T AT 01271867 T AT01271867 T AT 01271867T AT E341343 T1 ATE341343 T1 AT E341343T1
- Authority
- AT
- Austria
- Prior art keywords
- compositions containing
- insulin resistance
- improvement agent
- resistance improvement
- medical compositions
- Prior art date
Links
- 239000002934 diuretic Substances 0.000 title abstract 2
- 230000001882 diuretic effect Effects 0.000 title abstract 2
- 206010022489 Insulin Resistance Diseases 0.000 title 1
- 239000003795 chemical substances by application Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 208000001072 type 2 diabetes mellitus Diseases 0.000 title 1
- 229940122355 Insulin sensitizer Drugs 0.000 abstract 2
- 206010048612 Hydrothorax Diseases 0.000 abstract 1
- 206010030113 Oedema Diseases 0.000 abstract 1
- 210000001124 body fluid Anatomy 0.000 abstract 1
- 239000010839 body fluid Substances 0.000 abstract 1
- 230000000747 cardiac effect Effects 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000394424 | 2000-12-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE341343T1 true ATE341343T1 (de) | 2006-10-15 |
Family
ID=18860057
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01271867T ATE341343T1 (de) | 2000-12-26 | 2001-12-21 | Medizinische zusammensetzungen mit diuretischem und die insulinresistenz verbesserndem mittel |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US7199139B2 (de) |
| EP (2) | EP1354602B1 (de) |
| AT (1) | ATE341343T1 (de) |
| DE (1) | DE60123665T2 (de) |
| WO (1) | WO2002051441A1 (de) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8722668B2 (en) * | 1998-12-23 | 2014-05-13 | Daryl W. Hochman | Methods and compositions for the treatment of neuropathic pain and neuropsychiatric disorders |
| US8008283B2 (en) * | 1998-12-23 | 2011-08-30 | Neurotherapeutics Pharma, Inc. | Methods and compositions for the treatment of neuropsychiatric disorders |
| US7214711B2 (en) * | 1998-12-23 | 2007-05-08 | Neurotherapeutics Pharma Llc | Method of treating migraine headache without aura |
| US6414002B1 (en) | 1999-09-22 | 2002-07-02 | Bristol-Myers Squibb Company | Substituted acid derivatives useful as antidiabetic and antiobesity agents and method |
| US20070238740A1 (en) * | 2003-08-28 | 2007-10-11 | Nitromed, Inc. | Nitrosated And Nitrosylated Cardiovascular Compounds, Compositions And Methods Of Use |
| WO2005027967A1 (ja) * | 2003-09-17 | 2005-03-31 | Kaname Kawasugi | 医薬組成物 |
| US7420083B2 (en) * | 2003-09-25 | 2008-09-02 | Wyeth | Substituted aryloximes |
| CN1972715A (zh) * | 2004-03-29 | 2007-05-30 | 三共株式会社 | 含有胰岛素抵抗改善剂的糖尿病治疗剂 |
| AU2006216665A1 (en) * | 2005-02-24 | 2006-08-31 | Nicox S.A. | Nitric oxide enhancing diuretic compounds, compositions and methods of use |
| JP2009511629A (ja) * | 2005-10-17 | 2009-03-19 | ニューロセラピューティクス ファーマ, インコーポレイテッド | 中枢神経系疾患の調節に有用な利尿薬様化合物類似体 |
| EP2026659A4 (de) * | 2006-06-09 | 2010-06-30 | Wellstat Therapeutics Corp | Verbindungen zur behandlung von stoffwechselstörungen |
| JP5301465B2 (ja) | 2007-01-25 | 2013-09-25 | バーバ・ファーマシューティカルズ・リミテッド | インスリン抵抗性改善薬および治療方法 |
| ES2642586T3 (es) | 2009-07-27 | 2017-11-16 | Gilead Sciences, Inc. | Compuestos heterocíclicos condensados como moduladores de canales iónicos |
| EP2588197B1 (de) | 2010-07-02 | 2014-11-05 | Gilead Sciences, Inc. | Kondensierte heterozyklische verbindungen als ionenkanalmodulatoren |
| KR20140033377A (ko) | 2011-05-10 | 2014-03-18 | 길리애드 사이언시즈, 인코포레이티드 | 나트륨 채널 조절제로서의 융합된 헤테로시클릭 화합물 |
| NO3175985T3 (de) | 2011-07-01 | 2018-04-28 | ||
| UY34171A (es) | 2011-07-01 | 2013-01-31 | Gilead Sciences Inc | Compuestos heterocíclicos fusionados como moduladores del canal iónico |
| WO2013043925A1 (en) * | 2011-09-21 | 2013-03-28 | Gilead Sciences, Inc. | Sodium channel blockers reduce glucagon secretion |
Family Cites Families (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR240698A1 (es) | 1985-01-19 | 1990-09-28 | Takeda Chemical Industries Ltd | Procedimiento para preparar compuestos de 5-(4-(2-(5-etil-2-piridil)-etoxi)benzil)-2,4-tiazolidindiona y sus sales |
| FI91869C (fi) | 1987-03-18 | 1994-08-25 | Tanabe Seiyaku Co | Menetelmä antidiabeettisena aineena käytettävien bensoksatsolijohdannaisten valmistamiseksi |
| EP0842925A1 (de) | 1987-09-04 | 1998-05-20 | Beecham Group Plc | Substituierte Thiazolidindionderivate |
| JPH0713284Y2 (ja) * | 1987-09-21 | 1995-03-29 | 株式会社村田製作所 | 一体成形型誘電体フィルタの共振周波数調整構造 |
| US5594016A (en) | 1992-12-28 | 1997-01-14 | Mitsubishi Chemical Corporation | Naphthalene derivatives |
| HUT73431A (en) | 1993-04-30 | 1996-07-29 | Yamanouchi Pharma Co Ltd | Process for preparing novel bisoxadiazolidine derivatives and pharmaceutical compositions containing them |
| US5478852C1 (en) * | 1993-09-15 | 2001-03-13 | Sankyo Co | Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of impaired glucose tolerance in order to prevent or delay the onset of noninsulin-dependent diabetes mellitus |
| US5728720A (en) | 1993-12-27 | 1998-03-17 | Japan Tobacco Inc. | Isoxazolidinedione compounds and use thereof |
| ATE238297T1 (de) | 1994-10-20 | 2003-05-15 | Nippon Chemiphar Co | Chinolinderivat |
| WO1996028185A2 (en) * | 1995-03-16 | 1996-09-19 | Pfizer Inc. | Composition containing amlodipine, or a salt, or felodipine and an ace inhibitor |
| IL118474A (en) * | 1995-06-01 | 2001-08-08 | Sankyo Co | Benzimideol derivatives and pharmaceutical preparations containing them |
| JP3144624B2 (ja) | 1995-06-02 | 2001-03-12 | 杏林製薬株式会社 | N−ベンジルジオキソチアゾリジルベンズアミド誘導体及びその製造法 |
| ZA967800B (en) * | 1995-09-20 | 1997-04-03 | Yamanouchi Pharma Co Ltd | Heteroaryllsubstituted acryloylguanidine derivatives and pharmaceutical compositions comprising them |
| GB9604242D0 (en) | 1996-02-28 | 1996-05-01 | Glaxo Wellcome Inc | Chemical compounds |
| KR20000005224A (ko) * | 1996-04-04 | 2000-01-25 | 가와무라 요시부미 | 페닐알킬카르복실산 유도체_ |
| WO1999018066A1 (en) | 1997-10-02 | 1999-04-15 | Sankyo Company, Limited | Amidocarboxylic acid derivatives |
| WO1999019313A1 (en) | 1997-10-27 | 1999-04-22 | Dr. Reddy's Research Foundation | Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them |
| SE9801992D0 (sv) | 1998-06-04 | 1998-06-04 | Astra Ab | New 3-aryl-2-hydroxypropionic acid derivative I |
| RU2219172C2 (ru) | 1999-04-06 | 2003-12-20 | Санкио Компани, Лимитед | α-ЗАМЕЩЕННЫЕ ПРОИЗВОДНЫЕ КАРБОНОВЫХ КИСЛОТ |
| TWI249401B (en) * | 1999-04-14 | 2006-02-21 | Takeda Chemical Industries Ltd | Agent for improving ketosis |
| TWI284533B (en) | 1999-05-24 | 2007-08-01 | Sankyo Co | Pharmaceutical composition for treating hyperglycemia, impaired glucose tolerance, diabetes complications and for improving insulin resistant |
| PE20010580A1 (es) * | 1999-09-03 | 2001-05-25 | Takeda Chemical Industries Ltd | Composicion farmaceutica para tratar la diabetes |
| TWI302149B (en) | 1999-09-22 | 2008-10-21 | Bristol Myers Squibb Co | Substituted acid derivatives useful as antiodiabetic and antiobesity agents and method |
| JP2003518493A (ja) * | 1999-12-24 | 2003-06-10 | スミスクライン ビーチャム パブリック リミテッド カンパニー | 新規治療方法 |
| KR20070104953A (ko) * | 2000-03-17 | 2007-10-29 | 아지노모토 가부시키가이샤 | 신경 장애용 약제 |
| US20020013334A1 (en) * | 2000-06-15 | 2002-01-31 | Robl Jeffrey A. | HMG-CoA reductase inhibitors and method |
-
2001
- 2001-12-21 EP EP01271867A patent/EP1354602B1/de not_active Expired - Lifetime
- 2001-12-21 DE DE60123665T patent/DE60123665T2/de not_active Expired - Fee Related
- 2001-12-21 WO PCT/JP2001/011296 patent/WO2002051441A1/ja not_active Ceased
- 2001-12-21 EP EP06012545A patent/EP1695716A2/de not_active Withdrawn
- 2001-12-21 AT AT01271867T patent/ATE341343T1/de not_active IP Right Cessation
-
2003
- 2003-06-26 US US10/606,632 patent/US7199139B2/en not_active Expired - Fee Related
-
2005
- 2005-06-24 US US11/165,743 patent/US20050288339A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20050288339A1 (en) | 2005-12-29 |
| DE60123665T2 (de) | 2007-08-16 |
| EP1354602A1 (de) | 2003-10-22 |
| US7199139B2 (en) | 2007-04-03 |
| EP1354602A4 (de) | 2004-05-06 |
| EP1695716A2 (de) | 2006-08-30 |
| US20040053974A1 (en) | 2004-03-18 |
| DE60123665D1 (de) | 2006-11-16 |
| WO2002051441A1 (en) | 2002-07-04 |
| EP1354602B1 (de) | 2006-10-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |