ATE344265T1 - Derivate von benzothiazin und benzothiadiazin, verfahren zu ihrer herstellung und pharmazeutische zubereitungen diese enthaltend - Google Patents

Derivate von benzothiazin und benzothiadiazin, verfahren zu ihrer herstellung und pharmazeutische zubereitungen diese enthaltend

Info

Publication number: ATE344265T1
Authority: AT; Austria
Prior art keywords: benzothiadiazine; benzothiazine; derivatives; production; pharmaceutical preparations
Prior art date: 2003-06-13

Application number

AT04291435T

Other languages

English (en)

Inventor

Patrice Desos

Alex Cordi

Pierre Lestage

Original Assignee

Servier Lab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-06-13

Filing date

2004-06-09

Publication date

2006-11-15

2004-06-09 Application filed by Servier Lab filed Critical Servier Lab

2006-11-15 Application granted granted Critical

2006-11-15 Publication of ATE344265T1 publication Critical patent/ATE344265T1/de

Links

UJVBZCCNLAAMOV-UHFFFAOYSA-N 2h-1,2-benzothiazine Chemical class C1=CC=C2C=CNSC2=C1 UJVBZCCNLAAMOV-UHFFFAOYSA-N 0.000 title 1
HAVZTGSQJIEKPI-UHFFFAOYSA-N benzothiadiazine Chemical compound C1=CC=C2C=NNSC2=C1 HAVZTGSQJIEKPI-UHFFFAOYSA-N 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
238000000034 method Methods 0.000 title 1
239000000825 pharmaceutical preparation Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

AT04291435T 2003-06-13 2004-06-09 Derivate von benzothiazin und benzothiadiazin, verfahren zu ihrer herstellung und pharmazeutische zubereitungen diese enthaltend ATE344265T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0307118A FR2856065B1 (fr)	2003-06-13	2003-06-13	Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number	Publication Date
ATE344265T1 true ATE344265T1 (de)	2006-11-15

Family

ID=33186482

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04291435T ATE344265T1 (de)	2003-06-13	2004-06-09	Derivate von benzothiazin und benzothiadiazin, verfahren zu ihrer herstellung und pharmazeutische zubereitungen diese enthaltend

Country Status (27)

Country	Link
US (2)	US7253162B2 (de)
EP (1)	EP1486503B1 (de)
JP (1)	JP2005002114A (de)
KR (1)	KR100586683B1 (de)
CN (1)	CN1277823C (de)
AR (1)	AR044672A1 (de)
AT (1)	ATE344265T1 (de)
AU (1)	AU2004202586A1 (de)
BR (1)	BRPI0401956A (de)
CA (1)	CA2470263A1 (de)
CY (1)	CY1105939T1 (de)
DE (1)	DE602004002990T2 (de)
DK (1)	DK1486503T3 (de)
EA (1)	EA008797B1 (de)
EG (1)	EG24207A (de)
ES (1)	ES2276249T3 (de)
FR (1)	FR2856065B1 (de)
GE (1)	GEP20063815B (de)
HR (1)	HRP20070030T3 (de)
MA (1)	MA27092A1 (de)
MX (1)	MXPA04005580A (de)
NO (1)	NO20042422L (de)
NZ (1)	NZ533472A (de)
PL (1)	PL1486503T3 (de)
PT (1)	PT1486503E (de)
SG (1)	SG148023A1 (de)
SI (1)	SI1486503T1 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2879201B1 (fr) *	2004-12-10	2007-02-16	Servier Lab	Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
WO2007047397A2 (en)	2005-10-13	2007-04-26	Smithkline Beecham Corporation	Phenol ethers as modulators of the opioid receptors
EP2061761A1 (de) *	2006-09-07	2009-05-27	Millennium Pharmaceuticals, Inc.	Phenethylamid-derivate mit kinase-hemmungsaktivität
GB0821166D0 (en) *	2008-11-19	2008-12-24	Glaxo Group Ltd	Compounds
FR2955106B1 (fr) *	2010-01-08	2011-12-23	Servier Lab	Nouveaux derives de benzothiadiazines cyclopropylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
JP6134654B2 (ja) *	2012-02-08	2017-05-24	武田薬品工業株式会社	複素環化合物およびその用途
WO2019130229A1 (en) *	2017-12-28	2019-07-04	Mylan Laboratories Ltd	Methods and intermediates for preparing rucaparib

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR1377693A (fr) *	1962-12-06	1964-11-06	Geigy Ag J R	Nouveaux composés dibenzo [1.2] thiaziniques et produits pesticides qui en contiennent
FR2722502B1 (fr) *	1994-07-12	1996-08-23	Adir	Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent
HUP0101280A3 (en) *	1998-02-18	2003-02-28	Neurosearch As	Positive ampa receptor modulator compounds and their use
FR2823753B1 (fr) *	2001-04-18	2004-07-16	Servier Lab	Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine
FR2833950B1 (fr) *	2001-12-21	2005-12-16	Servier Lab	Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2833956B1 (fr) *	2001-12-21	2004-01-30	Servier Lab	Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

2003
- 2003-06-13 FR FR0307118A patent/FR2856065B1/fr not_active Expired - Fee Related
2004
- 2004-06-04 MA MA27721A patent/MA27092A1/fr unknown
- 2004-06-07 SG SG200404677-7A patent/SG148023A1/en unknown
- 2004-06-09 MX MXPA04005580A patent/MXPA04005580A/es active IP Right Grant
- 2004-06-09 AT AT04291435T patent/ATE344265T1/de not_active IP Right Cessation
- 2004-06-09 EP EP04291435A patent/EP1486503B1/de not_active Expired - Lifetime
- 2004-06-09 DK DK04291435T patent/DK1486503T3/da active
- 2004-06-09 PT PT04291435T patent/PT1486503E/pt unknown
- 2004-06-09 PL PL04291435T patent/PL1486503T3/pl unknown
- 2004-06-09 ES ES04291435T patent/ES2276249T3/es not_active Expired - Lifetime
- 2004-06-09 SI SI200430111T patent/SI1486503T1/sl unknown
- 2004-06-09 DE DE602004002990T patent/DE602004002990T2/de not_active Expired - Fee Related
- 2004-06-10 NO NO20042422A patent/NO20042422L/no not_active Application Discontinuation
- 2004-06-10 EG EG2004060261A patent/EG24207A/xx active
- 2004-06-10 US US10/865,184 patent/US7253162B2/en not_active Expired - Fee Related
- 2004-06-11 EA EA200400666A patent/EA008797B1/ru not_active IP Right Cessation
- 2004-06-11 AU AU2004202586A patent/AU2004202586A1/en not_active Abandoned
- 2004-06-11 CA CA002470263A patent/CA2470263A1/fr not_active Abandoned
- 2004-06-11 AR ARP040102023A patent/AR044672A1/es unknown
- 2004-06-11 GE GE5557A patent/GEP20063815B/en unknown
- 2004-06-11 NZ NZ533472A patent/NZ533472A/en unknown
- 2004-06-11 KR KR1020040042991A patent/KR100586683B1/ko not_active Expired - Fee Related
- 2004-06-14 BR BR0401956-3A patent/BRPI0401956A/pt not_active IP Right Cessation
- 2004-06-14 JP JP2004175278A patent/JP2005002114A/ja active Pending
- 2004-06-14 CN CNB2004100482744A patent/CN1277823C/zh not_active Expired - Fee Related
2007
- 2007-01-16 CY CY20071100074T patent/CY1105939T1/el unknown
- 2007-02-01 HR HR20070030T patent/HRP20070030T3/xx unknown
- 2007-06-27 US US11/823,439 patent/US7423034B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
EA200400666A3 (ru)	2005-10-27
ES2276249T3 (es)	2007-06-16
PT1486503E (pt)	2007-01-31
EG24207A (en)	2008-10-21
SI1486503T1 (sl)	2007-02-28
EA200400666A2 (ru)	2004-12-30
FR2856065B1 (fr)	2005-08-19
US20040254161A1 (en)	2004-12-16
US20070249594A1 (en)	2007-10-25
GEP20063815B (en)	2006-05-10
AR044672A1 (es)	2005-09-21
NZ533472A (en)	2005-09-30
KR20040107410A (ko)	2004-12-20
BRPI0401956A (pt)	2005-06-28
MA27092A1 (fr)	2004-12-20
CN1277823C (zh)	2006-10-04
CY1105939T1 (el)	2011-04-06
AU2004202586A1 (en)	2005-01-06
CN1572791A (zh)	2005-02-02
EA008797B1 (ru)	2007-08-31
DK1486503T3 (da)	2007-02-26
DE602004002990T2 (de)	2007-07-05
KR100586683B1 (ko)	2006-06-08
US7423034B2 (en)	2008-09-09
SG148023A1 (en)	2008-12-31
DE602004002990D1 (de)	2006-12-14
HK1071750A1 (en)	2005-07-29
EP1486503B1 (de)	2006-11-02
PL1486503T3 (pl)	2006-12-29
HRP20070030T3 (en)	2007-08-31
CA2470263A1 (fr)	2004-12-13
JP2005002114A (ja)	2005-01-06
NO20042422L (no)	2004-12-14
FR2856065A1 (fr)	2004-12-17
EP1486503A1 (de)	2004-12-15
MXPA04005580A (es)	2005-03-23
US7253162B2 (en)	2007-08-07

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2007-06-15

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