ATE346074T1 - Dna methyl transferase inhibitoren - Google Patents

Dna methyl transferase inhibitoren

Info

Publication number
ATE346074T1
ATE346074T1 AT01987166T AT01987166T ATE346074T1 AT E346074 T1 ATE346074 T1 AT E346074T1 AT 01987166 T AT01987166 T AT 01987166T AT 01987166 T AT01987166 T AT 01987166T AT E346074 T1 ATE346074 T1 AT E346074T1
Authority
AT
Austria
Prior art keywords
transferase inhibitors
methyl transferase
dna methyl
inhibitors
dna
Prior art date
Application number
AT01987166T
Other languages
English (en)
Inventor
Stephen J Benkovic
Lucille Shapiro
Stephen J Baker
Daphne C Wahnon
Mark Wall
Vincent K Shier
Charles P Scott
Justin Baboval
Original Assignee
Penn State Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Penn State Res Found filed Critical Penn State Res Found
Application granted granted Critical
Publication of ATE346074T1 publication Critical patent/ATE346074T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT01987166T 2000-11-30 2001-11-29 Dna methyl transferase inhibitoren ATE346074T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25020200P 2000-11-30 2000-11-30

Publications (1)

Publication Number Publication Date
ATE346074T1 true ATE346074T1 (de) 2006-12-15

Family

ID=22946721

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01987166T ATE346074T1 (de) 2000-11-30 2001-11-29 Dna methyl transferase inhibitoren

Country Status (7)

Country Link
EP (1) EP1339725B1 (de)
JP (1) JP2004524281A (de)
AT (1) ATE346074T1 (de)
AU (2) AU2002239407B2 (de)
CA (1) CA2430562C (de)
DE (1) DE60124759T2 (de)
WO (1) WO2002044184A2 (de)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2001289079A1 (en) * 2000-09-13 2002-03-26 Praecis Pharmaceuticals Incorporated Pharmaceutical compositions for sustained drug delivery
AU2003205089B2 (en) 2002-01-10 2007-01-25 The Pennsylvania State Research Foundation Methods for the preparation of alkyl diaryl borinates and complexed diarylborinic acids
JP5038912B2 (ja) 2005-02-16 2012-10-03 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子
US7767657B2 (en) 2005-02-16 2010-08-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
NZ570257A (en) 2006-02-16 2011-11-25 Anacor Pharmaceuticals Inc Boron-containing small molecules as anti-inflammatory agents
JP2009184988A (ja) * 2008-02-07 2009-08-20 Institute Of Physical & Chemical Research 新規ホウ素化合物及びそれを含む細胞内カルシウム濃度調節剤又は医薬組成物
BRPI0908565A2 (pt) 2008-03-06 2017-05-23 Anacor Pharmaceuticals Inc composto, formulação farmacêutica, métodos para reduzir a liberação de uma citocina ou de uma quimiocina, para tratar uma condição em um animal e para inibir uma fosfodiesterase
JP5606913B2 (ja) * 2008-08-11 2014-10-15 独立行政法人科学技術振興機構 蛋白質架橋阻害剤
EP2348863A4 (de) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc Borhaltige kleine moleküle
US8461336B2 (en) 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US9493489B2 (en) 2008-10-15 2016-11-15 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
MX2011006334A (es) 2008-12-17 2011-09-22 Anacor Pharmaceuticals Inc Polimorfos de (s)-3-amino-metil-7-(3-hidroxi-propoxi)-3h-benzo-[c] [1,2]-oxaborol-1-ol.
EP2445536B1 (de) 2009-06-22 2016-06-08 Burnham Institute for Medical Research Verfahren und zusammensetzungen mit peptiden und proteinen mit c-terminalen elementen
KR20130031233A (ko) 2009-07-28 2013-03-28 아나코르 파마슈티칼스 인코포레이티드 삼치환된 붕소 함유 분자
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011079304A1 (en) 2009-12-23 2011-06-30 Sanford-Burnham Medical Research Institute Methods and compositions related to annexin 1-binding compounds
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
CA2795289A1 (en) 2010-04-08 2011-10-13 Sanford-Burnham Medical Research Institute Methods and compositions for enhanced delivery of compounds
EP2598146A1 (de) 2010-07-29 2013-06-05 Corning Incorporated Verfahren zur identifizierung von zielen und molekülen zur purinosomenregulierung und ihre verwendung
SG10201507032YA (en) 2010-09-07 2015-10-29 Anacor Pharmaceuticals Inc Benzoxaborole derivatives for treating bacterial infections
WO2012118778A1 (en) 2011-02-28 2012-09-07 Sanford-Burnham Medical Research Institute Truncated car peptides and methods and compositions using truncated car peptides
WO2012166585A2 (en) 2011-05-31 2012-12-06 Airware, Inc. Re-calibration of ab ndir gas sensors
KR101756785B1 (ko) * 2015-03-10 2017-07-12 한국화학연구원 4배위 유기 붕소 화합물의 제조방법
US11981752B2 (en) 2017-05-02 2024-05-14 Sanford Burnham Prebys Medical Discovery Institute Tumor associated monocyte/macrophage binding peptide and methods of use thereof
US12583888B2 (en) 2019-02-04 2026-03-24 University Of Tartu Bi-specific extracellular matrix binding peptides and methods of use thereof
CN114703301B (zh) * 2022-01-11 2024-01-26 武汉明了生物科技有限公司 一种鉴定三种鲍特菌的引物组、试剂盒及其应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3485864A (en) * 1965-01-12 1969-12-23 Minnesota Mining & Mfg Diphenylborinic acid esters
FR2071171A6 (en) * 1969-12-19 1971-09-17 Rhone Poulenc Sa 1,1-diphenyl-azaborolidines - with insecticidal acaricidal - herbicidal and fungicidal activity
US4713346A (en) * 1986-02-03 1987-12-15 The Children's Medical Center Corporation Formation of analyzable boron containing adducts
DE19829949A1 (de) * 1998-07-04 2000-01-05 Bayer Ag Elektrolumineszierende Anordnungen unter Verwendung von Bor-Chelaten von 8-Aminochinolin-Derivaten
EP1155698A4 (de) * 1999-01-29 2003-01-15 Nitto Kasei Co Ltd Organoborverbindungen mit antikokzidischer aktivität
CN1370170A (zh) * 1999-05-25 2002-09-18 宾夕法尼亚州研究基金会 Dna甲基转移酶抑制剂

Also Published As

Publication number Publication date
AU3940702A (en) 2002-06-11
CA2430562A1 (en) 2002-06-06
JP2004524281A (ja) 2004-08-12
AU2002239407B2 (en) 2007-12-06
WO2002044184A2 (en) 2002-06-06
WO2002044184A3 (en) 2003-02-27
DE60124759D1 (en) 2007-01-04
EP1339725B1 (de) 2006-11-22
DE60124759T2 (de) 2007-03-15
EP1339725A2 (de) 2003-09-03
CA2430562C (en) 2010-02-02

Similar Documents

Publication Publication Date Title
DE60124759D1 (en) Dna methyl transferase inhibitoren
WO2000075142A3 (en) Dna methyltransferase inhibitors
EP1377587A4 (de) Proteinphosphatinhibitoren
NO20005224D0 (no) BTK inhibitorer og fremgangsmÕter for deres identifikasjon og anvendelse
EA200501928A1 (ru) Пирролодигидроизохинолины как ингибиторы pde10
CY1109006T1 (el) Παραγωγα πουρινης ως αναστολεις κινασης
SV2003001103A (es) Formulaciones autoemulsionantes de inhibidores de la proteina de transferencia de colesteril ester pc10894
BRPI0616630B8 (pt) compostos de pirazol substituídos
GB2386224A (en) Global electronic trading system
AU5553801A (en) Heterocycles that are inhibitors of impdh enzyme
DE60122216D1 (de) Zolpidem Hemitartrat Solvat
DE69913712D1 (de) Inhibitoren der bakteriellen nad synthetase
ATE311397T1 (de) Sulfonamidomethyl phosphonat beta-lactamase inhibitoren
WO2002018954A3 (en) Inhibition of cmv infection and dissemination
NO20033921L (no) Inhibitor av monoaminopptak
AU2576901A (en) Agents and methods for the treatment of proliferative diseases
SE0302965D0 (sv) Hämmare av DNA-Metyltransferasisoformer
MXPA03004878A (es) Nuevos inhibidores de la transferasa de la proteina farnesilo.
DK1438411T3 (da) Anvendelse af aminogylcosid-resistensgen
DE60037113D1 (de) Glycosyltransferase inhibitoren
CY1108517T1 (el) Σκεyασμα 2-μεθυλο-θειενο-βενζοδιαζεπiνης
EP1343870A4 (de) Bakterielle expressionssysteme
DE60232650D1 (de) Peptiddeformylaseinhibitoren
HN2000000084A (es) Inhibidores de metaloproteasa.
GB0128943D0 (en) Bacterial enzyme inhibitors

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties