ATE346074T1 - Dna methyl transferase inhibitoren - Google Patents

Dna methyl transferase inhibitoren

Info

Publication number
ATE346074T1
ATE346074T1 AT01987166T AT01987166T ATE346074T1 AT E346074 T1 ATE346074 T1 AT E346074T1 AT 01987166 T AT01987166 T AT 01987166T AT 01987166 T AT01987166 T AT 01987166T AT E346074 T1 ATE346074 T1 AT E346074T1
Authority
AT
Austria
Prior art keywords
transferase inhibitors
methyl transferase
dna methyl
inhibitors
dna
Prior art date
Application number
AT01987166T
Other languages
English (en)
Inventor
Stephen J Benkovic
Lucille Shapiro
Stephen J Baker
Daphne C Wahnon
Mark Wall
Vincent K Shier
Charles P Scott
Justin Baboval
Original Assignee
Penn State Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Penn State Res Found filed Critical Penn State Res Found
Application granted granted Critical
Publication of ATE346074T1 publication Critical patent/ATE346074T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT01987166T 2000-11-30 2001-11-29 Dna methyl transferase inhibitoren ATE346074T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US25020200P 2000-11-30 2000-11-30

Publications (1)

Publication Number Publication Date
ATE346074T1 true ATE346074T1 (de) 2006-12-15

Family

ID=22946721

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01987166T ATE346074T1 (de) 2000-11-30 2001-11-29 Dna methyl transferase inhibitoren

Country Status (7)

Country Link
EP (1) EP1339725B1 (de)
JP (1) JP2004524281A (de)
AT (1) ATE346074T1 (de)
AU (2) AU2002239407B2 (de)
CA (1) CA2430562C (de)
DE (1) DE60124759T2 (de)
WO (1) WO2002044184A2 (de)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7037889B2 (en) * 2000-09-13 2006-05-02 Praecis Pharmaceuticals Inc. Pharmaceutical compositions for sustained drug delivery
AU2003205089B2 (en) * 2002-01-10 2007-01-25 The Pennsylvania State Research Foundation Methods for the preparation of alkyl diaryl borinates and complexed diarylborinic acids
SI3424932T1 (sl) 2005-02-16 2021-08-31 Anacor Pharmaceuticals, Inc. Boronoftalidi za terapevtsko uporabo
WO2007078340A2 (en) 2005-12-30 2007-07-12 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
PT1988779E (pt) 2006-02-16 2015-09-04 Anacor Pharmaceuticals Inc Moléculas pequenas contendo boro como agentes antiinflamatórios
JP2009184988A (ja) * 2008-02-07 2009-08-20 Institute Of Physical & Chemical Research 新規ホウ素化合物及びそれを含む細胞内カルシウム濃度調節剤又は医薬組成物
NZ587955A (en) 2008-03-06 2012-10-26 Anacor Pharmaceuticals Inc Boron-containing small molecules as anti-inflammatory agents
WO2010018836A2 (ja) * 2008-08-11 2010-02-18 独立行政法人科学技術振興機構 ポリグルタミン凝集阻害剤
US8461336B2 (en) 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
EP2348863A4 (de) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc Borhaltige kleine moleküle
US9493489B2 (en) 2008-10-15 2016-11-15 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
MA32977B1 (fr) 2008-12-17 2012-01-02 Anacor Pharmaceuticals Inc Formes polymorphiques du (s)-3-aminomethyl-7-(3-hydroxy-propoxy)-3h-benzo(c(1,2)oxaborol-1-ol
EP2445536B1 (de) 2009-06-22 2016-06-08 Burnham Institute for Medical Research Verfahren und zusammensetzungen mit peptiden und proteinen mit c-terminalen elementen
RU2012107163A (ru) 2009-07-28 2013-09-10 Анакор Фармасьютикалз, Инк. Тризамещенные борсодержащие молекулы
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
US9346834B2 (en) 2009-10-20 2016-05-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110212918A1 (en) 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
SG10201704812TA (en) 2009-12-23 2017-07-28 Sanford-Burnham Medical Res Inst Methods and compositions related to annexin 1-binding compounds
US8716478B2 (en) 2010-01-27 2014-05-06 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
WO2011127405A1 (en) 2010-04-08 2011-10-13 Sanford-Burnham Medical Research Institute Methods and compositions for enhanced delivery of compounds
JP2013532990A (ja) 2010-07-29 2013-08-22 コーニング インコーポレイテッド プリノソームを調節する標的および分子を同定する方法ならびにそれらの使用
MX338209B (es) 2010-09-07 2016-04-07 Anacor Pharmaceuticals Inc Derivados de benzoxaborol para tratar infecciones bacterianas.
WO2012118778A1 (en) 2011-02-28 2012-09-07 Sanford-Burnham Medical Research Institute Truncated car peptides and methods and compositions using truncated car peptides
WO2012166585A2 (en) 2011-05-31 2012-12-06 Airware, Inc. Re-calibration of ab ndir gas sensors
KR101756785B1 (ko) * 2015-03-10 2017-07-12 한국화학연구원 4배위 유기 붕소 화합물의 제조방법
EP3628047A1 (de) 2017-05-02 2020-04-01 Sanford Burnham Prebys Medical Discovery Institute Tumorassoziiertes monozyten-/makrophagenbindendes peptid und verfahren zur verwendung davon
US12583888B2 (en) 2019-02-04 2026-03-24 University Of Tartu Bi-specific extracellular matrix binding peptides and methods of use thereof
CN114703301B (zh) * 2022-01-11 2024-01-26 武汉明了生物科技有限公司 一种鉴定三种鲍特菌的引物组、试剂盒及其应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3485864A (en) * 1965-01-12 1969-12-23 Minnesota Mining & Mfg Diphenylborinic acid esters
FR2071171A6 (en) * 1969-12-19 1971-09-17 Rhone Poulenc Sa 1,1-diphenyl-azaborolidines - with insecticidal acaricidal - herbicidal and fungicidal activity
US4713346A (en) * 1986-02-03 1987-12-15 The Children's Medical Center Corporation Formation of analyzable boron containing adducts
DE19829949A1 (de) * 1998-07-04 2000-01-05 Bayer Ag Elektrolumineszierende Anordnungen unter Verwendung von Bor-Chelaten von 8-Aminochinolin-Derivaten
EP1155698A4 (de) * 1999-01-29 2003-01-15 Nitto Kasei Co Ltd Organoborverbindungen mit antikokzidischer aktivität
CN1370170A (zh) * 1999-05-25 2002-09-18 宾夕法尼亚州研究基金会 Dna甲基转移酶抑制剂

Also Published As

Publication number Publication date
EP1339725B1 (de) 2006-11-22
WO2002044184A3 (en) 2003-02-27
CA2430562A1 (en) 2002-06-06
WO2002044184A2 (en) 2002-06-06
AU2002239407B2 (en) 2007-12-06
JP2004524281A (ja) 2004-08-12
DE60124759T2 (de) 2007-03-15
EP1339725A2 (de) 2003-09-03
AU3940702A (en) 2002-06-11
DE60124759D1 (en) 2007-01-04
CA2430562C (en) 2010-02-02

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