ATE349421T1 - Benzamidoacetonitrilderivate und ihre verwendung als antiparasitika - Google Patents
Benzamidoacetonitrilderivate und ihre verwendung als antiparasitikaInfo
- Publication number
- ATE349421T1 ATE349421T1 AT02745292T AT02745292T ATE349421T1 AT E349421 T1 ATE349421 T1 AT E349421T1 AT 02745292 T AT02745292 T AT 02745292T AT 02745292 T AT02745292 T AT 02745292T AT E349421 T1 ATE349421 T1 AT E349421T1
- Authority
- AT
- Austria
- Prior art keywords
- benzamidoacetonitril
- antiparasitics
- derivatives
- compounds
- enantiomers
- Prior art date
Links
- 229940125687 antiparasitic agent Drugs 0.000 title 1
- 239000003096 antiparasitic agent Substances 0.000 title 1
- LPKZSPQPPSEVSX-UHFFFAOYSA-N n-(cyanomethyl)benzamide Chemical class N#CCNC(=O)C1=CC=CC=C1 LPKZSPQPPSEVSX-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 244000045947 parasite Species 0.000 abstract 1
- 230000000361 pesticidal effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
- C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
- C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C251/32—Oximes
- C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
- C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
- C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D335/10—Dibenzothiopyrans; Hydrogenated dibenzothiopyrans
- C07D335/12—Thioxanthenes
- C07D335/14—Thioxanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
- C07D335/16—Oxygen atoms, e.g. thioxanthones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
- C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
- C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
- C07C2603/18—Fluorenes; Hydrogenated fluorenes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
- C07C2603/26—Phenanthrenes; Hydrogenated phenanthrenes
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH9192001 | 2001-05-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE349421T1 true ATE349421T1 (de) | 2007-01-15 |
Family
ID=4548043
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02745292T ATE349421T1 (de) | 2001-05-15 | 2002-05-14 | Benzamidoacetonitrilderivate und ihre verwendung als antiparasitika |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7705044B2 (de) |
| EP (1) | EP1390344B1 (de) |
| JP (1) | JP4124661B2 (de) |
| KR (1) | KR100628842B1 (de) |
| CN (1) | CN1241907C (de) |
| AT (1) | ATE349421T1 (de) |
| AU (1) | AU2002316903B2 (de) |
| BR (1) | BR0209828A (de) |
| CA (1) | CA2447084A1 (de) |
| CO (1) | CO5540291A2 (de) |
| DE (1) | DE60217099T2 (de) |
| MX (1) | MXPA03010404A (de) |
| NZ (1) | NZ529368A (de) |
| RU (1) | RU2284990C2 (de) |
| WO (1) | WO2002092552A2 (de) |
| ZA (1) | ZA200308592B (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE60126838T2 (de) * | 2000-12-20 | 2007-11-08 | Novartis Ag | Amidoacetonitrile zur Bekämpfung von Endoparasiten |
| TW200305556A (en) * | 2002-03-21 | 2003-11-01 | Novartis Ag | Organic compounds |
| GB0402677D0 (en) * | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| PT3088384T (pt) * | 2007-05-15 | 2019-03-22 | Aventis Agriculture | Compostos de ariloazol-2-il-cianoetilamino, método de fabrico e seu método de utilização |
| KR101782311B1 (ko) | 2008-10-21 | 2017-09-27 | 메리얼 인코포레이티드 | 티오아미드 화합물, 이의 제조 방법 및 사용 방법 |
| AR074024A1 (es) | 2008-11-14 | 2010-12-15 | Merial Ltd | Compuesto de arilazol-2-il-cianoetilamino enantiomericamente enriquecidos, composicion plaguicida y su uso para prevenir la infeccion parasitaria |
| US8822689B2 (en) | 2012-09-19 | 2014-09-02 | Merial Limited | Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4873224A (en) * | 1988-05-23 | 1989-10-10 | Merck & Co., Inc. | Avermectin derivatives |
| NZ231773A (en) * | 1988-12-23 | 1992-09-25 | Merck & Co Inc | Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof |
| RU2127256C1 (ru) * | 1992-07-15 | 1999-03-10 | Басф Аг | Замещенные простые оксимовые эфиры и фунгицидное, инсектицидное, арахноицидное средство |
| US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
| AR037746A1 (es) * | 2001-12-06 | 2004-12-01 | Novartis Ag | Compuestos derivados de amidoacetonitrilo, un procedimiento para su preparacion, un procedimiento para la preparacion de compuestos intermediarios, una composicion para combatir parasitos, un procedimiento para combatir dichos parasitos, y el empleo de dichos derivados para la preparacion de una com |
| TW200400932A (en) * | 2002-06-19 | 2004-01-16 | Novartis Ag | Organic compounds |
-
2002
- 2002-05-14 RU RU2003134179/04A patent/RU2284990C2/ru not_active IP Right Cessation
- 2002-05-14 US US10/477,289 patent/US7705044B2/en not_active Expired - Fee Related
- 2002-05-14 CA CA002447084A patent/CA2447084A1/en not_active Abandoned
- 2002-05-14 DE DE60217099T patent/DE60217099T2/de not_active Expired - Lifetime
- 2002-05-14 MX MXPA03010404A patent/MXPA03010404A/es unknown
- 2002-05-14 CN CNB028119355A patent/CN1241907C/zh not_active Expired - Fee Related
- 2002-05-14 WO PCT/EP2002/005294 patent/WO2002092552A2/en not_active Ceased
- 2002-05-14 KR KR1020037014727A patent/KR100628842B1/ko not_active Expired - Fee Related
- 2002-05-14 BR BR0209828-8A patent/BR0209828A/pt not_active IP Right Cessation
- 2002-05-14 JP JP2002589438A patent/JP4124661B2/ja not_active Expired - Fee Related
- 2002-05-14 AU AU2002316903A patent/AU2002316903B2/en not_active Ceased
- 2002-05-14 AT AT02745292T patent/ATE349421T1/de not_active IP Right Cessation
- 2002-05-14 NZ NZ529368A patent/NZ529368A/en not_active IP Right Cessation
- 2002-05-14 EP EP02745292A patent/EP1390344B1/de not_active Expired - Lifetime
-
2003
- 2003-11-04 ZA ZA200308592A patent/ZA200308592B/en unknown
- 2003-12-12 CO CO03108977A patent/CO5540291A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002092552A3 (en) | 2003-12-11 |
| CA2447084A1 (en) | 2002-11-21 |
| NZ529368A (en) | 2005-06-24 |
| DE60217099T2 (de) | 2007-08-09 |
| MXPA03010404A (es) | 2004-03-09 |
| CO5540291A2 (es) | 2005-07-29 |
| KR100628842B1 (ko) | 2006-09-29 |
| JP2004533451A (ja) | 2004-11-04 |
| AU2002316903B2 (en) | 2006-01-12 |
| US20040220055A1 (en) | 2004-11-04 |
| BR0209828A (pt) | 2004-06-15 |
| US7705044B2 (en) | 2010-04-27 |
| RU2284990C2 (ru) | 2006-10-10 |
| WO2002092552A2 (en) | 2002-11-21 |
| EP1390344B1 (de) | 2006-12-27 |
| RU2003134179A (ru) | 2005-06-10 |
| CN1531525A (zh) | 2004-09-22 |
| ZA200308592B (en) | 2004-09-03 |
| EP1390344A2 (de) | 2004-02-25 |
| KR20030094406A (ko) | 2003-12-11 |
| JP4124661B2 (ja) | 2008-07-23 |
| CN1241907C (zh) | 2006-02-15 |
| DE60217099D1 (de) | 2007-02-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |