ATE360015T1 - Protein tyrosin kinase inhibitoren - Google Patents

Protein tyrosin kinase inhibitoren

Info

Publication number
ATE360015T1
ATE360015T1 AT03771039T AT03771039T ATE360015T1 AT E360015 T1 ATE360015 T1 AT E360015T1 AT 03771039 T AT03771039 T AT 03771039T AT 03771039 T AT03771039 T AT 03771039T AT E360015 T1 ATE360015 T1 AT E360015T1
Authority
AT
Austria
Prior art keywords
tyrosine kinase
kinase inhibitors
protein tyrosine
compounds
stereoisomers
Prior art date
Application number
AT03771039T
Other languages
English (en)
Inventor
Ghenadie Rusu
Jianhua Zhong
Natalie Lazarowych
Martyn Brown
George Ma
Stephen Houldsworth
Original Assignee
Critical Outcome Technologies
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Critical Outcome Technologies filed Critical Critical Outcome Technologies
Application granted granted Critical
Publication of ATE360015T1 publication Critical patent/ATE360015T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT03771039T 2002-07-31 2003-07-31 Protein tyrosin kinase inhibitoren ATE360015T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US39940802P 2002-07-31 2002-07-31

Publications (1)

Publication Number Publication Date
ATE360015T1 true ATE360015T1 (de) 2007-05-15

Family

ID=31188578

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03771039T ATE360015T1 (de) 2002-07-31 2003-07-31 Protein tyrosin kinase inhibitoren

Country Status (7)

Country Link
US (2) US7585866B2 (de)
EP (1) EP1542989B1 (de)
AT (1) ATE360015T1 (de)
AU (1) AU2003250701A1 (de)
CA (1) CA2494061C (de)
DE (1) DE60313339T2 (de)
WO (1) WO2004011456A1 (de)

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ATE360015T1 (de) 2002-07-31 2007-05-15 Critical Outcome Technologies Protein tyrosin kinase inhibitoren
ATE380810T1 (de) 2002-10-09 2007-12-15 Critical Outcome Technologies Protein-tyrosine-kinase-inhibitoren
BRPI0519424B8 (pt) 2004-12-28 2021-05-25 Athenex Inc compostos, composição e uso dos ditos compostos para a preparação de um medicamento para prevenção ou tratamento de um distúrbio de proliferação celular ou infecção microbiana
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US7939529B2 (en) 2007-05-17 2011-05-10 Kinex Pharmaceuticals, Llc Process for the preparation of compositions for modulating a kinase cascade and methods of use thereof
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JP6499076B2 (ja) 2012-08-30 2019-04-10 アセネックス インコーポレイテッド タンパク質チロシンキナーゼ調節因子としてのｎ−（３−フルオロベンジル）−２−（５−（４−モルホリノフェニル）ピリジン−２−イル）アセトアミド

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Also Published As

Publication number Publication date
WO2004011456A1 (en) 2004-02-05
DE60313339D1 (de) 2007-05-31
CA2494061C (en) 2011-06-14
US20090298855A1 (en) 2009-12-03
WO2004011456A9 (en) 2005-06-02
WO2004011456A8 (en) 2004-08-05
CA2494061A1 (en) 2004-02-05
US20060069105A1 (en) 2006-03-30
EP1542989A1 (de) 2005-06-22
EP1542989B1 (de) 2007-04-18
US8252800B2 (en) 2012-08-28
DE60313339T2 (de) 2008-01-03
US7585866B2 (en) 2009-09-08
AU2003250701A1 (en) 2004-02-16

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