ATE360015T1 - Protein tyrosin kinase inhibitoren - Google Patents

Protein tyrosin kinase inhibitoren

Info

Publication number
ATE360015T1
ATE360015T1 AT03771039T AT03771039T ATE360015T1 AT E360015 T1 ATE360015 T1 AT E360015T1 AT 03771039 T AT03771039 T AT 03771039T AT 03771039 T AT03771039 T AT 03771039T AT E360015 T1 ATE360015 T1 AT E360015T1
Authority
AT
Austria
Prior art keywords
tyrosine kinase
kinase inhibitors
protein tyrosine
compounds
stereoisomers
Prior art date
Application number
AT03771039T
Other languages
English (en)
Inventor
Ghenadie Rusu
Jianhua Zhong
Natalie Lazarowych
Martyn Brown
George Ma
Stephen Houldsworth
Original Assignee
Critical Outcome Technologies
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Critical Outcome Technologies filed Critical Critical Outcome Technologies
Application granted granted Critical
Publication of ATE360015T1 publication Critical patent/ATE360015T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT03771039T 2002-07-31 2003-07-31 Protein tyrosin kinase inhibitoren ATE360015T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US39940802P 2002-07-31 2002-07-31

Publications (1)

Publication Number Publication Date
ATE360015T1 true ATE360015T1 (de) 2007-05-15

Family

ID=31188578

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03771039T ATE360015T1 (de) 2002-07-31 2003-07-31 Protein tyrosin kinase inhibitoren

Country Status (7)

Country Link
US (2) US7585866B2 (de)
EP (1) EP1542989B1 (de)
AT (1) ATE360015T1 (de)
AU (1) AU2003250701A1 (de)
CA (1) CA2494061C (de)
DE (1) DE60313339T2 (de)
WO (1) WO2004011456A1 (de)

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DE60313339T2 (de) 2002-07-31 2008-01-03 Critical Outcome Technologies, Inc. Protein tyrosin kinase inhibitoren
US7629347B2 (en) 2002-10-09 2009-12-08 Critical Outcome Technologies, Inc. Protein tyrosine kinase inhibitors
US7968574B2 (en) 2004-12-28 2011-06-28 Kinex Pharmaceuticals, Llc Biaryl compositions and methods for modulating a kinase cascade
ES2382068T3 (es) 2004-12-28 2012-06-05 Kinex Pharmaceuticals, Llc Composiciones y métodos para tratar trastornos de proliferación celular
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US7935697B2 (en) 2006-12-28 2011-05-03 Kinex Pharmaceuticals, Llc Compositions for modulating a kinase cascade and methods of use thereof
US7939529B2 (en) 2007-05-17 2011-05-10 Kinex Pharmaceuticals, Llc Process for the preparation of compositions for modulating a kinase cascade and methods of use thereof
EP2727909A1 (de) 2007-03-16 2014-05-07 The Scripps Research Institute Inhibitoren von focal adhesion kinase
CA2710039C (en) 2007-12-26 2018-07-03 Critical Outcome Technologies, Inc. Semicarbazones, thiosemicarbazones and related compounds and methods for treatment of cancer
EP2318406B1 (de) 2008-07-17 2016-01-27 Critical Outcome Technologies, Inc. Thiosemicarbazonhemmerverbindungen und krebsbehandlungsverfahren
GB0910537D0 (en) 2009-06-18 2009-07-29 Ivax Pharmaceuticals Ireland Inhaler
TW201103904A (en) * 2009-06-11 2011-02-01 Hoffmann La Roche Janus kinase inhibitor compounds and methods
EP2552915B1 (de) 2010-04-01 2017-07-19 Critical Outcome Technologies Inc. Verbindungen zur behandlung von hiv
WO2011129936A2 (en) 2010-04-16 2011-10-20 Kinex Pharmaceuticals, Llc Compositions and methods for the prevention and treatment of cancer
CN102477009B (zh) * 2010-11-23 2014-01-01 清华大学深圳研究生院 取代的（s）-苯甲磺酰基吡咯烷-3-氨基衍生物及其制备方法与应用
CA2883144C (en) 2012-08-30 2023-01-17 Kinex Pharmaceuticals, Llc N-(3-fluorobenzyl)-2-(5-(4-morpholinophenyl)pyridin-2-yl) acetamide as protein|tyrosine kinase modulators

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Also Published As

Publication number Publication date
US7585866B2 (en) 2009-09-08
DE60313339D1 (de) 2007-05-31
WO2004011456A9 (en) 2005-06-02
AU2003250701A1 (en) 2004-02-16
CA2494061C (en) 2011-06-14
DE60313339T2 (de) 2008-01-03
US8252800B2 (en) 2012-08-28
US20060069105A1 (en) 2006-03-30
US20090298855A1 (en) 2009-12-03
WO2004011456A8 (en) 2004-08-05
EP1542989A1 (de) 2005-06-22
EP1542989B1 (de) 2007-04-18
CA2494061A1 (en) 2004-02-05
WO2004011456A1 (en) 2004-02-05

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