ATE378421T1 - Glycosyltransferase inhibitoren - Google Patents

Glycosyltransferase inhibitoren

Info

Publication number
ATE378421T1
ATE378421T1 AT00936281T AT00936281T ATE378421T1 AT E378421 T1 ATE378421 T1 AT E378421T1 AT 00936281 T AT00936281 T AT 00936281T AT 00936281 T AT00936281 T AT 00936281T AT E378421 T1 ATE378421 T1 AT E378421T1
Authority
AT
Austria
Prior art keywords
inhibitors
glycosyltransferase
glycosyltransferase inhibitors
glyscosyltranferase
glycosyltransferases
Prior art date
Application number
AT00936281T
Other languages
English (en)
Inventor
Shawn Defrees
Original Assignee
Abaron Biosciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abaron Biosciences Inc filed Critical Abaron Biosciences Inc
Application granted granted Critical
Publication of ATE378421T1 publication Critical patent/ATE378421T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • A61K31/405Indole-alkanecarboxylic acids; Derivatives thereof, e.g. tryptophan, indomethacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT00936281T 1999-05-24 2000-05-24 Glycosyltransferase inhibitoren ATE378421T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13615099P 1999-05-24 1999-05-24
US57712099A 1999-05-24 1999-05-24

Publications (1)

Publication Number Publication Date
ATE378421T1 true ATE378421T1 (de) 2007-11-15

Family

ID=26834046

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00936281T ATE378421T1 (de) 1999-05-24 2000-05-24 Glycosyltransferase inhibitoren

Country Status (4)

Country Link
EP (1) EP1185269B1 (de)
AT (1) ATE378421T1 (de)
DE (1) DE60037113T2 (de)
WO (1) WO2001068095A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0421368D0 (en) * 2004-09-25 2004-10-27 Univ York Glycosyltransferase assay
EP2720044A1 (de) * 2012-10-15 2014-04-16 National University of Ireland, Galway Sialyltransferase ST3GAL6 als Marker für multiples Myelom
JP2016530265A (ja) 2013-08-12 2016-09-29 ベナロヤ リサーチ インスティテュート アット バージニア メイソン 免疫調節のための4−メチルウンベリフェロン処置
CN111437283A (zh) * 2020-03-09 2020-07-24 吉林大学 β1,4-半乳糖基转移酶抑制剂在制备治疗癌症的药物中的应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0576592B1 (de) * 1991-03-18 2000-05-31 The Scripps Research Institute Oligosaccharide als enzymsubstrate und -inhibitoren: verfahren und zusammensetzungen
CZ120398A3 (cs) * 1995-09-08 1998-12-16 Novo Nordisk A/S Použití 2-alkylpyrrolidinových derivátů pro přípravu léčiva pro léčbu diabetu, 2-alkylpyrrolidiné deriváty
US5770407A (en) * 1996-12-10 1998-06-23 The Scripps Research Institute Process for preparing nucleotide inhibitors of glycosyltransferases

Also Published As

Publication number Publication date
WO2001068095A1 (en) 2001-09-20
DE60037113T2 (de) 2008-09-18
EP1185269A1 (de) 2002-03-13
EP1185269B1 (de) 2007-11-14
DE60037113D1 (de) 2007-12-27
EP1185269A4 (de) 2004-12-01

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Legal Events

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