ATE386742T1 - Imidazonaphthyridine - Google Patents

Imidazonaphthyridine

Info

Publication number
ATE386742T1
ATE386742T1 AT99953956T AT99953956T ATE386742T1 AT E386742 T1 ATE386742 T1 AT E386742T1 AT 99953956 T AT99953956 T AT 99953956T AT 99953956 T AT99953956 T AT 99953956T AT E386742 T1 ATE386742 T1 AT E386742T1
Authority
AT
Austria
Prior art keywords
imidazonaphthyridines
tetrahydropyrido
substituents
prevention
compounds
Prior art date
Application number
AT99953956T
Other languages
English (en)
Inventor
Gerhard Grundler
Stefan Postius
Wolfgang-Alexander Simon
Wolfgang Kromer
Joerg Senn-Bilfinger
Original Assignee
Nycomed Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nycomed Gmbh filed Critical Nycomed Gmbh
Application granted granted Critical
Publication of ATE386742T1 publication Critical patent/ATE386742T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Luminescent Compositions (AREA)
AT99953956T 1998-11-03 1999-10-29 Imidazonaphthyridine ATE386742T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP98120834 1998-11-03

Publications (1)

Publication Number Publication Date
ATE386742T1 true ATE386742T1 (de) 2008-03-15

Family

ID=8232910

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99953956T ATE386742T1 (de) 1998-11-03 1999-10-29 Imidazonaphthyridine

Country Status (8)

Country Link
US (1) US6384048B1 (de)
EP (1) EP1127059B1 (de)
JP (1) JP2002528548A (de)
AT (1) ATE386742T1 (de)
AU (1) AU1044500A (de)
CA (1) CA2349476A1 (de)
DE (1) DE69938192D1 (de)
WO (1) WO2000026217A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2003528878A (ja) * 2000-03-29 2003-09-30 アルタナ ファルマ アクチエンゲゼルシャフト イミダゾピリジン誘導体のプロドラッグ
AU2002210563B2 (en) 2000-10-25 2007-03-01 Altana Pharma Ag Polysubstituted imidazopyridines as gastric secretion inhibitors
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
ATE336493T1 (de) 2001-08-02 2006-09-15 Altana Pharma Ag Tricyclische epoxide
US20040235882A1 (en) * 2001-08-03 2004-11-25 Jorg Senn-Bilfinger Amino-substituted imidazopyridines for the treatment of gastrointestial diseases
HRP20040834A2 (en) * 2002-02-15 2005-06-30 Altana Pharma Ag Tricyclic n-acyl compounds
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
TWI295575B (en) * 2002-04-24 2008-04-11 Altana Pharma Ag Nitrosated imidazopyridines
HRP20050528A2 (en) 2002-11-19 2006-06-30 Altana Pharma Ag 8-substituted imidazopyridines
BRPI0407541A (pt) * 2003-02-17 2006-02-14 Altana Pharma Ag combinações e uso de compostos farmaceuticamente ativos selecionados
EA009985B1 (ru) 2003-03-10 2008-04-28 Никомед Гмбх Новый способ получения рофлумиласта
CA2526566A1 (en) * 2003-05-27 2004-12-09 Altana Pharma Ag Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
EP1682133A1 (de) 2003-11-03 2006-07-26 AstraZeneca AB Imidazo-1,2-a-pyridin-derivate zur behandlung von beschwerdefreiem gastroösophagealem reflux
WO2005058894A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
WO2005089317A2 (en) * 2004-03-15 2005-09-29 3M Innovative Properties Company Immune response modifier formulations and methods
JP2008501766A (ja) * 2004-06-09 2008-01-24 ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング 置換された三環式のベンゾイミダゾール
AU2005291284A1 (en) * 2004-10-01 2006-04-13 Altana Pharma Ag Substituted tricyclic benzimidazoles
ES2421916T3 (es) * 2005-03-16 2013-09-06 Nycomed Gmbh Forma farmacéutica de sabor enmascarado que contiene roflumilast
EP2452680B1 (de) 2009-07-09 2019-12-18 RaQualia Pharma Inc. Säurepumpenantagonist zur behandlung von mit unnormalen magen-darm-bewegungen assoziierten erkrankungen

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
US4755524A (en) * 1986-01-31 1988-07-05 G. D. Searle & Co. Novel phenolic thioethers as inhibitors of 5-lipoxygenase
JPH07113924B2 (ja) 1986-02-14 1995-12-06 インターナショナル・ビジネス・マシーンズ・コーポレーション データ・ベース検索システム
BR9807883A (pt) * 1997-03-24 2000-02-22 Byk Gulden Lomberg Chem Fab Compostos de tetraidropirido
CA2289542A1 (en) 1997-05-28 1998-12-03 Byk Gulden Lomberg Chemische Fabrik Gmbh Fused dihydropyrans
HUP0001555A3 (en) 1997-10-30 2001-01-29 Altana Pharma Ag Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation

Also Published As

Publication number Publication date
AU1044500A (en) 2000-05-22
WO2000026217A1 (en) 2000-05-11
DE69938192D1 (en) 2008-04-03
CA2349476A1 (en) 2000-05-11
EP1127059B1 (de) 2008-02-20
US6384048B1 (en) 2002-05-07
JP2002528548A (ja) 2002-09-03
EP1127059A1 (de) 2001-08-29

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties