ATE386742T1 - Imidazonaphthyridine - Google Patents

Imidazonaphthyridine

Info

Publication number
ATE386742T1
ATE386742T1 AT99953956T AT99953956T ATE386742T1 AT E386742 T1 ATE386742 T1 AT E386742T1 AT 99953956 T AT99953956 T AT 99953956T AT 99953956 T AT99953956 T AT 99953956T AT E386742 T1 ATE386742 T1 AT E386742T1
Authority
AT
Austria
Prior art keywords
imidazonaphthyridines
tetrahydropyrido
substituents
prevention
compounds
Prior art date
Application number
AT99953956T
Other languages
English (en)
Inventor
Gerhard Grundler
Stefan Postius
Wolfgang-Alexander Simon
Wolfgang Kromer
Joerg Senn-Bilfinger
Original Assignee
Nycomed Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nycomed Gmbh filed Critical Nycomed Gmbh
Application granted granted Critical
Publication of ATE386742T1 publication Critical patent/ATE386742T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Luminescent Compositions (AREA)
AT99953956T 1998-11-03 1999-10-29 Imidazonaphthyridine ATE386742T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP98120834 1998-11-03

Publications (1)

Publication Number Publication Date
ATE386742T1 true ATE386742T1 (de) 2008-03-15

Family

ID=8232910

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99953956T ATE386742T1 (de) 1998-11-03 1999-10-29 Imidazonaphthyridine

Country Status (8)

Country Link
US (1) US6384048B1 (de)
EP (1) EP1127059B1 (de)
JP (1) JP2002528548A (de)
AT (1) ATE386742T1 (de)
AU (1) AU1044500A (de)
CA (1) CA2349476A1 (de)
DE (1) DE69938192D1 (de)
WO (1) WO2000026217A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK286850B6 (sk) * 2000-03-29 2009-06-05 Altana Pharma Ag Prekurzory imidazopyridínových derivátov, farmaceutický prostriedok s ich obsahom a ich použitie
EA008151B1 (ru) * 2000-10-25 2007-04-27 Алтана Фарма Аг Полизамещенные имидазопиридины в качестве ингибиторов желудочной секреции
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
HUP0400379A3 (en) 2001-08-02 2007-10-29 Altana Pharma Ag Tricyclic epoxides and their use for the preparation of pharmaceutically active agents
US20040235882A1 (en) * 2001-08-03 2004-11-25 Jorg Senn-Bilfinger Amino-substituted imidazopyridines for the treatment of gastrointestial diseases
US7314935B2 (en) * 2002-02-15 2008-01-01 Altana Pharma Ag Tricyclic n-acyl compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
TWI295575B (en) * 2002-04-24 2008-04-11 Altana Pharma Ag Nitrosated imidazopyridines
AU2003288071A1 (en) 2002-11-19 2004-06-15 Altana Pharma Ag 8-substituted imidazopyridines
MXPA05008490A (es) * 2003-02-17 2005-10-18 Altana Pharma Ag Combinaciones que contienen imidazopiridinas y su uso en el tratamiento de enfermedades gastrointestinales inflamatorias.
ES2335498T3 (es) 2003-03-10 2010-03-29 Nycomed Gmbh Nuevo proceso para la preparacion de reflumilast.
WO2004105795A1 (en) * 2003-05-27 2004-12-09 Altana Pharma Ag Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
KR20060099524A (ko) 2003-11-03 2006-09-19 아스트라제네카 아베 무증상 위식도 역류의 치료를 위한 이미다조[1,2-a]피리딘유도체
WO2005058894A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
CA2559607C (en) * 2004-03-15 2013-02-19 3M Innovative Properties Company Immune response modifier formulations and methods
AU2005251943A1 (en) * 2004-06-09 2005-12-22 Altana Pharma Ag Substituted tricyclic benzimidazoles
CA2582256A1 (en) * 2004-10-01 2006-04-13 Altana Pharma Ag Substituted tricyclic benzimidazoles
US8663694B2 (en) * 2005-03-16 2014-03-04 Takeda Gmbh Taste masked dosage form containing roflumilast
KR101605063B1 (ko) 2009-07-09 2016-03-21 라퀄리아 파마 인코포레이티드 소화관 운동이상이 관여하는 질환의 치료용 산 펌프 길항제

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
US4755524A (en) * 1986-01-31 1988-07-05 G. D. Searle & Co. Novel phenolic thioethers as inhibitors of 5-lipoxygenase
JPH07113924B2 (ja) 1986-02-14 1995-12-06 インターナショナル・ビジネス・マシーンズ・コーポレーション データ・ベース検索システム
EP0971922B1 (de) * 1997-03-24 2004-04-28 ALTANA Pharma AG Tetrahydropyridoverbindungen
EA002402B1 (ru) * 1997-03-24 2002-04-25 Бык Гульден Ломберг Хемише Фабрик Гмбх Тетрагидропиридо-соединения
JP2001526703A (ja) 1997-05-28 2001-12-18 ビイク グルデン ロンベルク ヒエーミツシエ フアブリーク ゲゼルシヤフト ミツト ベシユレンクテル ハフツング 縮合ジヒドロピラン

Also Published As

Publication number Publication date
DE69938192D1 (en) 2008-04-03
CA2349476A1 (en) 2000-05-11
AU1044500A (en) 2000-05-22
US6384048B1 (en) 2002-05-07
WO2000026217A1 (en) 2000-05-11
EP1127059A1 (de) 2001-08-29
EP1127059B1 (de) 2008-02-20
JP2002528548A (ja) 2002-09-03

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Legal Events

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