ATE386742T1 - Imidazonaphthyridine - Google Patents

Imidazonaphthyridine

Info

Publication number
ATE386742T1
ATE386742T1 AT99953956T AT99953956T ATE386742T1 AT E386742 T1 ATE386742 T1 AT E386742T1 AT 99953956 T AT99953956 T AT 99953956T AT 99953956 T AT99953956 T AT 99953956T AT E386742 T1 ATE386742 T1 AT E386742T1
Authority
AT
Austria
Prior art keywords
imidazonaphthyridines
tetrahydropyrido
substituents
prevention
compounds
Prior art date
Application number
AT99953956T
Other languages
English (en)
Inventor
Gerhard Grundler
Stefan Postius
Wolfgang-Alexander Simon
Wolfgang Kromer
Joerg Senn-Bilfinger
Original Assignee
Nycomed Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nycomed Gmbh filed Critical Nycomed Gmbh
Application granted granted Critical
Publication of ATE386742T1 publication Critical patent/ATE386742T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Luminescent Compositions (AREA)
AT99953956T 1998-11-03 1999-10-29 Imidazonaphthyridine ATE386742T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP98120834 1998-11-03

Publications (1)

Publication Number Publication Date
ATE386742T1 true ATE386742T1 (de) 2008-03-15

Family

ID=8232910

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99953956T ATE386742T1 (de) 1998-11-03 1999-10-29 Imidazonaphthyridine

Country Status (8)

Country Link
US (1) US6384048B1 (de)
EP (1) EP1127059B1 (de)
JP (1) JP2002528548A (de)
AT (1) ATE386742T1 (de)
AU (1) AU1044500A (de)
CA (1) CA2349476A1 (de)
DE (1) DE69938192D1 (de)
WO (1) WO2000026217A1 (de)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100860627B1 (ko) * 2000-03-29 2008-09-29 니코메드 게엠베하 이미다조피리딘 유도체의 프로드러그
KR20040011423A (ko) * 2000-10-25 2004-02-05 알타나 파마 아게 위액 분비 억제제로서의 다중치환된 이미다조피리딘
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
WO2003014119A1 (en) 2001-08-02 2003-02-20 Altana Pharma Ag Tricyclic epoxides
WO2003014120A1 (en) * 2001-08-03 2003-02-20 Altana Pharma Ag Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases
US7314935B2 (en) * 2002-02-15 2008-01-01 Altana Pharma Ag Tricyclic n-acyl compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
TWI295575B (en) * 2002-04-24 2008-04-11 Altana Pharma Ag Nitrosated imidazopyridines
KR20050086584A (ko) 2002-11-19 2005-08-30 알타나 파마 아게 8-치환 이미다조피리딘
PL377581A1 (pl) * 2003-02-17 2006-02-06 Altana Pharma Ag Połączenia zawierające imidazopirydyny oraz ich zastosowanie do leczenia chorób zapalnych przewodu pokarmowego
DK1606261T3 (da) 2003-03-10 2010-01-18 Nycomed Gmbh Hidtil ukendt fremgangsmåde til fremstilling af roflumilast
US20060241134A1 (en) * 2003-05-27 2006-10-26 Altana Pharma Ga Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
WO2005041961A1 (en) 2003-11-03 2005-05-12 Astrazeneca Ab Imidazo [1,2-a] pyridine derivatives for the treatment of silent gastro-esophageal reflux
US7326784B2 (en) 2003-12-19 2008-02-05 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano-imidazo-pyridines derivatives
ES2665342T3 (es) * 2004-03-15 2018-04-25 Meda Ab Formulaciones y métodos para modificadores de la respuesta inmune
WO2005121139A1 (en) * 2004-06-09 2005-12-22 Altana Pharma Ag Substituted tricyclic benzimidazoles
CA2582256A1 (en) * 2004-10-01 2006-04-13 Altana Pharma Ag Substituted tricyclic benzimidazoles
AU2006224619B2 (en) * 2005-03-16 2012-06-07 Takeda Gmbh Taste masked dosage form containing roflumilast
US8648080B2 (en) 2009-07-09 2014-02-11 Raqualia Pharma Inc. Acid pump antagonist for the treatment of diseases involved in abnormal gastrointestinal motility

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4468400A (en) 1982-12-20 1984-08-28 Schering Corporation Antiulcer tricyclic imidazo [1,2-a]pyridines
US4755524A (en) * 1986-01-31 1988-07-05 G. D. Searle & Co. Novel phenolic thioethers as inhibitors of 5-lipoxygenase
JPH07113924B2 (ja) 1986-02-14 1995-12-06 インターナショナル・ビジネス・マシーンズ・コーポレーション データ・ベース検索システム
IL131407A0 (en) * 1997-03-24 2001-01-28 Byk Gulden Lomberg Chem Fab Tetrahydropyrido compounds medicaments containing the same and the use thereof
AU736767B2 (en) 1997-05-28 2001-08-02 Altana Pharma Ag Fused dihydropyrans
HUP0001555A3 (en) 1997-10-30 2001-01-29 Altana Pharma Ag Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation

Also Published As

Publication number Publication date
US6384048B1 (en) 2002-05-07
AU1044500A (en) 2000-05-22
CA2349476A1 (en) 2000-05-11
EP1127059B1 (de) 2008-02-20
JP2002528548A (ja) 2002-09-03
EP1127059A1 (de) 2001-08-29
DE69938192D1 (en) 2008-04-03
WO2000026217A1 (en) 2000-05-11

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties