ATE311389T1 - Wirkstoffvorläufer von imidazopyridin-derivaten - Google Patents

Wirkstoffvorläufer von imidazopyridin-derivaten

Info

Publication number: ATE311389T1
Authority: AT; Austria
Prior art keywords: precursor; imidazopyridine derivatives; imidazopyridine; derivatives; substituents
Prior art date: 2000-03-29

Application number

AT01933769T

Other languages

English (en)

Inventor

Wolfgang-Alexander Simon

Stefan Postius

Reinhard Huber

Wolfgang Kromer

Joerg Senn-Bilfinger

Wilm Buhr

Original Assignee

Altana Pharma Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-29

Filing date

2001-03-28

Publication date

2005-12-15

2001-03-28 Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag

2005-12-15 Application granted granted Critical

2005-12-15 Publication of ATE311389T1 publication Critical patent/ATE311389T1/de

Links

150000005232 imidazopyridines Chemical class 0.000 title 1
239000002243 precursor Substances 0.000 title 1
208000018522 Gastrointestinal disease Diseases 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AT01933769T 2000-03-29 2001-03-28 Wirkstoffvorläufer von imidazopyridin-derivaten ATE311389T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00106695		2000-03-29
PCT/EP2001/003514 WO2001072756A1 (en)	2000-03-29	2001-03-28	Prodrugs of imidazopyridine derivatives

Publications (1)

Publication Number	Publication Date
ATE311389T1 true ATE311389T1 (de)	2005-12-15

Family

ID=8168271

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01933769T ATE311389T1 (de)	2000-03-29	2001-03-28	Wirkstoffvorläufer von imidazopyridin-derivaten

Country Status (25)

Country	Link
US (2)	US20030125327A1 (de)
EP (1)	EP1313740B1 (de)
JP (1)	JP2003528878A (de)
KR (1)	KR100860627B1 (de)
CN (1)	CN1214030C (de)
AT (1)	ATE311389T1 (de)
AU (1)	AU783633B2 (de)
BR (1)	BR0109483A (de)
CA (1)	CA2404474A1 (de)
CZ (1)	CZ20023194A3 (de)
DE (1)	DE60115466T2 (de)
DK (1)	DK1313740T3 (de)
EA (1)	EA005597B1 (de)
ES (1)	ES2253376T3 (de)
HR (1)	HRP20020854A2 (de)
HU (1)	HUP0302331A2 (de)
IL (2)	IL151200A0 (de)
MX (1)	MXPA02009551A (de)
NO (1)	NO20024662L (de)
NZ (1)	NZ520837A (de)
PL (1)	PL365116A1 (de)
SI (1)	SI1313740T1 (de)
SK (1)	SK286850B6 (de)
WO (1)	WO2001072756A1 (de)
ZA (1)	ZA200207637B (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ20023116A3 (cs) *	2000-03-29	2003-01-15	Altana Pharma Ag	Alkylované imidazopyridinové sloučeniny
AU2002210563B2 (en)	2000-10-25	2007-03-01	Altana Pharma Ag	Polysubstituted imidazopyridines as gastric secretion inhibitors
WO2003043614A2 (en) *	2001-11-19	2003-05-30	Altana Pharma Ag	Reversible proton pump inhibitors for the treatment of airway disorders
HRP20040834A2 (en)	2002-02-15	2005-06-30	Altana Pharma Ag	Tricyclic n-acyl compounds
TWI295575B (en) *	2002-04-24	2008-04-11	Altana Pharma Ag	Nitrosated imidazopyridines
WO2003094967A2 (en) *	2002-05-07	2003-11-20	Altana Pharma Ag	New combination of reversible proton pump inhibitors and airway therapeutics for treating airway disorders
HRP20050528A2 (en)	2002-11-19	2006-06-30	Altana Pharma Ag	8-substituted imidazopyridines
PL375933A1 (en) *	2002-12-20	2005-12-12	Altana Pharma Ag	8-trialkylsiloxy-2-methyl-9-phenyl-7-oxo-7,8,9,10-tetrahydroimidazo[1,2-h][1,7]naphthyridines
BRPI0407541A (pt) *	2003-02-17	2006-02-14	Altana Pharma Ag	combinações e uso de compostos farmaceuticamente ativos selecionados
AR044129A1 (es)	2003-05-06	2005-08-24	Altana Pharma Ag	Compuestos intermedios de imidazopiridina. proceso de preparacion.
SA04250092B1 (ar) *	2003-05-14	2008-05-04	التانا فاروا ايه جي	مركب وسيط جديد لتحضير مركبات إيميدازوبيريدين imidazopyridines فعالة علاجياً
CA2526566A1 (en) *	2003-05-27	2004-12-09	Altana Pharma Ag	Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility
EP1682133A1 (de)	2003-11-03	2006-07-26	AstraZeneca AB	Imidazo-1,2-a-pyridin-derivate zur behandlung von beschwerdefreiem gastroösophagealem reflux
AR046893A1 (es) *	2003-12-16	2005-12-28	Altana Pharma Ag	Bencimidazoles triciclicos
WO2005058894A1 (en)	2003-12-19	2005-06-30	Altana Pharma Ag	Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
CN101027277A (zh) *	2004-07-23	2007-08-29	帝斯曼知识产权资产管理有限公司	(2r,3r)－2－羟基－3－氨基－3－芳基－丙酰胺和(2r,3r)－2－羟基－3－氨基－3－芳基－丙酸烷基酯的制备方法
AU2005291284A1 (en) *	2004-10-01	2006-04-13	Altana Pharma Ag	Substituted tricyclic benzimidazoles
EP2452680B1 (de)	2009-07-09	2019-12-18	RaQualia Pharma Inc.	Säurepumpenantagonist zur behandlung von mit unnormalen magen-darm-bewegungen assoziierten erkrankungen

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4468400A (en) *	1982-12-20	1984-08-28	Schering Corporation	Antiulcer tricyclic imidazo [1,2-a]pyridines
US4673679A (en) *	1986-05-14	1987-06-16	E. I. Du Pont De Nemours And Company	Use of prodrugs of 3-hydroxymorphinans to prevent bitter taste upon buccal, nasal or sublingual administration
JPH06502659A (ja) *	1991-05-31	1994-03-24	ファイザー　インク	免疫抑制剤としてのラパマイシンプロドラッグの使用
DE4308095A1 (de) *	1993-03-13	1994-09-15	Hoechst Ag	Prodrug-Derivate von Arzneimittelwirkstoffen mit Hydroxylgruppen, Verfahren zu deren Herstellung und ihre Verwendung
SE9401197D0 (sv) *	1994-04-11	1994-04-11	Astra Ab	Active compounds
US6073004A (en)	1996-12-17	2000-06-06	Ericsson Inc.	Emergency call initiator
BR9807883A (pt) *	1997-03-24	2000-02-22	Byk Gulden Lomberg Chem Fab	Compostos de tetraidropirido
CA2289542A1 (en) *	1997-05-28	1998-12-03	Byk Gulden Lomberg Chemische Fabrik Gmbh	Fused dihydropyrans
HUP0001555A3 (en) *	1997-10-30	2001-01-29	Altana Pharma Ag	Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation
WO2000017200A1 (en) *	1998-09-23	2000-03-30	Byk Gulden Lomberg Chemische Fabrik Gmbh	Tetrahydropyridoethers
CA2349476A1 (en) *	1998-11-03	2000-05-11	Byk Gulden Lomberg Chemische Fabrik Gmbh	Imidazonaphthyridines
CZ20023116A3 (cs) *	2000-03-29	2003-01-15	Altana Pharma Ag	Alkylované imidazopyridinové sloučeniny

2001
- 2001-03-28 JP JP2001570665A patent/JP2003528878A/ja not_active Withdrawn
- 2001-03-28 DK DK01933769T patent/DK1313740T3/da active
- 2001-03-28 HR HRP20020854 patent/HRP20020854A2/hr not_active Application Discontinuation
- 2001-03-28 WO PCT/EP2001/003514 patent/WO2001072756A1/en not_active Ceased
- 2001-03-28 SI SI200130498T patent/SI1313740T1/sl unknown
- 2001-03-28 CZ CZ20023194A patent/CZ20023194A3/cs unknown
- 2001-03-28 CA CA002404474A patent/CA2404474A1/en not_active Abandoned
- 2001-03-28 US US10/182,619 patent/US20030125327A1/en not_active Abandoned
- 2001-03-28 HU HU0302331A patent/HUP0302331A2/hu unknown
- 2001-03-28 EA EA200200875A patent/EA005597B1/ru not_active IP Right Cessation
- 2001-03-28 EP EP01933769A patent/EP1313740B1/de not_active Expired - Lifetime
- 2001-03-28 MX MXPA02009551A patent/MXPA02009551A/es active IP Right Grant
- 2001-03-28 KR KR1020027012842A patent/KR100860627B1/ko not_active Expired - Fee Related
- 2001-03-28 IL IL15120001A patent/IL151200A0/xx unknown
- 2001-03-28 PL PL01365116A patent/PL365116A1/xx not_active Application Discontinuation
- 2001-03-28 AU AU60166/01A patent/AU783633B2/en not_active Ceased
- 2001-03-28 SK SK1385-2002A patent/SK286850B6/sk not_active IP Right Cessation
- 2001-03-28 ES ES01933769T patent/ES2253376T3/es not_active Expired - Lifetime
- 2001-03-28 NZ NZ520837A patent/NZ520837A/en unknown
- 2001-03-28 BR BR0109483-1A patent/BR0109483A/pt not_active Application Discontinuation
- 2001-03-28 CN CNB018071635A patent/CN1214030C/zh not_active Expired - Fee Related
- 2001-03-28 DE DE60115466T patent/DE60115466T2/de not_active Expired - Fee Related
- 2001-03-28 AT AT01933769T patent/ATE311389T1/de not_active IP Right Cessation
2002
- 2002-08-12 IL IL151200A patent/IL151200A/en not_active IP Right Cessation
- 2002-09-23 ZA ZA200207637A patent/ZA200207637B/en unknown
- 2002-09-27 NO NO20024662A patent/NO20024662L/no not_active Application Discontinuation
2004
- 2004-04-19 US US10/826,337 patent/US7189736B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
ZA200207637B (en)	2004-04-08
DE60115466D1 (de)	2006-01-05
AU783633B2 (en)	2005-11-17
AU6016601A (en)	2001-10-08
NO20024662D0 (no)	2002-09-27
HK1056175A1 (en)	2004-02-06
KR100860627B1 (ko)	2008-09-29
HRP20020854A2 (en)	2004-12-31
BR0109483A (pt)	2003-06-10
US20030125327A1 (en)	2003-07-03
SK13852002A3 (sk)	2003-02-04
NO20024662L (no)	2002-09-27
CN1214030C (zh)	2005-08-10
WO2001072756A1 (en)	2001-10-04
US20040198764A1 (en)	2004-10-07
HUP0302331A2 (hu)	2003-12-29
DE60115466T2 (de)	2006-07-20
CN1426414A (zh)	2003-06-25
KR20020084262A (ko)	2002-11-04
US7189736B2 (en)	2007-03-13
EP1313740A1 (de)	2003-05-28
NZ520837A (en)	2005-01-28
ES2253376T3 (es)	2006-06-01
IL151200A0 (en)	2003-04-10
EA200200875A1 (ru)	2003-04-24
JP2003528878A (ja)	2003-09-30
DK1313740T3 (da)	2006-04-03
SI1313740T1 (sl)	2006-04-30
CA2404474A1 (en)	2001-10-04
MXPA02009551A (es)	2004-05-14
PL365116A1 (en)	2004-12-27
EA005597B1 (ru)	2005-04-28
IL151200A (en)	2009-11-18
SK286850B6 (sk)	2009-06-05
EP1313740B1 (de)	2005-11-30
CZ20023194A3 (cs)	2003-01-15

Legal Events

Date

Code

Title

Description

2006-07-15

UEP

Publication of translation of european patent specification

Ref document number: 1313740

Country of ref document: EP

2010-12-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
YU21401A (sh)	2004-03-12	Tetrahidropiridoetri
ATE332302T1 (de)	2006-07-15	Alkylierte imidazopyridinderivate
DE60115466D1 (de)	2006-01-05	Wirkstoffvorläufer von imidazopyridin-derivaten
ATE386742T1 (de)	2008-03-15	Imidazonaphthyridine
ATE265455T1 (de)	2004-05-15	Tetrahydropyridoverbindungen
DE60127131D1 (de)	2007-04-19	Tricyclische imidazopyridine
DE60131968D1 (de)	2008-01-31	PYRANOÄ2,3-cÜIMIDAZOÄ1,2-aÜPYRIDIN-DERIVATE ZUR BEHANDLUNG VON GASTROINTESTINALEN ERKRANKUNGEN
ATE328883T1 (de)	2006-06-15	Imidazopyridin-8-one
IS8034A (is)	2005-09-16	Imídasó[4,5-B]kínólínafleiður og notkun þeirra sem NO-myndunarhemla
EA200500903A1 (ru)	2005-12-29	Силиловые простые эфиры
PE61999A1 (es)	1999-06-19	Compuestos de tetrahidropiridina