ATE387430T1 - Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffe - Google Patents
Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffeInfo
- Publication number
- ATE387430T1 ATE387430T1 AT00986516T AT00986516T ATE387430T1 AT E387430 T1 ATE387430 T1 AT E387430T1 AT 00986516 T AT00986516 T AT 00986516T AT 00986516 T AT00986516 T AT 00986516T AT E387430 T1 ATE387430 T1 AT E387430T1
- Authority
- AT
- Austria
- Prior art keywords
- compositions
- compounds
- active ingredients
- delivering active
- delivering
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000004480 active ingredient Substances 0.000 title 1
- 239000013543 active substance Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C235/58—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C235/60—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C235/58—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring
- C07C235/64—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring with carbon atoms of carboxamide groups and singly-bound oxygen atoms, bound in ortho-position to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
- C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
- C07C235/84—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
- C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton
- C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17121399P | 1999-12-16 | 1999-12-16 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE387430T1 true ATE387430T1 (de) | 2008-03-15 |
Family
ID=22622945
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00986516T ATE387430T1 (de) | 1999-12-16 | 2000-12-18 | Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffe |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US6693208B2 (de) |
| EP (1) | EP1237872B1 (de) |
| JP (1) | JP4850379B2 (de) |
| AT (1) | ATE387430T1 (de) |
| AU (1) | AU2274201A (de) |
| DE (1) | DE60038183T2 (de) |
| ES (1) | ES2298168T3 (de) |
| WO (1) | WO2001044199A1 (de) |
Families Citing this family (47)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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| AU2595697A (en) * | 1996-03-29 | 1997-10-22 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| US6991798B1 (en) | 1998-08-07 | 2006-01-31 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| IL140930A0 (en) * | 1998-08-07 | 2002-02-10 | Emisphere Tech Inc | Compounds and compositions for delivering active agents |
| EP1237872B1 (de) * | 1999-12-16 | 2008-02-27 | Emisphere Technologies, Inc. | Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffe |
| US7151191B2 (en) | 2000-01-13 | 2006-12-19 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| UA80248C2 (en) | 2000-06-29 | 2007-09-10 | Compounds and compositions for delivering active agents | |
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| WO2002069937A1 (en) * | 2001-03-01 | 2002-09-12 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| NZ527157A (en) * | 2001-03-01 | 2005-04-29 | Emisphere Tech Inc | Compositions for delivering bisphosphonates |
| JP5196701B2 (ja) * | 2001-11-29 | 2013-05-15 | エミスフィアー テクノロジーズ インコーポレイテッド | クロモリンナトリウムの経口投与用製剤 |
| CN1332711C (zh) | 2002-02-20 | 2007-08-22 | 埃米球科技有限公司 | 施用glp－1分子的方法 |
| US8088734B2 (en) | 2003-01-21 | 2012-01-03 | Unigene Laboratories Inc. | Oral delivery of peptides |
| US7288253B2 (en) | 2003-08-08 | 2007-10-30 | Amgen Fremont, Inc. | Antibodies directed to parathyroid hormone (PTH) and uses thereof |
| US7318925B2 (en) | 2003-08-08 | 2008-01-15 | Amgen Fremont, Inc. | Methods of use for antibodies against parathyroid hormone |
| CN100398536C (zh) | 2003-08-20 | 2008-07-02 | 爱密斯菲尔科技公司 | 用于口服传递glp-1化合物或mc4激动剂肽的化合物、方法和制剂 |
| JP4767850B2 (ja) | 2003-08-20 | 2011-09-07 | エミスフィアー テクノロジーズ インコーポレイテッド | グルカゴン様ペプチド（ｇｌｐ）−１化合物またはメラノコルチン４受容体（ｍｃ４）アゴニストペプチドの経口デリバリーのための化合物、方法および製剤 |
| US20060286129A1 (en) | 2003-12-19 | 2006-12-21 | Emisphere Technologies, Inc. | Oral GLP-1 formulations |
| JP2005209106A (ja) * | 2004-01-26 | 2005-08-04 | Nec Corp | 携帯通信端末、受信メール管理方法、プログラムおよび記録媒体 |
| BRPI0510226A (pt) * | 2004-05-06 | 2007-10-23 | Emisphere Tech Inc | composição farmacêutica sólida, forma de dosagem sólida, método para administrar heparina a um animal, método para tratar ou evitar trombose em um animal, método para preparar uma forma de dosagem sólida de heparina umidecida |
| CA2566161C (en) | 2004-05-14 | 2013-10-01 | Emisphere Technologies, Inc. | Aryl ketone compounds and compositions for delivering active agents |
| WO2005112633A2 (en) | 2004-05-14 | 2005-12-01 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| RU2403237C2 (ru) * | 2004-05-14 | 2010-11-10 | Эмисфире Текнолоджис, Инк. | Составы и смеси для доставки активных агентов |
| AU2005244986B2 (en) | 2004-05-19 | 2011-01-27 | Emisphere Technologies, Inc. | Topical cromolyn formulations |
| US20080132527A1 (en) | 2004-05-19 | 2008-06-05 | Emisphere Technologies, Inc. | Compositions For Delivering Acyclovir |
| CA2573856A1 (en) | 2004-08-03 | 2006-02-16 | Emisphere Technologies, Inc. | Antidiabetic oral insulin-biguanide combination |
| US7659289B2 (en) * | 2004-09-17 | 2010-02-09 | Comentis, Inc. | Hydroxyethylene-based β-secretase inhibitors and use thereof |
| WO2006034277A1 (en) * | 2004-09-17 | 2006-03-30 | Comentis, Inc. | Bicyclic compounds which inhibit beta-secretase activity and methods of use thereof |
| US9345725B2 (en) * | 2004-12-29 | 2016-05-24 | Emisphere Technologies, Inc. | Pharmaceutical formulations of gallium salts |
| US8110547B2 (en) | 2005-01-12 | 2012-02-07 | Emisphere Technologies, Inc. | Compositions for buccal delivery of parathyroid hormone |
| NZ562314A (en) * | 2005-04-08 | 2010-02-26 | Comentis Inc | Compounds which inhibit beta-secretase activity and methods of use thereof |
| US8975227B2 (en) | 2005-07-15 | 2015-03-10 | Emisphere Technologies, Inc. | Intraoral dosage forms of glucagon |
| US8927015B2 (en) | 2006-04-12 | 2015-01-06 | Emisphere Technologies, Inc. | Formulations for delivering insulin |
| US8771712B2 (en) | 2006-05-09 | 2014-07-08 | Emisphere Technologies, Inc. | Topical administration of acyclovir |
| CA2656019C (en) | 2006-06-28 | 2016-09-13 | Emisphere Technologies, Inc. | Gallium nitrate formulations |
| WO2008027958A2 (en) | 2006-08-31 | 2008-03-06 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
| WO2008112706A1 (en) | 2007-03-13 | 2008-09-18 | Nutrition 21, Inc. | Methods and compositions for the sustained release of chromium |
| WO2009002867A2 (en) | 2007-06-26 | 2008-12-31 | Nutrition 21, Inc. | Multiple unit dosage form having a therapeutic agents in combination with a nutritional supplement |
| KR20100051668A (ko) * | 2007-07-26 | 2010-05-17 | 코멘티스, 인코포레이티드 | 베타-세크레타제 활성을 억제하는 이소프탈아미드 유도체 |
| CA2699787A1 (en) * | 2007-09-24 | 2009-04-02 | Comentis, Inc. | (3-hydroxy-4-amino-butan-2-yl)-3-(2-thiazol-2-yl-pyrrolidine-1-carbonyl) benzamide derivatives and related compounds as beta-secretase inhibitors for treating |
| EP2461803B1 (de) | 2009-08-03 | 2018-10-17 | Emisphere Technologies, Inc. | Schnell wirkende naproxenzusammensetzung mit reduzierter wirkung auf magen und darm |
| US20130150323A1 (en) * | 2010-02-04 | 2013-06-13 | Urigen Pharmaceuticals, Inc | Use of oral heparin preparations to treat urinary tract diseases and conditions |
| ES2927800T3 (es) | 2011-03-01 | 2022-11-11 | Nutrition 21 Llc | Composición de insulina y cromo para el tratamiento y la prevención de diabetes, hipoglicemia y trastornos relacionados |
| PT2897620T (pt) | 2012-09-21 | 2020-09-03 | Intensity Therapeutics Inc | Método de tratamento de cancro |
| GB2564295A (en) | 2016-02-11 | 2019-01-09 | Nutrition 21 Llc | Chromium containing compositions for improving health and fitness |
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| JP2002534363A (ja) * | 1999-01-08 | 2002-10-15 | エミスフェアー・テクノロジーズ・インク | ポリマー性デリバリー剤及びデリバリー剤化合物 |
| EP1237872B1 (de) * | 1999-12-16 | 2008-02-27 | Emisphere Technologies, Inc. | Verbindungen und zusammensetzungen zur abgabe aktiver wirkstoffe |
-
2000
- 2000-12-18 EP EP00986516A patent/EP1237872B1/de not_active Expired - Lifetime
- 2000-12-18 AU AU22742/01A patent/AU2274201A/en not_active Abandoned
- 2000-12-18 US US10/168,275 patent/US6693208B2/en not_active Expired - Lifetime
- 2000-12-18 AT AT00986516T patent/ATE387430T1/de not_active IP Right Cessation
- 2000-12-18 DE DE60038183T patent/DE60038183T2/de not_active Expired - Lifetime
- 2000-12-18 JP JP2001544689A patent/JP4850379B2/ja not_active Expired - Fee Related
- 2000-12-18 ES ES00986516T patent/ES2298168T3/es not_active Expired - Lifetime
- 2000-12-18 WO PCT/US2000/034329 patent/WO2001044199A1/en not_active Ceased
-
2003
- 2003-12-31 US US10/750,138 patent/US20050042274A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP4850379B2 (ja) | 2012-01-11 |
| US6693208B2 (en) | 2004-02-17 |
| EP1237872A1 (de) | 2002-09-11 |
| US20030216589A1 (en) | 2003-11-20 |
| WO2001044199A1 (en) | 2001-06-21 |
| EP1237872B1 (de) | 2008-02-27 |
| AU2274201A (en) | 2001-06-25 |
| DE60038183T2 (de) | 2009-02-19 |
| EP1237872A4 (de) | 2005-06-15 |
| ES2298168T3 (es) | 2008-05-16 |
| JP2003516971A (ja) | 2003-05-20 |
| DE60038183D1 (de) | 2008-04-10 |
| US20050042274A1 (en) | 2005-02-24 |
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