ATE414083T1 - Ocaperidonsalze und pharmazeutische zusammensetzungen, die diese enthalten - Google Patents

Ocaperidonsalze und pharmazeutische zusammensetzungen, die diese enthalten

Info

Publication number
ATE414083T1
ATE414083T1 AT06710597T AT06710597T ATE414083T1 AT E414083 T1 ATE414083 T1 AT E414083T1 AT 06710597 T AT06710597 T AT 06710597T AT 06710597 T AT06710597 T AT 06710597T AT E414083 T1 ATE414083 T1 AT E414083T1
Authority
AT
Austria
Prior art keywords
pharmaceutical compositions
ocaperidone
salt
compositions containing
containing same
Prior art date
Application number
AT06710597T
Other languages
English (en)
Inventor
Stefano Biondi
Arnold Demailly
Cesare Mondadori
Jean-Laurent Paparin
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE414083T1 publication Critical patent/ATE414083T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT06710597T 2005-02-24 2006-02-24 Ocaperidonsalze und pharmazeutische zusammensetzungen, die diese enthalten ATE414083T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05290428A EP1695973A1 (de) 2005-02-24 2005-02-24 Ocaperidonsalz und dieser enthaltende pharmazeutische Zubereitung

Publications (1)

Publication Number Publication Date
ATE414083T1 true ATE414083T1 (de) 2008-11-15

Family

ID=35431923

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06710597T ATE414083T1 (de) 2005-02-24 2006-02-24 Ocaperidonsalze und pharmazeutische zusammensetzungen, die diese enthalten

Country Status (15)

Country Link
US (1) US20080200479A1 (de)
EP (2) EP1695973A1 (de)
JP (1) JP2008531544A (de)
KR (1) KR20070105354A (de)
CN (1) CN101142214B (de)
AT (1) ATE414083T1 (de)
AU (1) AU2006217540C1 (de)
BR (1) BRPI0608560A2 (de)
CA (1) CA2598327A1 (de)
DE (1) DE602006003652D1 (de)
EA (1) EA012039B1 (de)
ES (1) ES2317507T3 (de)
MX (1) MX2007010245A (de)
NZ (1) NZ556748A (de)
WO (1) WO2006090285A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8227430B2 (en) * 2007-09-04 2012-07-24 Meiji Seika Pharma Co., Ltd Injectable, injection solution, and injection kit preparation
KR101501253B1 (ko) * 2014-12-22 2015-03-12 제이투에이치바이오텍 (주) 결정성 페북소스타트 피돌레이트 염 및 이의 제조 방법
KR101829706B1 (ko) 2016-09-21 2018-02-19 씨제이헬스케어 주식회사 벤즈이미다졸 유도체의 산부가염

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU65921A1 (de) * 1972-08-18 1974-02-21
US4575509A (en) * 1983-01-31 1986-03-11 Bristol-Myers Company Water-soluble formulations of m-AMSA with pyroglutamic acid
US5034397A (en) * 1985-12-12 1991-07-23 Bristol-Myers Squibb Co. Stable, water soluble salt compositions of M-AMSA in 1-methyl-2-pyrrolidinone
GB9008850D0 (en) * 1990-04-19 1990-06-13 Janssen Pharmaceutica Nv Novel 2,9-disubstituted-4h-pyridol(1,2-a)pyrimidin-4-ones
TW376319B (en) * 1993-04-28 1999-12-11 Janssen Pharmaceutica Nv Pharmaceutical composition containing risperidone pamoate and having a long acting activity for treating psychoses induced by the release of dopamine
US20030191141A1 (en) * 2002-03-28 2003-10-09 Inigo Pfeiffer Polymorphic form of 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-alpha]pyrimidin-4-one and formulations thereof
KR100467669B1 (ko) * 2002-08-21 2005-01-24 씨제이 주식회사 암로디핀의 유기산염
EP1543023B1 (de) * 2002-09-18 2010-03-17 Prosidion Limited Sekundäre bindungsstelle von dipeptidylpeptidase iv (dp iv)
US20040127733A1 (en) * 2002-10-31 2004-07-01 Boehringer Ingelheim Pharma Gmbh & Co. Kg New beta-agonists, processes for preparing them and their use as pharmaceutical compositions
EP1615924A1 (de) * 2003-04-22 2006-01-18 Synthon B.V. Wasserlöslich salze von risperidon
US20040254173A1 (en) * 2003-06-13 2004-12-16 Leventer Steven M. Modulation of dopamine responses with substituted (S)-2,3-benzodiazepines
TW200524864A (en) * 2003-11-10 2005-08-01 Wyeth Corp Sulfonyltetrahydro-3H-benzo(E)indole-8-amine compounds as 5-hydroxytryptamine-6 ligands
GEP20094781B (en) * 2004-01-22 2009-09-25 Pfizer Sulfonamide derivatives for the treatment of diseases
US7649002B2 (en) * 2004-02-04 2010-01-19 Pfizer Inc (3,5-dimethylpiperidin-1yl)(4-phenylpyrrolidin-3-yl)methanone derivatives as MCR4 agonists
AU2005243153A1 (en) * 2004-05-07 2005-11-24 Janssen Pharmaceutica N.V. Scalable synthesis of imidazole derivatives
UY29016A1 (es) * 2004-07-20 2006-02-24 Boehringer Ingelheim Int Analogos de dipeptidos inhibidores de la hepatitis c
US7329763B1 (en) * 2006-09-11 2008-02-12 New Cell Formulations Ltd Creatine pyroglutamic acid salts and methods for their production and use in individuals

Also Published As

Publication number Publication date
WO2006090285A1 (en) 2006-08-31
MX2007010245A (es) 2007-09-07
BRPI0608560A2 (pt) 2010-01-12
CN101142214B (zh) 2011-02-23
ES2317507T3 (es) 2009-04-16
DE602006003652D1 (de) 2008-12-24
US20080200479A1 (en) 2008-08-21
EP1888577A1 (de) 2008-02-20
EA200701797A1 (ru) 2008-02-28
AU2006217540C1 (en) 2011-11-03
JP2008531544A (ja) 2008-08-14
EP1888577B1 (de) 2008-11-12
AU2006217540A1 (en) 2006-08-31
AU2006217540B2 (en) 2011-05-12
EA012039B1 (ru) 2009-06-30
KR20070105354A (ko) 2007-10-30
CA2598327A1 (en) 2006-08-31
NZ556748A (en) 2009-08-28
EP1695973A1 (de) 2006-08-30
CN101142214A (zh) 2008-03-12

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