ATE449773T1 - Homomorpholinoxazolidinone als antibakterielle mittel - Google Patents

Homomorpholinoxazolidinone als antibakterielle mittel

Info

Publication number
ATE449773T1
ATE449773T1 AT06779767T AT06779767T ATE449773T1 AT E449773 T1 ATE449773 T1 AT E449773T1 AT 06779767 T AT06779767 T AT 06779767T AT 06779767 T AT06779767 T AT 06779767T AT E449773 T1 ATE449773 T1 AT E449773T1
Authority
AT
Austria
Prior art keywords
sup
sub
antibacterial agents
homomorpholinoxazolidinones
het
Prior art date
Application number
AT06779767T
Other languages
English (en)
Inventor
Vara Prasad Venkata Nagendra Josyula
Frederick Earl Boyer Jr
Ji-Young Kim
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Application granted granted Critical
Publication of ATE449773T1 publication Critical patent/ATE449773T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
AT06779767T 2005-06-29 2006-06-20 Homomorpholinoxazolidinone als antibakterielle mittel ATE449773T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69486205P 2005-06-29 2005-06-29
PCT/IB2006/001730 WO2007000644A1 (en) 2005-06-29 2006-06-20 Homomorpholine oxazolidinones as antibacterial agents

Publications (1)

Publication Number Publication Date
ATE449773T1 true ATE449773T1 (de) 2009-12-15

Family

ID=37101665

Family Applications (1)

Application Number Title Priority Date Filing Date
AT06779767T ATE449773T1 (de) 2005-06-29 2006-06-20 Homomorpholinoxazolidinone als antibakterielle mittel

Country Status (8)

Country Link
EP (1) EP1899331B1 (de)
JP (1) JP2008544979A (de)
AT (1) ATE449773T1 (de)
CA (1) CA2610978A1 (de)
DE (1) DE602006010702D1 (de)
DK (1) DK1899331T3 (de)
ES (1) ES2335307T3 (de)
WO (1) WO2007000644A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2181993A1 (de) 2006-03-31 2010-05-05 Research Foundation Itsuu Laboratory Antimikrobielle Oxazolidinonderivate
WO2009020616A1 (en) * 2007-08-06 2009-02-12 Micurx Pharmaceuticals, Inc. Antimicrobial ortho-fluorophenyl oxazolidinones for treatment of bacterial infections
CN101883768A (zh) * 2007-10-02 2010-11-10 财团法人乙卯研究所 具有7元杂环的噁唑烷酮衍生物
EP3107923B1 (de) 2014-02-21 2021-11-03 Shanghai MicuRx Pharmaceutical Co., Ltd. Wasserlösliche o-carbonyl-phosphoramidat-prodrugs zur therapeutischen verabreichung
WO2017015106A1 (en) * 2015-07-17 2017-01-26 The Global Alliance For Tb Drug Development, Inc. Substituted phenyloxazolidinones for antimicrobial therapy

Family Cites Families (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SK283420B6 (sk) 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
MY115155A (en) 1993-09-09 2003-04-30 Upjohn Co Substituted oxazine and thiazine oxazolidinone antimicrobials.
NZ295528A (en) 1994-11-15 1999-03-29 Upjohn Co Bicyclic oxazine and thiazine oxazolidinone antibacterials
CA2303959A1 (en) 1997-11-12 1999-05-20 Pharmacia & Upjohn Company Oxazolidinone derivatives and pharmaceutical compositions
JP2000204084A (ja) 1998-11-11 2000-07-25 Hokuriku Seiyaku Co Ltd チオカルバミド酸誘導体
EP1133493A1 (de) 1998-11-27 2001-09-19 PHARMACIA & UPJOHN COMPANY Thiocarbonylgruppe enthaltende oxazolidinone als antibakterielle mittel
US6297242B1 (en) 1999-08-12 2001-10-02 Ortho-Mcneil Pharmaceutical, Inc. N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof
HUP0203869A2 (hu) 1999-12-21 2003-07-28 Pharmacia & Upjohn Co. Szulfoximin funkcionalitással rendelkező oxazolidinok és alkalmazásuk mikrobaellenes szerként, a vegyületeket tartalmazó gyógyszerkészítmények
AU2001253113B2 (en) 2000-04-20 2005-02-03 Pharmacia & Upjohn Company Use of thioamide oxazolidinones for the treatment of bone resorption and osteoporosis
WO2002002095A2 (en) 2000-06-30 2002-01-10 Pharmacia & Upjohn Company Compositions for treating bacterial infections containing oxazolidinone compound, sulbactam and an ampicillin
GB0017225D0 (en) 2000-07-14 2000-08-30 Really Useful Products Limited Container
AU6937001A (en) 2000-07-17 2002-01-30 Ranbaxy Lab Ltd Oxazolidinone derivatives as antimicrobials
DE10034627A1 (de) 2000-07-17 2002-01-31 Bayer Ag Aryl-substituierte Oxazolidinone mit Cytokin inhibitorischer Wirkung
US6466161B2 (en) 2000-08-24 2002-10-15 Sirf Technology, Inc. Location services system that reduces auto-correlation or cross-correlation in weak signals
AR031135A1 (es) 2000-10-10 2003-09-10 Upjohn Co Composiciones de antibiotico topico para el tratamiento de infecciones oculares
MXPA03006958A (es) 2001-02-05 2003-11-18 Upjohn Co Composicion para administracion rectal de farmaco antibacterial de oxazolidinona.
DE10105989A1 (de) 2001-02-09 2002-08-14 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
GB0108793D0 (en) 2001-04-07 2001-05-30 Astrazeneca Ab Chemical compounds
US20050032861A1 (en) 2001-04-07 2005-02-10 Betts Michael John Oxazolidines containing a sulfonimid group as antibiotics
US6956040B2 (en) 2001-07-16 2005-10-18 Ranbaxy Laboratories Limited Oxazolidinone piperazinyl derivatives as potential antimicrobials
EP1409464A4 (de) 2001-07-16 2005-11-02 Ranbaxy Lab Ltd Oxazolidinonderivate als potentielle antimikrobielle mittel
TW200302095A (en) 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
WO2003072081A1 (en) 2002-02-22 2003-09-04 Pharmacia Corporation Ophthalmic formulation with gum system
MXPA04008173A (es) 2002-02-22 2004-11-26 Pharmacia Corp Formulaciones de farmaco antibiotico oftalmico que contienen un compuesto de ciclodextrina y cloruro de cetil piridinio.
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
RU2004129278A (ru) 2002-02-28 2005-06-10 Астразенека Аб (Se) Химические соединения
US7473699B2 (en) 2002-02-28 2009-01-06 Astrazeneca Ab 3-cyclyl-5-(nitrogen-containing 5-membered ring)methyl-oxazolidinone derivatives and their use as antibacterial agents
IL164195A0 (en) 2002-03-29 2005-12-18 Upjohn Co Parenteral, intravenous, and oral administration of oxazolidinones for treating diabetic foot infections
WO2003093247A2 (en) 2002-04-30 2003-11-13 Orchid Chemicals & Pharmaceuticals Ltd Antibacterial agents
TW200403240A (en) 2002-06-28 2004-03-01 Upjohn Co Difluorothioacetamides of oxazolidinones as antibacterial agents
WO2004009587A1 (en) 2002-07-22 2004-01-29 Orchid Chemicals & Pharmaceuticals Ltd Oxazolidinone derivatives as antibacterial agents
EA200500283A1 (ru) 2002-07-29 2005-08-25 Рэнбакси Лабораториз Лимитед Производные оксазолидинона как противомикробные средства
EP1578734A1 (de) 2002-08-22 2005-09-28 Orchid Chemicals and Pharmaceuticals Ltd Neue antibakterielle wirkstoffe

Also Published As

Publication number Publication date
JP2008544979A (ja) 2008-12-11
WO2007000644A1 (en) 2007-01-04
EP1899331B1 (de) 2009-11-25
DK1899331T3 (da) 2010-03-08
DE602006010702D1 (de) 2010-01-07
ES2335307T3 (es) 2010-03-24
CA2610978A1 (en) 2007-01-04
EP1899331A1 (de) 2008-03-19

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties