BR0215921A - Derivados de oxazolidinona utilizáveis como antimicrobianos e processo de sua preparação - Google Patents

Derivados de oxazolidinona utilizáveis como antimicrobianos e processo de sua preparação

Info

Publication number
BR0215921A
BR0215921A BR0215921-0A BR0215921A BR0215921A BR 0215921 A BR0215921 A BR 0215921A BR 0215921 A BR0215921 A BR 0215921A BR 0215921 A BR0215921 A BR 0215921A
Authority
BR
Brazil
Prior art keywords
antimicrobials
spp
oxazolidinone derivatives
mycobacterium
compounds
Prior art date
Application number
BR0215921-0A
Other languages
English (en)
Inventor
Anita Mehta
Sonali Rudra
Ajjarapu Venkata Subrahman Rao
Ajay Singh Yadav
Ashok Rattan
Original Assignee
Ranbaxy Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Lab Ltd filed Critical Ranbaxy Lab Ltd
Publication of BR0215921A publication Critical patent/BR0215921A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

"DERIVADOS DE OXAZOLIDINONA UTILIZáVEIS COMO ANTIMICROBIANOS E PROCESSO DE SUA PREPARAçãO". A presente invenção se refere a certas oxazolidinonas fenil substituídas e a processos para a síntese das mesmas. Esta invenção também se refere a composições farmacêuticas contendo os compostos da presente invenção como antimicrobianos. Os compostos são utilizáveis como agentes antimicrobianos, eficazes contra uma série de patógenos para indivíduos humanos e veterinários, incluindo bactérias aeróbias gram-positivas tais como estafilococos, estreptococos e enterococos bem como organismos anaeróbios tais como Bacterioides spp. e Clostridia spp., e organismos de produção ácida rápida, tais como Mycobacterium tuberculosis, Mycobacterium avium e Mycobacterium spp.
BR0215921-0A 2002-07-29 2002-07-29 Derivados de oxazolidinona utilizáveis como antimicrobianos e processo de sua preparação BR0215921A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IB2002/002940 WO2004014392A1 (en) 2002-07-29 2002-07-29 Oxazolidinone derivatives as antimicrobials

Publications (1)

Publication Number Publication Date
BR0215921A true BR0215921A (pt) 2005-09-13

Family

ID=31503894

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0215921-0A BR0215921A (pt) 2002-07-29 2002-07-29 Derivados de oxazolidinona utilizáveis como antimicrobianos e processo de sua preparação

Country Status (8)

Country Link
US (1) US20060293307A1 (pt)
EP (1) EP1542696A4 (pt)
CN (1) CN1668308A (pt)
AU (1) AU2002319848A1 (pt)
BR (1) BR0215921A (pt)
EA (1) EA200500283A1 (pt)
MX (1) MXPA05001199A (pt)
WO (1) WO2004014392A1 (pt)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL371335A1 (en) 2002-01-22 2005-06-13 Pharmacia & Upjohn Company Infection-resistant medical devices
US6875784B2 (en) * 2002-10-09 2005-04-05 Pharmacia & Upjohn Company Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
WO2005082899A1 (en) * 2004-01-28 2005-09-09 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
WO2006043121A1 (en) * 2004-10-20 2006-04-27 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
WO2006051408A1 (en) * 2004-11-11 2006-05-18 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
EP1874782A1 (en) 2005-04-15 2008-01-09 Ranbaxy Laboratories Limited Oxazolidinone derivatives as antimicrobials
WO2007023507A2 (en) * 2005-06-20 2007-03-01 Wockhardt Limited Oxazolidinones bearing antimicrobial activity composition and methods of preparation
WO2007000644A1 (en) 2005-06-29 2007-01-04 Pharmacia & Upjohn Company Llc Homomorpholine oxazolidinones as antibacterial agents
JP2009523764A (ja) * 2006-01-19 2009-06-25 ラボラトリオス・サルバト・ソシエダッド・アノニマ 抗菌活性を有するジカルボニル化合物
KR20080110877A (ko) 2006-03-31 2008-12-19 재단법인 이쯔우 연구소 헤테로환을 갖는 신규 화합물
WO2009044777A1 (ja) 2007-10-02 2009-04-09 Research Foundation Itsuu Laboratory ７員ヘテロ環を有するオキサゾリジノン誘導体
EP2367820B1 (en) 2008-11-20 2016-09-21 Panacea Biotec Limited Novel antimicrobial agents
BR112012000657A2 (pt) 2009-06-26 2016-11-16 Panacea Biotec Ltd novos azabicilohexanos
WO2013044845A1 (zh) * 2011-09-29 2013-04-04 山东轩竹医药科技有限公司 联芳基杂环取代的噁唑烷酮抗菌药
CN104364240B (zh) * 2012-06-08 2017-02-22 四川贝力克生物技术有限责任公司 一种用于预防或治疗分支杆菌疾病的药物
WO2014180562A1 (en) 2013-05-07 2014-11-13 Galapagos Nv Novel compounds and pharmaceutical compositions thereof for the treatment of cystic fibrosis
PT3030568T (pt) 2013-08-08 2018-12-24 Galapagos Nv Tieno[2,3-c]piranos como moduladores de cftr
WO2020113094A1 (en) 2018-11-30 2020-06-04 Nuvation Bio Inc. Pyrrole and pyrazole compounds and methods of use thereof
WO2021258013A1 (en) 2020-06-18 2021-12-23 Akagera Medicines, Inc. Oxazolidinone compounds, liposome compositions comprising oxazolidinone compounds and methods of use thereof

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH23565A (en) * 1986-09-05 1989-08-25 Sumitomo Chemical Co Novel pyrimidinylpyrimidine derivatives and a plant disease protectant containing them as the active ingredient
CA1288433C (en) * 1986-12-03 1991-09-03 Tsuguhiro Katoh Pyridinylpyrimidine derivatives, method for production thereof and a fungicide containing them as the active ingredient
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4921869A (en) * 1987-10-09 1990-05-01 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
ZA969622B (en) * 1995-12-13 1998-05-15 Upjohn Co Oxazolidinone antibacterial agents having a six-membered heteroaromatic ring.
MY116093A (en) * 1996-02-26 2003-11-28 Upjohn Co Azolyl piperazinyl phenyl oxazolidinone antimicrobials
CN1138765C (zh) * 1997-05-30 2004-02-18 法玛西雅厄普约翰美国公司 带有硫代羰基功能基的噁唑烷酮抗菌剂
BR0112826A (pt) * 2000-07-17 2003-06-24 Ranbaxy Lab Ltd Derivados da oxazolidinona como antimicrobianos

Also Published As

Publication number Publication date
AU2002319848A1 (en) 2004-02-25
EP1542696A1 (en) 2005-06-22
US20060293307A1 (en) 2006-12-28
EA200500283A1 (ru) 2005-08-25
WO2004014392A1 (en) 2004-02-19
EP1542696A4 (en) 2006-08-02
CN1668308A (zh) 2005-09-14
MXPA05001199A (es) 2005-05-16

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Legal Events

Date Code Title Description
B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE A 3O, 5O, 6O E 7O ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2038 DE 26/01/2010