ATE493423T1 - Verfahren zur steuerung der kristallstruktur von risedronat - Google Patents
Verfahren zur steuerung der kristallstruktur von risedronatInfo
- Publication number
- ATE493423T1 ATE493423T1 AT04778281T AT04778281T ATE493423T1 AT E493423 T1 ATE493423 T1 AT E493423T1 AT 04778281 T AT04778281 T AT 04778281T AT 04778281 T AT04778281 T AT 04778281T AT E493423 T1 ATE493423 T1 AT E493423T1
- Authority
- AT
- Austria
- Prior art keywords
- risedronate
- controlling
- crystal structure
- hydrate
- ethylidene
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- IIDJRNMFWXDHID-UHFFFAOYSA-N Risedronic acid Chemical compound OP(=O)(O)C(P(O)(O)=O)(O)CC1=CC=CN=C1 IIDJRNMFWXDHID-UHFFFAOYSA-N 0.000 title abstract 2
- 229940089617 risedronate Drugs 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 239000013078 crystal Substances 0.000 abstract 1
- 230000006911 nucleation Effects 0.000 abstract 1
- 238000010899 nucleation Methods 0.000 abstract 1
- 238000010979 pH adjustment Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/58—Pyridine rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Glass Compositions (AREA)
- Crystals, And After-Treatments Of Crystals (AREA)
- Steroid Compounds (AREA)
- Pyridine Compounds (AREA)
- Seasonings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Yarns And Mechanical Finishing Of Yarns Or Ropes (AREA)
- Pens And Brushes (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49122203P | 2003-07-30 | 2003-07-30 | |
| PCT/US2004/022703 WO2005012314A1 (en) | 2003-07-30 | 2004-07-15 | Process for controlling crystal structure of risedronate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE493423T1 true ATE493423T1 (de) | 2011-01-15 |
Family
ID=34115482
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT04778281T ATE493423T1 (de) | 2003-07-30 | 2004-07-15 | Verfahren zur steuerung der kristallstruktur von risedronat |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US7002014B2 (de) |
| EP (1) | EP1651656B1 (de) |
| JP (1) | JP4423614B2 (de) |
| KR (1) | KR100786044B1 (de) |
| CN (1) | CN100439377C (de) |
| AT (1) | ATE493423T1 (de) |
| AU (1) | AU2004261561B9 (de) |
| BR (1) | BRPI0413067A (de) |
| CA (1) | CA2529470C (de) |
| CO (1) | CO5660304A2 (de) |
| DE (1) | DE602004030801D1 (de) |
| IL (1) | IL172676A (de) |
| IS (1) | IS2915B (de) |
| MA (1) | MA27914A1 (de) |
| MX (1) | MXPA06001129A (de) |
| NO (1) | NO335393B1 (de) |
| NZ (1) | NZ544030A (de) |
| RU (1) | RU2319706C2 (de) |
| SG (1) | SG144151A1 (de) |
| WO (1) | WO2005012314A1 (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1775302A1 (de) | 2005-10-11 | 2007-04-18 | Sandoz A/S | Methode zur Herstellung von kristallinem Natriumrisedronat |
| JP5052816B2 (ja) * | 2006-04-26 | 2012-10-17 | 株式会社パーマケム・アジア | ３−ピリジル−１−ヒドロキシエチリデン−１、１−ビスホスホン酸ナトリウム塩２．５水和物ａ型結晶の製造方法 |
| JP5354858B2 (ja) * | 2006-05-09 | 2013-11-27 | 株式会社Ａｄｅｋａ | スルホンアミド化合物の金属塩を含有するポリエステル樹脂組成物 |
| JP2009536639A (ja) | 2006-05-11 | 2009-10-15 | アイエヌディー−スイフト ラボラトリーズ リミテッド | 純リセドロン酸または塩を調製するための方法 |
| WO2008044245A2 (en) * | 2006-10-10 | 2008-04-17 | Matrix Laboratories Ltd | A process for the preparation of risedronate sodium hemipentahydrate |
| KR100828705B1 (ko) * | 2006-12-04 | 2008-05-09 | 씨제이제일제당 (주) | 리세드론산 나트륨 수화물의 제조방법 |
| KR100775440B1 (ko) | 2006-12-20 | 2007-11-12 | 동우신테크 주식회사 | 리세드로네이트 나트륨 헤미펜타히드레이트의 제조방법 |
| KR100798855B1 (ko) * | 2007-02-14 | 2008-01-28 | 주식회사 엔지켐 | 리세드론산 나트륨 헤미펜타하이드레이트의 제조방법 |
| KR100812528B1 (ko) * | 2007-04-12 | 2008-03-12 | 보령제약 주식회사 | 리세드로네이트 나트륨염의 헤미펜타히드레이트의 선택적결정화방법 |
| WO2009050731A2 (en) * | 2007-06-20 | 2009-04-23 | Alkem Laboratories Ltd | Novel process for preparing risedronic acid |
| WO2009034580A1 (en) * | 2007-09-11 | 2009-03-19 | Fleming Laboratories Limited | Improved process for the preparation of risedronate sodium hemipentahydrate |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3428524A1 (de) * | 1984-08-02 | 1986-02-13 | Boehringer Mannheim Gmbh, 6800 Mannheim | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
| IL77243A (en) * | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
| RU2120798C1 (ru) * | 1991-11-22 | 1998-10-27 | Проктер энд Гэмбл Фармасьютикалз, Инк. | Твердая фармацевтическая композиция для перорального введения |
| PE20011061A1 (es) * | 2000-02-01 | 2001-11-20 | Procter & Gamble | Cristalizacion selectiva del acido 3-piridil-1-hidroxi-etiliden-1,1-bisfosfonico sodio como el hemipentahidrato o el monohidrato |
-
2004
- 2004-07-15 BR BRPI0413067-7A patent/BRPI0413067A/pt not_active Application Discontinuation
- 2004-07-15 EP EP04778281A patent/EP1651656B1/de not_active Expired - Lifetime
- 2004-07-15 MX MXPA06001129A patent/MXPA06001129A/es active IP Right Grant
- 2004-07-15 AU AU2004261561A patent/AU2004261561B9/en not_active Expired
- 2004-07-15 DE DE602004030801T patent/DE602004030801D1/de not_active Expired - Lifetime
- 2004-07-15 JP JP2006521878A patent/JP4423614B2/ja not_active Expired - Lifetime
- 2004-07-15 CN CNB2004800205190A patent/CN100439377C/zh not_active Expired - Lifetime
- 2004-07-15 NZ NZ544030A patent/NZ544030A/en not_active IP Right Cessation
- 2004-07-15 RU RU2006102357/04A patent/RU2319706C2/ru active
- 2004-07-15 SG SG200804444-8A patent/SG144151A1/en unknown
- 2004-07-15 CA CA2529470A patent/CA2529470C/en not_active Expired - Lifetime
- 2004-07-15 KR KR1020067000683A patent/KR100786044B1/ko not_active Expired - Lifetime
- 2004-07-15 AT AT04778281T patent/ATE493423T1/de not_active IP Right Cessation
- 2004-07-15 WO PCT/US2004/022703 patent/WO2005012314A1/en not_active Ceased
- 2004-07-29 US US10/901,692 patent/US7002014B2/en not_active Expired - Lifetime
-
2005
- 2005-12-18 IL IL172676A patent/IL172676A/en active IP Right Grant
-
2006
- 2006-01-25 IS IS8262A patent/IS2915B/is unknown
- 2006-01-26 MA MA28754A patent/MA27914A1/fr unknown
- 2006-02-27 CO CO06019211A patent/CO5660304A2/es not_active Application Discontinuation
- 2006-02-27 NO NO20060950A patent/NO335393B1/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN100439377C (zh) | 2008-12-03 |
| RU2006102357A (ru) | 2006-07-27 |
| MXPA06001129A (es) | 2006-04-11 |
| KR20060054297A (ko) | 2006-05-22 |
| AU2004261561A1 (en) | 2005-02-10 |
| IS8262A (is) | 2006-01-25 |
| JP4423614B2 (ja) | 2010-03-03 |
| NZ544030A (en) | 2008-05-30 |
| CA2529470C (en) | 2010-11-23 |
| CO5660304A2 (es) | 2006-07-31 |
| EP1651656B1 (de) | 2010-12-29 |
| CN1823078A (zh) | 2006-08-23 |
| IS2915B (is) | 2014-12-15 |
| SG144151A1 (en) | 2008-07-29 |
| RU2319706C2 (ru) | 2008-03-20 |
| JP2007500189A (ja) | 2007-01-11 |
| WO2005012314A1 (en) | 2005-02-10 |
| IL172676A (en) | 2010-12-30 |
| US7002014B2 (en) | 2006-02-21 |
| NO20060950L (no) | 2006-02-27 |
| DE602004030801D1 (de) | 2011-02-10 |
| IL172676A0 (en) | 2006-04-10 |
| AU2004261561B9 (en) | 2008-10-30 |
| BRPI0413067A (pt) | 2006-10-17 |
| KR100786044B1 (ko) | 2007-12-17 |
| US20050026869A1 (en) | 2005-02-03 |
| EP1651656A1 (de) | 2006-05-03 |
| MA27914A1 (fr) | 2006-05-02 |
| CA2529470A1 (en) | 2005-02-10 |
| NO335393B1 (no) | 2014-12-08 |
| AU2004261561B2 (en) | 2008-06-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |