ATE497499T1 - Verfahren zur herstellung von hexahydrofuroä2,3- büfuran-3-ol - Google Patents

Verfahren zur herstellung von hexahydrofuroä2,3- büfuran-3-ol

Info

Publication number: ATE497499T1
Authority: AT; Austria
Prior art keywords: bufuran; producing; hexahydrofuro; furan; methods
Prior art date: 2006-11-09

Application number

AT07822416T

Other languages

English (en)

Inventor

Sebastien Francois Emmanuel Lemaire

Andras Horvath

Wim Albert Alex Aelterman

Thomas Joachim Landewald Rammeloo

Original Assignee

Tibotec Pharm Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-11-09

Filing date

2007-11-09

Publication date

2011-02-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37692659&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE497499(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-11-09 Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd

2011-02-15 Application granted granted Critical

2011-02-15 Publication of ATE497499T1 publication Critical patent/ATE497499T1/de

Links

238000004519 manufacturing process Methods 0.000 title 1
RCDXYCHYMULCDZ-HCWXCVPCSA-N (3as,4r,6ar)-2,3,3a,4,5,6a-hexahydrofuro[2,3-b]furan-4-ol Chemical compound O1CC[C@H]2[C@@H](O)CO[C@H]21 RCDXYCHYMULCDZ-HCWXCVPCSA-N 0.000 abstract 1
RCDXYCHYMULCDZ-UHFFFAOYSA-N 2,3,3a,4,5,6a-hexahydrofuro[2,3-b]furan-4-ol Chemical compound O1CCC2C(O)COC21 RCDXYCHYMULCDZ-UHFFFAOYSA-N 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/20—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Furan Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

AT07822416T 2006-11-09 2007-11-09 Verfahren zur herstellung von hexahydrofuroä2,3- büfuran-3-ol ATE497499T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP06123752		2006-11-09
PCT/EP2007/062119 WO2008055970A2 (en)	2006-11-09	2007-11-09	Methods for the preparation of hexahydrofuro[2,3-b]furan-3-ol

Publications (1)

Publication Number	Publication Date
ATE497499T1 true ATE497499T1 (de)	2011-02-15

Family

ID=37692659

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT07822416T ATE497499T1 (de)	2006-11-09	2007-11-09	Verfahren zur herstellung von hexahydrofuroä2,3- büfuran-3-ol

Country Status (22)

Country	Link
US (1)	US8153829B2 (de)
EP (1)	EP2089371B1 (de)
JP (1)	JP5491862B2 (de)
CN (2)	CN101541775B (de)
AT (1)	ATE497499T1 (de)
AU (1)	AU2007316562B2 (de)
BR (1)	BRPI0718706B8 (de)
CA (1)	CA2669014C (de)
CY (1)	CY1111407T1 (de)
DE (1)	DE602007012365D1 (de)
DK (1)	DK2089371T3 (de)
ES (1)	ES2359949T3 (de)
HR (1)	HRP20110258T1 (de)
IL (1)	IL198270A (de)
ME (1)	ME01232B (de)
MX (1)	MX2009004957A (de)
PL (1)	PL2089371T3 (de)
PT (1)	PT2089371E (de)
RS (1)	RS51675B (de)
RU (1)	RU2464266C2 (de)
SI (1)	SI2089371T1 (de)
WO (1)	WO2008055970A2 (de)

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EP2571355B1 (de)	2010-05-20	2016-09-07	Hetero Research Foundation	Kristallines hydrochloridsalz von darunavir
CN102617586B (zh) *	2011-01-26	2016-04-06	浙江九洲药业股份有限公司	地瑞那韦中间体的制备方法
ES2755087T3 (es)	2012-08-22	2020-04-21	Merck Sharp & Dohme	Derivados de benzimidazol hexahidrofuro[3,2-b]furano útiles como activadores de proteína cinasa activada por AMP
CN103864813B (zh) *	2012-12-18	2017-02-22	上海迪赛诺化学制药有限公司	一种合成六氢呋喃并[2,3‑b]呋喃‑3‑醇及其对映体的方法
CN103896886A (zh) *	2012-12-31	2014-07-02	上海迪赛诺化学制药有限公司	一种达鲁那韦中间体及其制备方法和应用
TW201514188A (zh) *	2013-03-13	2015-04-16	Lantheus Medical Imaging Inc	製備釓磷維塞三鈉單水合物之方法
CN103664976B (zh) *	2013-12-12	2015-11-04	惠州市莱佛士制药技术有限公司	一种顺式六氢呋喃并[2,3-b]呋喃-3-醇的制备方法
CN113307783B (zh) *	2016-05-07	2023-04-07	成都博腾药业有限公司	一种制备地瑞那韦中间体的方法
CN112300186B (zh) *	2019-08-01	2024-04-30	浙江九洲药业股份有限公司	六氢呋喃并呋喃醇衍生物的制备方法、其中间体及其制备方法

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ES2338538T3 (es) *	2001-09-10	2010-05-10	Tibotec Pharmaceuticals	Metodo para la preparacion de hexahidrofuro(2,3-b)furan-3-ol.
WO2003024974A2 (en)	2001-09-20	2003-03-27	Smithkline Beecham Corporation	Process for preparing protease inhibitor intermediates
ES2503551T5 (es) *	2002-05-16	2021-10-28	Janssen Sciences Ireland Unlimited Co	Formas pseudopolimórficas de un inhibidor de la proteasa de VIH
DK1532127T3 (da) *	2002-06-27	2007-02-05	Smithkline Beecham Corp	Fremstilling af stereoisomerer af (3alfa,3alfa/beta,6alfa/beta)hexahydrofuro(2,3-b)furan-3-ol
WO2004033462A2 (en)	2002-10-09	2004-04-22	The Board Of Trustees Of The University Of Illinois	METHOD OF PREPARING (3R, 3aS, 6aR) -3- HYDROXYHEXAHYDROFURO [2, 3-b] FURAN AND RELATED COMPOUNDS
WO2004060895A1 (ja)	2002-12-27	2004-07-22	Sumitomo Chemical Company, Limited	ヘキサヒドロフロフラノール誘導体の製造方法、その中間体及びその製造方法
DE602004021640D1 (de) *	2003-12-23	2009-07-30	Tibotec Pharm Ltd	Verfahren zur herstellung von (1s,2r)-3-ää(4-aminophenyl)sulfonylü(isobutyl)aminoü-1-benzyl-2-hydroxypropylcarbamidsäure-(3r,3as,6ar)-hexahydrofuroä2,3-büfuran-3-ylester
TWI383975B (zh)	2004-03-31	2013-02-01	悌柏泰克醫藥有限公司	製備（３Ｒ，３ａＳ，６ａＲ）六氫-呋喃并〔２，３-ｂ〕呋喃-３-醇之方法

2007
- 2007-11-09 ES ES07822416T patent/ES2359949T3/es active Active
- 2007-11-09 DE DE602007012365T patent/DE602007012365D1/de active Active
- 2007-11-09 SI SI200730567T patent/SI2089371T1/sl unknown
- 2007-11-09 DK DK07822416.9T patent/DK2089371T3/da active
- 2007-11-09 PL PL07822416T patent/PL2089371T3/pl unknown
- 2007-11-09 CN CN2007800418345A patent/CN101541775B/zh active Active
- 2007-11-09 AT AT07822416T patent/ATE497499T1/de active
- 2007-11-09 PT PT07822416T patent/PT2089371E/pt unknown
- 2007-11-09 AU AU2007316562A patent/AU2007316562B2/en active Active
- 2007-11-09 BR BRPI0718706A patent/BRPI0718706B8/pt active IP Right Grant
- 2007-11-09 WO PCT/EP2007/062119 patent/WO2008055970A2/en not_active Ceased
- 2007-11-09 RS RS20110169A patent/RS51675B/sr unknown
- 2007-11-09 EP EP07822416A patent/EP2089371B1/de active Active
- 2007-11-09 JP JP2009535738A patent/JP5491862B2/ja active Active
- 2007-11-09 HR HR20110258T patent/HRP20110258T1/hr unknown
- 2007-11-09 RU RU2009121792/04A patent/RU2464266C2/ru active
- 2007-11-09 US US12/447,537 patent/US8153829B2/en active Active
- 2007-11-09 CN CN201110342987.1A patent/CN102432621B/zh active Active
- 2007-11-09 ME MEP-2011-65A patent/ME01232B/me unknown
- 2007-11-09 CA CA2669014A patent/CA2669014C/en active Active
- 2007-11-09 MX MX2009004957A patent/MX2009004957A/es active IP Right Grant
2009
- 2009-04-21 IL IL198270A patent/IL198270A/en active IP Right Grant
2011
- 2011-05-02 CY CY20111100423T patent/CY1111407T1/el unknown

Also Published As

Publication number	Publication date
JP5491862B2 (ja)	2014-05-14
ES2359949T3 (es)	2011-05-30
RU2009121792A (ru)	2010-12-20
CA2669014A1 (en)	2008-05-15
PL2089371T3 (pl)	2011-06-30
EP2089371A2 (de)	2009-08-19
EP2089371B1 (de)	2011-02-02
BRPI0718706B1 (pt)	2021-03-23
CA2669014C (en)	2016-01-26
AU2007316562A1 (en)	2008-05-15
ME01232B (me)	2013-06-20
CN101541775B (zh)	2011-12-28
US8153829B2 (en)	2012-04-10
CN102432621A (zh)	2012-05-02
BRPI0718706A2 (pt)	2014-01-07
WO2008055970A3 (en)	2008-06-26
AU2007316562B2 (en)	2013-02-21
HRP20110258T1 (hr)	2011-05-31
JP2010509290A (ja)	2010-03-25
SI2089371T1 (sl)	2011-05-31
DK2089371T3 (da)	2011-05-16
CN101541775A (zh)	2009-09-23
WO2008055970A2 (en)	2008-05-15
BRPI0718706B8 (pt)	2021-05-25
RS51675B (sr)	2011-10-31
PT2089371E (pt)	2011-04-18
CY1111407T1 (el)	2015-08-05
IL198270A (en)	2014-02-27
RU2464266C2 (ru)	2012-10-20
IL198270A0 (en)	2009-12-24
DE602007012365D1 (de)	2011-03-17
US20100094028A1 (en)	2010-04-15
MX2009004957A (es)	2009-05-19
CN102432621B (zh)	2016-02-17

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2011-08-15

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