ATE502914T1 - Therapeutische amide und entsprechende verbindungen - Google Patents

Therapeutische amide und entsprechende verbindungen

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Publication number
ATE502914T1
ATE502914T1 AT07840723T AT07840723T ATE502914T1 AT E502914 T1 ATE502914 T1 AT E502914T1 AT 07840723 T AT07840723 T AT 07840723T AT 07840723 T AT07840723 T AT 07840723T AT E502914 T1 ATE502914 T1 AT E502914T1
Authority
AT
Austria
Prior art keywords
corresponding compounds
therapeutic
amides
therapeutic amides
disclosed
Prior art date
Application number
AT07840723T
Other languages
English (en)
Inventor
David Old
Danny Dinh
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Application granted granted Critical
Publication of ATE502914T1 publication Critical patent/ATE502914T1/de

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    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/52—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
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    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

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US7985767B2 (en) * 2006-09-06 2011-07-26 Allergan, Inc. Therapeutic amides
US7956051B2 (en) * 2008-01-24 2011-06-07 Allergan, Inc. Therapeutic amides and related compounds
US8198318B2 (en) 2008-03-18 2012-06-12 Allergen, Inc. Therapeutic amides
CN104341367B (zh) * 2014-10-07 2016-08-17 张远强 一类四氮唑乙酸类化合物、其制备方法及用途
CN104262276B (zh) * 2014-10-07 2016-06-22 张远强 含卤代苯的四氮唑乙酸类化合物、其制备方法及用途
CN104262277B (zh) * 2014-10-07 2016-06-22 张远强 含硝基和卤苯取代的四氮唑乙酸类化合物、其制备方法及用途
CN104292176B (zh) * 2014-10-07 2016-06-29 张远强 一种含卤代苯的四氮唑乙酸类化合物、其制备方法和用途
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CN104292178B (zh) * 2014-10-07 2016-06-22 张远强 含四氮唑乙酸类化合物、其制备方法及用途
CN104292177B (zh) * 2014-10-07 2016-08-17 张远强 含腈基和卤苯取代的四氮唑乙酸类化合物、其制备方法及用途

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US6437146B1 (en) * 1998-09-25 2002-08-20 Fujisawa Pharmaceutical Co., Ltd. Oxazole compounds as prostaglandin e2 agonists or antagonists
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ES2254726T3 (es) * 2001-07-16 2006-06-16 F. Hoffmann-La Roche Ag Analogos de prostaglandina como agonistas receptores de ep4.
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ES2246419T3 (es) * 2001-11-05 2006-02-16 Allergan, Inc. Analogos de omega-cicloalquil-17-heteroaril-prostaglandina e2 como agonistas del receptor ep-2.
CA2372731A1 (en) * 2002-02-22 2003-08-22 Claudiu T. Supuran Oligo-amine/oligo-carboxy sulfonamides
US6573294B1 (en) * 2002-05-14 2003-06-03 Allergan, Inc. 8-azaprostaglandin analogs as agents for lowering intraocular pressure
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AU2007284085A1 (en) 2008-02-21
BRPI0716643A2 (pt) 2017-05-16
EP2049467A2 (de) 2009-04-22
US20080051374A1 (en) 2008-02-28
WO2008021804A3 (en) 2008-04-10
EP2049467B1 (de) 2011-03-23
WO2008021804A2 (en) 2008-02-21
JP2010500976A (ja) 2010-01-14
ES2361131T3 (es) 2011-06-14
US7468360B2 (en) 2008-12-23
CA2660396A1 (en) 2008-02-21

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