ATE50578T1 - Imidazo(1,2-a>chinolinderivate, ihre herstellung und therapeutische anwendung. - Google Patents

Imidazo(1,2-a>chinolinderivate, ihre herstellung und therapeutische anwendung.

Info

Publication number
ATE50578T1
ATE50578T1 AT87400073T AT87400073T ATE50578T1 AT E50578 T1 ATE50578 T1 AT E50578T1 AT 87400073 T AT87400073 T AT 87400073T AT 87400073 T AT87400073 T AT 87400073T AT E50578 T1 ATE50578 T1 AT E50578T1
Authority
AT
Austria
Prior art keywords
see diagramm
compound
formula
alkylamino
alpha
Prior art date
Application number
AT87400073T
Other languages
English (en)
Inventor
Pascal George
Peretti Daniele De
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Application granted granted Critical
Publication of ATE50578T1 publication Critical patent/ATE50578T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Optical Fibers, Optical Fiber Cores, And Optical Fiber Bundles (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
AT87400073T 1986-01-22 1987-01-14 Imidazo(1,2-a>chinolinderivate, ihre herstellung und therapeutische anwendung. ATE50578T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8600834A FR2593179B1 (fr) 1986-01-22 1986-01-22 Derives d'imidazo(1,2-a)quinoleines, leur preparation et leur application en therapeutique
EP87400073A EP0233800B1 (de) 1986-01-22 1987-01-14 Imidazo[1,2-a]chinolinderivate, ihre Herstellung und therapeutische Anwendung

Publications (1)

Publication Number Publication Date
ATE50578T1 true ATE50578T1 (de) 1990-03-15

Family

ID=9331353

Family Applications (1)

Application Number Title Priority Date Filing Date
AT87400073T ATE50578T1 (de) 1986-01-22 1987-01-14 Imidazo(1,2-a>chinolinderivate, ihre herstellung und therapeutische anwendung.

Country Status (18)

Country Link
EP (1) EP0233800B1 (de)
JP (1) JPS62169783A (de)
AT (1) ATE50578T1 (de)
AU (1) AU585688B2 (de)
CA (1) CA1286668C (de)
DE (1) DE3761770D1 (de)
DK (1) DK31887A (de)
ES (1) ES2014306B3 (de)
FI (1) FI85476C (de)
FR (1) FR2593179B1 (de)
GR (1) GR3000463T3 (de)
HU (1) HU194232B (de)
IE (1) IE59173B1 (de)
IL (1) IL81335A (de)
NO (1) NO164596C (de)
NZ (1) NZ219008A (de)
PT (1) PT84159B (de)
ZA (1) ZA87442B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2593180B1 (fr) * 1986-01-22 1990-10-26 Synthelabo Derives d'acylaminomethyl-1 imidazo (1,2-a)quinoleines, leur preparation et leur application en therapeutique
US5935970A (en) * 1995-06-15 1999-08-10 Pharmacia & Upjohn Company Use of imidazo 1,5-a!quinolones as neuroprotective agents
FR2759700B1 (fr) * 1997-02-20 1999-03-19 Synthelabo Derives d'imidazo [2,1-c][1,4] benzothiazine, leur preparation et leur application en therapeutique
FR2783828B1 (fr) * 1998-09-29 2000-11-10 Synthelabo Derives d'acide 5,6-dihydro-4h-imidazo[1,2-a][1] benzazepine -1-acetique, leur preparation et leur application en therapeutique
WO2004058758A1 (en) * 2002-12-18 2004-07-15 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
ES2336126T3 (es) * 2004-06-22 2010-04-08 Mallinckrodt, Inc. Sintesis de heteroarilacetamidas a partir de mezclas de reaccion que tienen un contenido reducido de agua.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2492382A1 (fr) * 1980-10-22 1982-04-23 Synthelabo Derives d'imidazo (1,2-a) pyridine, leur preparation et leur application en therapeutique
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593180B1 (fr) * 1986-01-22 1990-10-26 Synthelabo Derives d'acylaminomethyl-1 imidazo (1,2-a)quinoleines, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
PT84159A (pt) 1987-02-01
NO164596C (no) 1990-10-24
DK31887A (da) 1987-07-23
FI85476C (fi) 1992-04-27
FR2593179A1 (fr) 1987-07-24
AU585688B2 (en) 1989-06-22
IE870155L (en) 1987-07-22
ZA87442B (en) 1987-09-30
IE59173B1 (en) 1994-01-26
NO870249D0 (no) 1987-01-21
GR3000463T3 (en) 1991-06-28
AU6789887A (en) 1987-07-23
IL81335A (en) 1990-07-12
FI85476B (fi) 1992-01-15
FI870252A7 (fi) 1987-07-23
NZ219008A (en) 1989-08-29
FI870252A0 (fi) 1987-01-21
JPS62169783A (ja) 1987-07-25
DE3761770D1 (de) 1990-04-05
ES2014306B3 (es) 1990-07-01
EP0233800A1 (de) 1987-08-26
IL81335A0 (en) 1987-08-31
HUT43063A (en) 1987-09-28
PT84159B (pt) 1989-07-31
NO870249L (no) 1987-07-23
EP0233800B1 (de) 1990-02-28
HU194232B (en) 1988-01-28
NO164596B (no) 1990-07-16
DK31887D0 (da) 1987-01-21
CA1286668C (en) 1991-07-23
FR2593179B1 (fr) 1988-04-01

Similar Documents

Publication Publication Date Title
US4473692A (en) Camptothecin derivatives and process for preparing same
US4513138A (en) Camptothecin-1-oxide derivatives
ATE289608T1 (de) Herstellung von camptothecinderivaten durch intramolekulare cyclisierung
KR880000439A (ko) 1,8-다리 걸친 4-퀴놀론-3-카르복실산의 제조방법
AU585688B2 (en) Imidazo``1,2-a`` quinoline derivatives, their preparation and their application in therapy
IE873469L (en) Resolution of 1,4-dihydropyridine derivatives
US4387223A (en) Process for preparing 2(1H)-quinazolinone derivatives
ES8502993A1 (es) Un procedimiento para producir derivados de dihidropirazolo (3,4-b) piridina
FI76337B (fi) Foerfarande foer framstaellning av nya, farmakologiskt aktiva 4,7-dihydropyrazolo/3,4-b/pyridin-5- karboxylsyraderivat.
ATE53034T1 (de) Verfahren zur herstellung von cephemverbindungen.
NO892821D0 (no) Fremgangsmaate for fremstilling av o2, 2'-anhydro-1-(b-d-arabinofuranosyl) tymin.
NO301012B1 (no) Fremgangsmåte for fremstilling av benzo£b|naftyridiner
DK162602C (da) Fremgangsmaade til fremstilling af 7-acylamino-3-(thio-substitueret)methyl-3-cephem-4-carboxylsyre-1-oxid-derivater
KR830010089A (ko) 1,4-티아잔-카르복시산 유도체의 제조방법
NO143534B (no) Analogifremgangsmaate for fremstilling av terapeutisk virksomme derivater av oxatiino(1,4)(2,3-c)pyrrol
DK24088A (da) Fremgangsmaade og mellemprodukter til fremstilling af thiazolobenzimidazoler
IL73998A (en) Preparation of 3-(n-tosyl-l-alaninyloxy)-pyrrole compounds
ATE67194T1 (de) Thiadiazolylacetamid-derivate, verfahren zu ihrer herstellung und ihre verwendung.
DE3760058D1 (en) 3,4-dihydro-2,5,7,8-tetramethyl-2h-1-benzopyran derivatives and processes for their preparation
JPS646265A (en) Production of thiazepine derivative
JPS6425781A (en) 7-deazapurine derivative and production thereof
WO2000034286A3 (en) Process for the preparation of pyrimidinone derivatives

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee