ATE534649T1 - Imidazothiazole und imidazoxazolderivative als inhibitoren von p38 - Google Patents

Imidazothiazole und imidazoxazolderivative als inhibitoren von p38

Info

Publication number: ATE534649T1
Authority: AT; Austria
Prior art keywords: imidazoxazole; imidazothiazoles; inhibitors; derivatives; inhibiting
Prior art date: 2003-05-15

Application number

AT04752390T

Other languages

English (en)

Inventor

Mark Ashwell

Syed Ali

Jifeng Liu

Yanbin Liu

Peter Lohse

Belew Mekonnen

Robert Selliah

Manish Tandon

Woj Wrona

Valery Antonenko

Original Assignee

Arqule Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-05-15

Filing date

2004-05-14

Publication date

2011-12-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=33555294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE534649(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-05-14 Application filed by Arqule Inc filed Critical Arqule Inc

2011-12-15 Application granted granted Critical

2011-12-15 Publication of ATE534649T1 publication Critical patent/ATE534649T1/de

Links

239000003112 inhibitor Substances 0.000 title 1
102000002574 p38 Mitogen-Activated Protein Kinases Human genes 0.000 abstract 3
230000000694 effects Effects 0.000 abstract 2
230000002401 inhibitory effect Effects 0.000 abstract 2
238000000034 method Methods 0.000 abstract 2
102000004127 Cytokines Human genes 0.000 abstract 1
108090000695 Cytokines Proteins 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
238000000338 in vitro Methods 0.000 abstract 1
238000001727 in vivo Methods 0.000 abstract 1

Classifications

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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
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General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
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Oncology (AREA)
Immunology (AREA)
Communicable Diseases (AREA)
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Rheumatology (AREA)
Pulmonology (AREA)
Molecular Biology (AREA)
Orthopedic Medicine & Surgery (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
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Psychology (AREA)
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Urology & Nephrology (AREA)
Cardiology (AREA)
Vascular Medicine (AREA)
Transplantation (AREA)
Biotechnology (AREA)
Hospice & Palliative Care (AREA)
Obesity (AREA)
Hematology (AREA)

AT04752390T 2003-05-15 2004-05-14 Imidazothiazole und imidazoxazolderivative als inhibitoren von p38 ATE534649T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US47073503P	2003-05-15	2003-05-15
US51229803P	2003-10-17	2003-10-17
PCT/US2004/015368 WO2004110990A2 (en)	2003-05-15	2004-05-14	Imidazothiazoles and imidazoxazole derivatives as inhibitors of p38

Publications (1)

Publication Number	Publication Date
ATE534649T1 true ATE534649T1 (de)	2011-12-15

Family

ID=33555294

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT04752390T ATE534649T1 (de)	2003-05-15	2004-05-14	Imidazothiazole und imidazoxazolderivative als inhibitoren von p38

Country Status (9)

Country	Link
US (2)	US7902192B2 (de)
EP (2)	EP2251343A1 (de)
JP (1)	JP4939220B2 (de)
KR (1)	KR20060025141A (de)
AT (1)	ATE534649T1 (de)
AU (1)	AU2004247626B8 (de)
CA (1)	CA2526285A1 (de)
MX (1)	MXPA05012377A (de)
WO (1)	WO2004110990A2 (de)

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KR101948805B1 (ko) *	2016-07-05	2019-02-15	한국과학기술연구원	항종양 효과를 갖는 이미다조옥사졸 유도체 및 이를 포함하는 약학적 조성물
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CN113121564A (zh) *	2019-12-31	2021-07-16	韩国科学技术研究院	具有抗肿瘤效果的咪唑并恶唑衍生物及包括其的药物组合物
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- 2004-05-14 KR KR1020057021750A patent/KR20060025141A/ko not_active Ceased
- 2004-05-14 WO PCT/US2004/015368 patent/WO2004110990A2/en not_active Ceased
- 2004-05-14 MX MXPA05012377A patent/MXPA05012377A/es active IP Right Grant
- 2004-05-14 EP EP10175256A patent/EP2251343A1/de not_active Withdrawn
- 2004-05-14 AU AU2004247626A patent/AU2004247626B8/en not_active Ceased
- 2004-05-14 EP EP04752390A patent/EP1633758B1/de not_active Expired - Lifetime
- 2004-05-14 AT AT04752390T patent/ATE534649T1/de active
- 2004-05-14 US US10/556,161 patent/US7902192B2/en not_active Expired - Fee Related
- 2004-05-14 JP JP2006533130A patent/JP4939220B2/ja not_active Expired - Lifetime
2010
- 2010-12-03 US US12/960,079 patent/US20110301160A1/en not_active Abandoned

Also Published As

Publication number	Publication date
AU2004247626A1 (en)	2004-12-23
US20070270418A1 (en)	2007-11-22
US20110301160A1 (en)	2011-12-08
CA2526285A1 (en)	2004-12-23
AU2004247626B8 (en)	2011-05-19
MXPA05012377A (es)	2006-05-25
JP2006528983A (ja)	2006-12-28
WO2004110990A2 (en)	2004-12-23
EP2251343A1 (de)	2010-11-17
US7902192B2 (en)	2011-03-08
EP1633758B1 (de)	2011-11-23
WO2004110990A3 (en)	2005-03-24
JP4939220B2 (ja)	2012-05-23
EP1633758A2 (de)	2006-03-15
KR20060025141A (ko)	2006-03-20
AU2004247626B2 (en)	2011-01-20

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